“angiotensin receptors”的搜索结果

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  1. Angiotensin III

    Catalog No. A18943
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    angiotensin 1 (AT1) and AT2 receptor agonist
    Angiotensin III is an angiotensin 1 (AT1) and AT2 receptor agonist. 了解更多
  2. Angiotensin II human Acetate

    Catalog No. A17993
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    Angiotensin II human is a vasoconstrictor that acts on the AT1 and the AT2 receptor. 了解更多
  3. Angiotensin

    Catalog No. AP4258
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  4. Angiotensin 1/2 + A (2 - 8)

    Catalog No. A14888
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    Angiotensin 1/2 + A (2 - 8)有效的内源性血管收缩肽;血管紧张素(Ang)的衍生物II。 了解更多
  5. Angiotensin 1/2 (1-6)

    Catalog No. A14887
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    Angiotensin 1/2 (1-6)是一种包含氨基酸1-6的肽,是从血管紧张素I/II肽转化而来的。 了解更多
  6. Angiotensin 1/2 (1-5)

    Catalog No. A14886
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    Angiotensin 1/2 (1-5)是一种包含氨基酸1-5的肽,是从血管紧张素I/II转化而来的。 了解更多
  7. Angiotensin 1/2 (1-9)

    Catalog No. A14873
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    Angiotensin 1/2 (1-9)是一种肽(ASP-ARG-VAL-TYR-ILE-HIS-PRO-PHE-HIS),包含从血管紧张素I/II肽转换而来的氨基酸1-9。 了解更多
  8. Angiotensin III (human, mouse)

    Catalog No. A14864
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    Angiotensin III (human,mouse)是在血管紧张素II的N末端裂解形成的六肽,血管紧张素II是位于红细胞和大多数组织血管床中的血管紧张素酶在肾素-血管紧张素-醛固酮(RAAS)系统中的关键因素。 了解更多
  9. Angiotensin II

    Catalog No. A14863
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    Angiotensin II是一种八肽激素,在心血管稳态中起着核心作用。 了解更多
  10. Angiotensin (1-7)

    Catalog No. A14862
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    Angiotensin (1-7)是一种内源性肽片段,可以分别通过内切肽酶或羧肽酶从Ang I或Ang II产生。 了解更多
  11. Fimasartan

    Catalog No. A17477
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    non-peptide angiotensin II receptor antagonist
    Fimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of angiotensin II, such as systemic vasoconstriction and water retention by the kidneys. 了解更多
  12. Losartan

    Catalog No. A17510
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    Angiotensin II receptor antagonist
    Losartan is an angiotensin II receptor antagonist, competing with the binding of angiotensin II to AT1 receptors with IC50 of 20 nM. 了解更多
  13. Angiotensin I (human, mouse, rat)

    Catalog No. A14859
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    Angiotensin I (human,mouse,rat)是由肾素对血管紧张素原的作用形成的。 了解更多
  14. EMD-66684

    Catalog No. A22609
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    angiotensin II receptor antagonist
    EMD-66684 is a non-peptide angiotensin II receptor antagonist. 了解更多
  15. L-159282

    Catalog No. A20703
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    nonpeptide angiotensin II receptor antagonist
    L-159282 is a highly potent, orally active, nonpeptide angiotensin II receptor antagonist, with anti-hypertensive activity. 了解更多
  16. L162389

    Catalog No. A20297
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    angiotensin AT1 receptor antagonist
    L162389 is a potent antagonist of angiotensin AT1 receptor with Ki of 28 nM. 了解更多
  17. CGP48369

    Catalog No. A19745
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    angiotensin II receptor antagonist
    CGP48369 is a nonpeptidic angiotensin II receptor antagonist, used for anti-hypertensive research. 了解更多
  18. Pratosartan

    Catalog No. A19381
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    angiotensin II receptor antagonist
    Pratosartan is a selective angiotensin II receptor antagonist. 了解更多
  19. AVE 0991

    Catalog No. A20997
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    angiotensin-(1-7) receptor agonist
    AVE 0991 is a nonpeptide and orally active angiotensin-(1-7) receptor agonist with an IC50 of 21 nM. 了解更多
  20. Azilsartan D5

    Catalog No. A21600
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    angiotensin II type 1 receptor antagonist
    Azilsartan D5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. 了解更多
  21. Losartan (D4 Carboxylic Acid)

    Catalog No. A21578
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    angiotensin II receptor antagonist
    Losartan D4 Carboxylic Acid is the deuterium labeled Losartan(EXP-3174), which is an angiotensin II receptor antagonist. 了解更多
  22. CGP-42112

    Catalog No. A21575
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    Angiotensin-II subtype 2 receptor(AT2 R) agonist
    CGP-42112(CGP-42112A) is a potent Angiotensin-II subtype 2 receptor(AT2 R) agonist. 了解更多
  23. Lisinopril

    Catalog No. A21064
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    angiotensin-converting enzyme inhibitor
    Lisinopril (MK-521) is angiotensin-converting enzyme inhibitor, used in treatment of hypertension, congestive heart failure, and heart attacks. 了解更多
  24. Sparsentan

    Catalog No. A20879
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    angiotensin II and endothelin A receptor antagonist
    Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. 了解更多
  25. Azilsartan medoxomil monopotassium

    Catalog No. A20860
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    angiotensin II receptor type 1 antagonist
    Azilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. 了解更多
  26. Valsartan

    Catalog No. A10962
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    angiotensin II receptor antagonist
    Valsartan (CGP-48933) is an angiotensin II receptor antagonist for the treatment of high blood pressure and heart failure. 了解更多
  27. SL910102

    Catalog No. A13591
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    Angiotensin AT1 receptor antagonist
    SL910102 is a nonpeptide angiotensin AT1 receptor antagonist. 了解更多
  28. SYM 2081

    Catalog No. A20332
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    kainate receptors agonist
    SYM 2081 is a high-affinity ligand and potent, selective agonist of kainate receptors, inhibits [3H]-kainate binding with an IC50 of 35 nM, almost 3000- and 200-fold selectivity for kainate receptors over AMPA and NMDA receptors respectively. 了解更多
  29. Alniditan

    Catalog No. A19801
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    5-HT1B/1D receptors agonist
    Alniditan is a potent 5-HT1B/1D receptors agonist, with IC50 of 1.7 and 1.3 nM in HEK?293 cells, and pKi value of 8.96 and 9.40 for 5-HT1B/1D receptors, respectively. 了解更多
  30. PSN632408

    Catalog No. A20902
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    GPR119 receptors agonist
    PSN632408 is an optimized agonist of GPR119 receptors that shows similar potency to OEA at both recombinant mouse and human GPR119 receptors, exhibiting EC50 values of 5.6 and 7.9 uM, respectively. 了解更多
  31. Deramciclane

    Catalog No. A13011
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    5-HT2A and 5-HT2C receptors antagonist
    Deramciclane has a high affinity for 5-HT2A and 5-HT2C receptors; it acts as an antagonist at both receptor subtypes and has inverse agonist properties at the 5-HT2C receptors without direct stimulatory agonist. 了解更多
  32. DPI-3290

    Catalog No. A13699
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    opioid receptors agonist
    DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively. 了解更多
  33. MHP 133

    Catalog No. A20058
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    AChE /M1/M2/5HT4/I2 inhibitor
    MHP 133 is a drug with multiple CNS targets, and inhibits acetylcholinesterase (AChE) with Ki of 69 μM; also active against muscarinic M1 and M2 receptors, serotonin 5HT4 receptors, and imidazole I2 receptors. 了解更多
  34. Dihydroergotamine Mesylate

    Catalog No. A17764
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    Serotonin receptors agonist
    Dihydroergotamine Mesylate, also known as DHE or Migranal, is an ergot alkaloid used to treat migraines. It has similar actions to the triptans, acting as an agonist to the serotonin receptors and causing vasoconstriction of the intracranial blood vessels, but also interacts centrally with dopamine and adrenergic receptors. 了解更多
  35. Elisartan

    Catalog No. A20697
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    Elisartan is an orally active non-peptide pro-drug of angiotensin II AT1 receptor antagonist HN-12206, and shows anti-hypertension activities. 了解更多
  36. Rentiapril

    Catalog No. A20233
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    ACE inhibitor
    Rentiapril is an orally active angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity. 了解更多
  37. ZD 7155 hydrochloride

    Catalog No. A19959
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    AT1 receptor antagonist
    ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist. 了解更多
  38. Utibapril

    Catalog No. A19907
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    ACE inhibitor
    Utibapril is an angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activities. 了解更多
  39. NCX899

    Catalog No. A19352
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    ACE inhibitor
    NCX899 is a NO-releasing derivative of enalapril, and shows inhibitory activity against angiotensin-converting enzyme (ACE) activity. 了解更多
  40. H-Ile-Pro-Pro-OH

    Catalog No. A19177
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    H-Ile-Pro-Pro-OH, a milk-derived peptide, inhibits angiotensin-converting enzyme (ACE)with an IC50 of 5 μM. Antihypertensive tripeptides. 了解更多
  41. Olodanrigan

    Catalog No. A21691
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    AT2R antagonist
    Olodanrigan (EMA401) is a highly selective, orally active, peripherally restricted angiotensin II type 2 receptor (AT2R) antagonist. 了解更多
  42. Dihexa

    Catalog No. A20933
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    Dihexa, an oligopeptide drug, is an orally active and blood-brain barrier-permeable angiotensin IV analog. 了解更多
  43. Imidaprilate

    Catalog No. A20003
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    ACE inhibitor
    Imidaprilate is an active metabolite of TA-6366, acts as a potent angiotensin converting enzyme (ACE) inhibitor, with an IC50 of 2.6 nM, and is used in the research of hypertensive disease. 了解更多
  44. Zofenopril

    Catalog No. A13615
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    ACE inhibitor
    Zofenopril is an angiotensin-converting enzyme (ACE) inhibitor with an IC50 of 81 μM. 了解更多
  45. TD-0212

    Catalog No. A13715
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    neprilysin (NEP) inhibitor
    TD-0212 (compound 35) is an orally active dual pharmacology angiotensin II type 1 receptor (AT1) antagonist and neprilysin (NEP) inhibitor, with a pKi of 8.9 for AT1 and a pIC50 of 9.2 for NEP. 了解更多
  46. H-Val-Pro-Pro-OH

    Catalog No. A18868
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    ACE inhibitor
    H-Val-Pro-Pro-OH, a milk-derived proline peptides derivative, is an inhibitor of Angiotensin I converting enzyme (ACE), with an IC50 of 9 μM. 了解更多
  47. Apelin agonist 1

    Catalog No. A19035
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    apelin agonist
    Apelin agonist 1 is an oral selective apelin agonist AM-2995, a agonist of the APJ (APLNR, angiotensin receptor like-1) receptor, may be used in the treatment of cardiovascular conditions. 了解更多
  48. Azilsartan Medoxomil

    Catalog No. A16420
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    angiotensin II receptor type 1 拮抗剂
    Azilsartan medoxomil是一种口服给药的1型血管紧张素II受体拮抗剂,IC50为0.62 nM。 了解更多
  49. BIBS39

    Catalog No. A14154
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    angiotensin II receptor 拮抗剂
    BIBS39是一种非肽血管紧张素II(AII)受体拮抗剂,可从其特异性结合位点置换[125I] AII,其AII亚型(AT1)受体和K(i)的K(i)值为29+/-7 nM。)AII亚型2(AT2)受体的480+/-110 nM)值。 了解更多
  50. LCZ696 (Valsartan)

    Catalog No. A14206
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    angiotensin receptor-neprilysin 抑制剂
    LCZ696 (Valsartan)是一种生物利用型双效血管紧张素受体-中性溶血素抑制剂(ARNi),用于治疗高血压和心力衰竭。 了解更多

产品 1 到 50 共 209个

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