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Bcl-2 Inhibitor包含两种互变异构体的混合物。一种有效的,细胞可渗透的Bcl-2抑制剂与Bak BH3肽竞争体外结合Bcl-2和Bcl-XL的作用(分别为IC50 = 10 uM和7 uM)。
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 33.3 mL | 166.5 mL | 333 mL |
0.5 mM | 6.66 mL | 33.3 mL | 66.6 mL |
1 mM | 3.33 mL | 16.65 mL | 33.3 mL |
5 mM | 0.67 mL | 3.33 mL | 6.66 mL |
*The above data is based on the productmolecular weight 300.3. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
目录号 | A13580 |
---|---|
作用机制 | Inhibitor (抑制剂) |
M. Wt | 300.3 |
Formula | C16H16N2O4 |
Purity | >99% |
Storage | Store lyophilized at -20ºC, keep desiccated. |
CAS No. | 383860-03-5 |
Synonyms | TW-37 |
SMILES | COC1=CC(=C(C=C1)N=O)CCC2=C(C=CC(=C2)OC)N=O |
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