ADL5859 HCl

Name: ADL5859 HCl
SKU: A11072

目录号: A11072

Opioid Receptor 激动剂

ADL5859 HCl Chemical Structure

CAS NO. 850173-95-4

ADL5859 HCl是高效的选择性δ阿片受体激动剂，Ki值为0.84 nM，ED50值为20 nM。

库存：现货

规格	价格	数量
5 mg	￥ 1,200.00
10 mg	￥ 2,000.00
50 mg	￥ 5,800.00
100 mg	￥ 8,800.00
10mM * 1mL in DMSO	￥ 1,400.00

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生物活性

ADL5859 HCl是高效的选择性δ阿片受体激动剂，Ki值为0.84 nM，ED50值为20 nM。

靶点信息

δ-opioid receptor	μ-opioid receptor	κ-opioid receptor
0.8 nM(Ki)	32 nM(Ki)	37 nM(Ki)

溶解度 *

In vitro (25°C)	DMSO	76 mg/mL (177.17 mM)
	Water	4 mg/mL (9.32 mM)
	Ethanol	1 mg/mL (2.33 mM)
In vivo	0.5% hydroxyethyl cellulose+0.1% Tween 80	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	23.31 mL	116.55 mL	233.1 mL
0.5 mM	4.66 mL	23.31 mL	46.62 mL
1 mM	2.33 mL	11.66 mL	23.31 mL
5 mM	0.47 mL	2.33 mL	4.66 mL

*The above data is based on the productmolecular weight 429. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11072
作用机制	Agonist (激动剂)
M. Wt	429
Formula	C24H28N2O3.HCl
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	850173-95-4
Synonyms	ADL-5859
SMILES	CCN(CC)C(=O)C1=CC=C(C=C1)C2=CC3(CCNCC3)OC4=C2C(=CC=C4)O.Cl