GPCR / G Protein

产品 1 到 50 共 860个

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  1. R-121919

    Catalog No. A13535
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    CRF1 receptor 拮抗剂
    R121919是有效的小分子CRF1受体拮抗剂。 了解更多
  2. Verucerfont

    Catalog No. A16950
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    CRF-1 拮抗剂
    Verucerfont,也称为GSK561679和NBI77860,是CRF-1拮抗剂。Verucerfont阻止CRH-1受体,因此减少了慢性应激后ACTH的释放。 了解更多
  3. Emicerfont

    Catalog No. A14047
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    CRF-1 拮抗剂
    Emicerfont,也称为GW876008,是一种CRF-1拮抗剂。Emicerfont阻止CRH-1受体,因此减少了ACTH的释放。 了解更多
  4. Pexacerfont

    Catalog No. A14105
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    CRF1 receptor antagonist
    Pexacerfont is a selective corticotropin-releasing factor (CRF1) receptor antagonist with IC50 of 6.1??0.6 nM for human CRF1 receptor. 了解更多
  5. NVS-CRF38

    Catalog No. A21770
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    CRF1 antagonist
    NVS-CRF38 is a novel corticotropin-releasing factor receptor 1 (CRF1) antagonist with low water solubility. 了解更多
  6. CP 376395

    Catalog No. A21973
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    CRF1 receptor antagonist
    CP 376395 is a potent and selective Corticotropin releasing factor 1 (CRF1) receptor antagonist. 了解更多
  7. CP 316311

    Catalog No. A21983
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    CRF1 receptor antagonist
    CP 316311 is a potent and selective CRF1 receptor antagonist with an IC50 value of 6.8 nM. 了解更多
  8. TGR5-Receptor-Agonist

    Catalog No. A13732
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    TGR5(GPCR19) 激动剂
    TGR5 Receptor Agonist是一种有效的TGR5(GPCR19)激动剂,在U2-OS细胞分析(pEC50 = 6.8)和黑素细胞(pEC50 = 7.5)中显示出增强的效力。 了解更多
    • 最新产品

    SBI-115

    Catalog No. A17235
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    GPCR19 antagonist
    SBI-115 is a TGR5 (GPCR19) antagonist. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5. 了解更多
  9. SB756050

    Catalog No. A12759
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    TGR5 agonist
    SB756050 is a selective TGR5 agonist currently in phase 1clinical trials for the treatment of type 2 diabetes. 了解更多
  10. INT-777

    Catalog No. A21168
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    TGR5 agonist
    INT-777 is a potent TGR5 agonist with an EC50 of 0.82 μM. 了解更多
  11. INT-767

    Catalog No. A21494
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    dual FXR/TGR5 agonist
    INT-767 is a dual farnesoid X receptor (FXR)/TGR5 agonist with mean EC50s of 30 and 630 nM, respectively. 了解更多
  12. NPS-2143 (SB-262470)

    Catalog No. A11140
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    CaSR 拮抗剂
    NPS-2143 (SB-262470)是一种选择性的Ca2+感应受体拮抗剂,显示可阻止HEK293细胞中表达的人Ca2+受体引起的细胞质Ca2+浓度增加,IC50为43 nM。 了解更多
  13. AMG-073 HCl (Cinacalcet HCl)

    Catalog No. A10219
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    CaSR activator
    AMG-073 HCl(Cinacalcet HCl)是一种用于治疗甲状旁腺功能亢进的化合物,称为拟钙剂,通过增加甲状旁腺钙敏感受体(CaR)对细胞外钙的敏感性来减少甲状旁腺激素(PTH)的合成和分泌 。 了解更多
  14. Strontium ranelate (Protelos)

    Catalog No. A11681
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    CaSR 激动剂
    Strontium ranelate是一种抗骨质疏松剂,可增加骨形成并减少骨吸收,从而导致骨转换平衡,有利于骨形成。这类似于胆碱稳定的原硅酸的作用。 了解更多
  15. AMG 073 (Cinacalcet)

    Catalog No. A11314
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    CaSR activator
    AMG 073 (Cinacalcet)是一类治疗甲状旁腺功能亢进的新型化合物。 了解更多
  16. Evocalcet

    Catalog No. A17003
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    CaSR 激动剂
    Evocalcet是一种钙敏感受体激动剂。钙敏感受体(CaSR)是C类G蛋白偶联受体,可感应细胞外钙离子水平。 了解更多
  17. NPS-2143 hydrochloride

    Catalog No. A11505
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    CaSR antagonist
    NPS-2143 hydrochloride (SB-262470A hydrochloride), an orally active calcilytic agent, is a selective and potent calcium ion-sensing receptor (CaSR) antagonist. 了解更多
  18. Lixisenatide

    Catalog No. A14076
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    GLP-1 receptor 激动剂
    Lixisenatide抑制胰高血糖素释放,显着降低餐后胰高血糖素。对糖尿病(T2DM)有促进作用。 了解更多
  19. BETP

    Catalog No. A13781
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    GLP-1 receptor 激动剂
    BETP是胰高血糖素样肽1(GLP-1)受体的选择性正构构调节剂和部分激动剂。 了解更多
  20. Liraglutide

    Catalog No. A16115
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    GLP-1 receptor 激动剂
    Liraglutide是一种长效胰高血糖素样肽1(GLP-1)受体激动剂。 了解更多
  21. Albiglutide

    Catalog No. A16823
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    GLP-1 激动剂
    Albiglutide是一种胰高血糖素样肽1激动剂(GLP-1激动剂)。 了解更多
  22. Dulaglutide

    Catalog No. A16987
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    GLP-1 receptor 激动剂
    Dulaglutide是胰高血糖素样肽1(GLP-1)受体激动剂。 了解更多
  23. VU0453379

    Catalog No. A18796
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    GLP-1R modulator
    VU0453379 is a CNS-penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric modulator (PAM) with an EC50 of 1.3 μM. 了解更多
  24. Semaglutide

    Catalog No. A18908
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    GLP-1 receptor agonist
    Semaglutide, a long-acting GLP-1 analogue, is a glucagon-like peptide-1 (GLP-1) receptor agonist that can be used in the treatment of type 2 diabetes. 了解更多
  25. NNC0640

    Catalog No. A18900
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    GLP-1R modulator
    NNC0640 is a negative allosteric modulator of glucagon-like peptide-1 receptor (GLP-1R). 了解更多
  26. Loxiglumide (CR1505)

    Catalog No. A11769
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    CCK-A receptor 拮抗剂
    Loxiglumide (CR1505)是一种胆囊收缩素拮抗剂。 了解更多
  27. Proglumide sodium salt

    Catalog No. A13713
    CCK 拮抗剂
    Proglumide sodium salt是一种非选择性胆囊收缩素(CCK)拮抗剂。它抑制CCK刺激的淀粉酶分泌,并防止CCK诱导的小鼠胰腺腺泡中的2-脱氧葡萄糖摄取。 了解更多
  28. Z-360 calcium salt (Nastorazepide calcium salt)

    Catalog No. A13671
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    CCK-2 receptor 拮抗剂
    Z-360 calcium salt (Nastorazepide calcium salt)是一种选择性口服可口服的1,5-苯并二氮杂卓衍生物胃泌素/胆囊收缩素2(CCK-2)受体拮抗剂,具有潜在的抗肿瘤活性。 了解更多
  29. Nastorazepide (Z-360)

    Catalog No. A15984
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    CCK-2 receptor 拮抗剂
    Nastorazepide (Z-360) 是一种选择性的,口服的1,5-苯二氮杂卓衍生物胃泌素/胆囊收缩素2(CCK-2)受体拮抗剂,具有潜在的抗肿瘤活性。 了解更多
  30. Proglumide

    Catalog No. A18171
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    CCK antagonist
    Proglumide is a drug that exerts an inhibitory effect on gastric secretion and reduces gastrointestinal motility. IProglumide is a known cholecystokinin (CCK) antagonist. 了解更多
  31. Dexloxiglumide

    Catalog No. A18541
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    CCKA receptor antagonist
    Dexloxiglumide is a selective cholecystokinin type A (CCKA) receptor antagonist. Dexloxiglumide, the active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). 了解更多
  32. Moxonidine HCl

    Catalog No. A11741
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    imidazoline receptor 1 激动剂
    Moxonidine HCl是咪唑啉受体亚型1(I1)的选择性激动剂。Moxonidine引起交感神经系统活动的减少,因此导致血压的降低。 了解更多
  33. Rilmenidine Phosphate

    Catalog No. A14256
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    I(1) imidazoline receptor 激动剂
    Rilmenidine Phosphate是一种选择性的I(1)咪唑啉受体激动剂。 了解更多
  34. KU14R

    Catalog No. A13987
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    I3 receptor 拮抗剂
    KU14R是胰腺β细胞非典型咪唑啉结合位点(可能的I3受体)的拮抗剂。KU14R也已显示出选择性阻断依法氧烷诱导的胰岛素分泌。 了解更多
  35. Moxonidine Hydrochloride

    Catalog No. A13416
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    imidazoline receptor 1 激动剂
    Moxonidine Hydrochloride (BDF5895)是咪唑啉1型受体(I1-R)选择性激动剂,为降压剂。 了解更多
  36. Bombesin

    Catalog No. A13488
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    Bombesin是一种神经肽,具有许多生物学作用,包括激素释放,刺激胰酶分泌,抑制胃排空和调节胃酸分泌。 了解更多
  37. Anamorelin HCl

    Catalog No. A12345
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    Anamorelin HCl目前正在开发中,是口服活性的饥饿素受体(ghrelin receptor)激动剂。用于治疗与恶病质/厌食症相关的非小肺癌。 了解更多
  38. Anamorelin

    Catalog No. A12346
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    Anamorelin是一种新型 ghrelin receptor激动剂,FLIPR 检测中,EC50 为 0.74 nM,用于治疗与恶病质/厌食症相关的非小肺癌。 了解更多
  39. Capromorelin

    Catalog No. A14350
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    Capromorelin用作生长激素促分泌素和生长素释放肽模拟物,使人体以青春期和成年期常见的方式分泌人体生长激素。 了解更多
  40. Anamorelin Fumarate

    Catalog No. A15000
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    GHSR stimulator
    Anamorelin Fumarate是一种合成的口服活性ghrelin受体激动剂,正在开发中,用于治疗与小肺癌相关的恶病质/厌食症。 了解更多
  41. Capromorelin Tartrate

    Catalog No. A21238
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    GHSR agonist
    Capromorelin Tartrate is an orally active, potent growth hormone secretagogue receptor (GHSR) agonist, with Ki of 7 nM for hGHS-R1a. 了解更多
  42. MK 0893

    Catalog No. A11495
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    GCGR 抑制剂
    MK 0893是胰高血糖素受体拮抗剂作为抗糖尿病药物,IC50 值为 6.6 nM。 了解更多
  43. ESI-09

    Catalog No. A14233
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    EPAC1/EPAC2 抑制剂
    ESI-09是一种直接由cAMP(EPAC)抑制剂激活的特异性交换蛋白,对于EPAC1和EPAC2,IC50为3.2 uM和1.4 uM。 了解更多
  44. HJC0350

    Catalog No. A14266
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    EPAC2 抑制剂
    HJC0350是一种有效的选择性EPAC2抑制剂,IC50为0.3μM,对Epac1无抑制作用。 了解更多
  45. cAMPS-Sp, triethylammonium salt

    Catalog No. A16060
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    cAMPS-Sp, triethylammonium salt是一种可透过细胞的cAMP类似物,可激活cAMP受体蛋白,例如PKA和cAMP调节的鸟嘌呤核苷酸交换因子。 了解更多
  46. SQ22536

    Catalog No. A16116
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    adenylyl cyclase 抑制剂
    SQ22536是腺苷酸环化酶的抑制剂,IC50为1.4 uM。它可以抑制完整人血小板中PGE1刺激的cAMP水平升高。 了解更多
  47. Bithionol

    Catalog No. A14941
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    Bithionol是一种有效的可溶性腺苷酸环化酶抑制剂,具有抗菌和驱虫特性以及除藻活性。 了解更多
  48. ESI-05

    Catalog No. A18644
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    EPAC2 antagonist
    ESI-05 (NSC 116966) is a specific antagonist of EPAC2 (exchange protein directly activated by cAMP 2), with an IC50 of 0.4 ?M. ESI-05 (NSC 116966) inhibits cAMP-mediated activation of EPAC2 as well as EAPC2 mediated Rap1 activation. 了解更多
  49. Riociguat (BAY 63-2521)

    Catalog No. A11549
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    sGC stimulator
    Riociguat (BAY 63-2521)是可溶性鸟苷酸环化酶(sGC)的刺激物。 了解更多

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