Alcaftadine

Name: Alcaftadine
SKU: A16393

目录号: A16393

H1 histamine receptor 拮抗剂

Alcaftadine Chemical Structure

CAS NO. 147084-10-4

Alcaftadine是H1受体的高亲和力配体，其pKi（8.5）与其他H1抗组胺药相当。Alcaftadine还是H2和H4受体的拮抗剂，对H3受体没有亲和力。

库存：现货

规格	价格	数量
10 mg	￥ 400.00
25 mg	￥ 800.00
100 mg	￥ 2,200.00

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生物活性

Alcaftadine是H1受体的高亲和力配体，其pKi（8.5）与其他H1抗组胺药相当。Alcaftadine还是H2和H4受体的拮抗剂，对H3受体没有亲和力。

溶解度 *

In vitro	DMSO	26 mg/mL (84.57 mM)
	Water	Insoluble
	Ethanol	57 mg/mL (185.43 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	32.53 mL	162.66 mL	325.32 mL
0.5 mM	6.51 mL	32.53 mL	65.06 mL
1 mM	3.25 mL	16.27 mL	32.53 mL
5 mM	0.65 mL	3.25 mL	6.51 mL

*The above data is based on the productmolecular weight 307.39. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A16393
作用机制	Antagonist (拮抗剂)
M. Wt	307.39
Formula	C19H21N3O
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	147084-10-4
Synonyms	R89674, R 89674, R-89674
SMILES	CN1CC/C(CC1)=C2C3=CC=CC=C3CCN4C(C=O)=CN=C/24