“MK-2206 dihydrochloride”的搜索结果

产品 1 到 50 共 117个

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  1. MK-2206 2HCl

    Catalog No. A10003
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    AKT 抑制剂
    MK-2206 2HCl是Akt1/2/3的高选择性抑制剂,IC50分别为8 nM/12 nM/65 nM。 了解更多
  2. SYM2206

    Catalog No. A20843
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    AMPA receptor antagonist
    SYM 2206 is a novel, potent, non-competitive AMPA receptor antagonist. 了解更多
  3. Quisinostat dihydrochloride

    Catalog No. A22453
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    pan-HDAC inhibitor
    Quisinostat dihydrochloride (JNJ-26481585 dihydrochloride) is an orally available, potent pan-HDAC inhibitor with IC50s of 0.11 nM, 0.33 nM, 0.64 nM, 0.46 nM, and 0.37 nM for HDAC1, HDAC2, HDAC4, HDAC10 and HDAC11, respectively. Quisinostat dihydrochloride has a broad spectrum antitumoral activity. 了解更多
  4. PAβN dihydrochloride

    Catalog No. A22016
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    efflux pump inhibitor
    PAβN dihydrochloride (MC-207110 dihydrochloride) is an efflux pump inhibitor. 了解更多
  5. Banoxantrone D12 dihydrochloride

    Catalog No. A21438
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    Banoxantrone D12 dihydrochloride (AQ4N D12 dihydrochloride) is the deuterium labeled banoxantrone dihydrochloride. Banoxantrone is a novel bioreductive agent that can be reduced to a stable, DNA-affinic compound AQ4, which is a potent topoisomerase II inhibitor. 了解更多
  6. Ipatasertib dihydrochloride

    Catalog No. A21734
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    pan-Akt inhibitor
    Ipatasertib dihydrochloride (GDC-0068 dihydrochloride) is a highly selective pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 5/18/8 nM, 620-fold selectivity over PKA. 了解更多
  7. GDC-0575 dihydrochloride

    Catalog No. A21567
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    CHK1 inhibitor
    GDC-0575 dihydrochloride (ARRY-575 dihydrochloride) is an orally bioavailable CHK1 inhibitor, with an IC50 of 1.2 nM, and has antitumor activity. 了解更多
  8. GSK3368715 dihydrochloride

    Catalog No. A21733
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    PRMT inhibitor
    GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50=3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)). 了解更多
  9. LCL521 dihydrochloride

    Catalog No. A21656
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    ACDase inhibitor
    LCL521 dihydrochloride (1,3DMG-B13 dihydrochloride) is an acid ceramidase (ACDase) inhibitor. 了解更多
  10. Lerociclib dihydrochloride

    Catalog No. A21577
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    CDK4/CDK6 inhibitor
    Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 1 nM and 2 nM for CDK4/CyclinD1 and CDK6/CyclinD3, respectively. 了解更多
  11. NVP-BSK805 dihydrochloride

    Catalog No. A21406
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    JAK2 inhibitor
    NVP-BSK805 dihydrochloride (BSK805 dihydrochloride) is an ATP-competitive JAK2 inhibitor, with IC50s of 0.48 nM, 31.63 nM, 18.68 nM, and 10.76 nM for JAK2 JH1 (JAK homology 1), JAK1 JH1, JAK3 JH1, and TYK2 JH1, respectively. 了解更多
  12. Mirodenafil dihydrochloride

    Catalog No. A18047
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    PDE-5 inhibitor
    Mirodenafil dihydrochloride (SK3530 dihydrochloride) is a phosphodiesterase type 5 (PDE-5) inhibitor developed for the treatment of erectile dysfunction. 了解更多
  13. Canertinib dihydrochloride

    Catalog No. A11344
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    EGFR inhibitor
    Canertinib dihydrochloride (CI-1033 dihydrochloride) is a potent and irreversible EGFR inhibitor; inhibits cellular EGFR and ErbB2 autophosphorylation with IC50s of 7.4 and 9 nM. 了解更多
  14. Azaphen dihydrochloride monohydrate

    Catalog No. A15009
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    serotonin reuptake 抑制剂
    Azaphen dihydrochloride monohydrate是5-羟色胺再摄取的有效抑制剂。 了解更多
  15. DAPI dihydrochloride

    Catalog No. A22602
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    fluorescent probe
    DAPI Dihydrochloride is a cell-permeable fluorescent probe used to stain DNA and chromosomes, with a preference for adenine and thymine rich DNA. 了解更多
  16. Banoxantrone dihydrochloride

    Catalog No. A21432
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    Banoxantrone dihydrochloride is a novel bioreductive agent that can be reduced to a stable, DNA-affinic compound AQ4, which is a potent topoisomerase II inhibitor. 了解更多
  17. MW-150 dihydrochloride dihydrate

    Catalog No. A21860
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    p38α MAPK inhibitor
    MW-150 dihydrochloride dihydrate (MW01-18-150SRM dihydrochloride dihydrate) is a selective, CNS penetrant, and orally active inhibitor of p38α MAPK with a Ki of 101 nM. 了解更多
  18. Liarozole dihydrochloride

    Catalog No. A21853
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    CYP450 dependent inhibitor
    Liarozole dihydrochloride (R75251; R85246) is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase). 了解更多
  19. Philanthotoxin 74 dihydrochloride

    Catalog No. A21739
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    AMPAR antagonist
    Philanthotoxin 74 dihydrochloride (PhTx 74) is an AMPAR antagonist; inhibits GluR3 and GluR1 with IC50s of 263 and 296 nM, respectively. 了解更多
  20. SB-277011 dihydrochloride

    Catalog No. A21353
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    dopamine D3 receptor antagonist
    SB-277011 dihydrochloride (SB-277011A dihydrochloride) is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor antagonist, with pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively. 了解更多
  21. Retigabine dihydrochloride

    Catalog No. A15222
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    KCNQ channel opener
    Retigabine dihydrochloride是具有抗惊厥活性的Kv7.2-7.5(KCNQ2-5)神经元钾通道开放剂。 了解更多
  22. LDK378 (Ceritinib) dihydrochloride

    Catalog No. A15142
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    ALK 抑制剂
    LDK378 (Ceritinib) dihydrochloride是有效的抗ALK抑制剂,IC50为0.2 nM,对IGF-1R和InsR的选择性分别为40倍和35倍。 了解更多
  23. LMPTP INHIBITOR 1 dihydrochloride

    Catalog No. A22227
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    LMPTP inhibitor
    LMPTP INHIBITOR 1 (dihydrochloride) is a selective inhibitor of low molecular weight protein tyrosine phosphatase (LMPTP), with an IC50 of 0.8 μM LMPTP-A. 了解更多
  24. LYN-1604 dihydrochloride

    Catalog No. A22230
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    ULK1 activator
    LYN-1604 dihydrochloride is a potent UNC-51-like kinase 1 (ULK1) activator (EC50=18.94 nM) for the research of triple negative breast cancer (TNBC). 了解更多
  25. Iso-H7 dihydrochloride

    Catalog No. A22368
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    inhibitor of phosphokinase C
    Iso-H7 dihydrochloride is an inhibitor of phosphokinase C. 了解更多
  26. IT1t dihydrochloride

    Catalog No. A22027
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    CXCR4 antagonist
    IT1t dihydrochloride is a potent CXCR4 antagonist; inhibits CXCL12/CXCR4 interaction with an IC50 of 2.1 nM. 了解更多
  27. SB-772077B dihydrochloride

    Catalog No. A20090
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    ROCK inhibitor
    SB-772077B dihydrochloride is an aminofurazan-based Rho kinase (ROCK) inhibitor with IC50s of 5.6 nM and 6 nM toward ROCK1 and ROCK2, respevtively. 了解更多
  28. ABT-702 dihydrochloride

    Catalog No. A19624
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    AK inhibitor
    ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor (IC50=1.7 nM). 了解更多
  29. N-Desethyl amodiaquine dihydrochloride

    Catalog No. A21695
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    N-Desethyl amodiaquine dihydrochloride is the major biologically active metabolite of Amodiaquine. N-Desethyl amodiaquine dihydrochloride is an antiparasitic agent. 了解更多
  30. d-Atabrine dihydrochloride

    Catalog No. A21654
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    d-Atabrine dihydrochloride is an active enantiomer of quinacrine which displays antiprion activity. 了解更多
  31. Veliparib dihydrochloride

    Catalog No. A21356
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    PARP inhibitor
    Veliparib dihydrochloride is a potent PARP inhibitor, inhibiting PARP1 and PARP2 with Kis of 5.2 and 2.9 nM, respectively. 了解更多
  32. Ro 10-5824 dihydrochloride

    Catalog No. A21986
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    dopamine D4 receptor partial agonist
    Ro 10-5824 dihydrochloride is a selective dopamine D4 receptor partial agonist, with Ki of 5.2 nM. 了解更多
  33. GSK-LSD1 dihydrochloride

    Catalog No. A21815
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    LSD1 inhibitor
    GSK-LSD1 dihydrochloride is a potent, selective and irreversible lysine specific demethylase 1 (LSD1) inhibitor with an IC50 of 16 nM. 了解更多
  34. K-604 dihydrochloride

    Catalog No. A21773
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    ACAT-1 inhibitor
    K-604 dihydrochloride is a potent and selective acyl-CoA:cholesterol acyltransferase 1 (ACAT-1) inhibitor with an IC50 of 0.45??0.06 μM. 了解更多
  35. N8-Acetylspermidine dihydrochloride

    Catalog No. A21720
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    N8-Acetylspermidine dihydrochloride is a polyamine. 了解更多
  36. TLR7/8 agonist 1 dihydrochloride

    Catalog No. A21700
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    TLR7/8 agonist
    TLR7/8 agonist 1 dihydrochloride is a toll-like receptor (TLR7)/TLR8 dual-agonistic imidazoquinoline. 了解更多
  37. MRT68921 dihydrochloride

    Catalog No. A21650
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    ULK1/ULK2 inhibitor
    MRT68921 dihydrochloride is the most potent inhibitor of ULK1 and ULK2, with IC50 values of 2.9 nM and 1.1 nM, respectively. 了解更多
  38. l-Atabrine dihydrochloride

    Catalog No. A21646
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    l-Atabrine dihydrochloride is a less active enantiomer of quinacrine which displays antiprion activity. 了解更多
  39. JNJ-37822681 dihydrochloride

    Catalog No. A21470
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    dopamine D2 receptor antagonist
    JNJ-37822681 dihydrochloride is a potent, specific, centrally active, fast-dissociating dopamine D2 receptor antagonist with a moderate binding affinity for the dopamine D2L receptor (Ki =158 nM), which has potential for the treatment of schizophrenia and bipolar disorder. 了解更多
  40. PF429242 dihydrochloride

    Catalog No. A21386
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    S1P inhibitor
    PF429242 dihydrochloride is a reversible and competitive S1P inhibitor with an IC50 of 175 nM. 了解更多
  41. JDTic dihydrochloride

    Catalog No. A11469
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    KOR antagonist
    JDTic (dihydrochloride) is a potent antagonist of kappa-opioid receptors (KOR), blocking the κ-agonist U50, 488-induced antinociception. 了解更多
  42. Lesopitron dihydrochloride

    Catalog No. A12950
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    5-HT1A receptor agonist
    Lesopitron dihydrochloride is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes. 了解更多
  43. AQ-13 dihydrochloride

    Catalog No. A12178
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    AQ-13 dihydrochloride is an aminoquinoline antimalarial drug that is effective against chloroquine-resistant strains of Plasmodium falciparum. 了解更多
  44. Ranolazine dihydrochloride

    Catalog No. A10781
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    Ranolazine dihydrochloride (CVT 303 dihydrochloride) is an anti-angina drug that achieves its effects by inhibiting the late phase of inward sodium current (INa and IKr with IC50 values of 6 μM and 12 μM, respectively) without affecting heart rate or blood pressure (BP). 了解更多
  45. L-NIO dihydrochloride

    Catalog No. A13027
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    NOS inhibitor
    L-NIO dihydrochloride is a potent, non-selective and NADPH-dependent nitric oxide synthase (NOS) inhibitor. 了解更多
  46. Levocetirizine Dihydrochloride

    Catalog No. A17440
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    L-isomer of cetirizine and histamine H1 receptor antagonist
    Levocetirizine dihydrochloride is a L-isomer of cetirizine and histamine H1 receptor antagonist. It incrases levels of CD4+ CD25+ T cells and decreases levels of eosinophils, decreasing allergy symptoms. 了解更多
  47. LY2801653 dihydrochloride

    Catalog No. A15150
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    MET 抑制剂
    LY2801653 dihydrochloride是一种有效的,口服可生物利用的c-MET激酶小分子抑制剂(Ki = 2 nM)。 了解更多
  48. H-1152 dihydrochloride

    Catalog No. A15102
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    ROCK 抑制剂
    H-1152 dihydrochloride是一种异喹啉磺酰胺衍生物,是Rho激酶的一种更特异,更强且可透过膜的抑制剂,Ki值为1.6 nM,但对其他丝氨酸/苏氨酸激酶的抑制作用较弱。 了解更多
  49. Pramipexole dihydrochloride monohyrate

    Catalog No. A10747
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    Dopamine Receptor 激动剂
    Pramipexole dihydrochloride monohyrate是非麦角灵类的多巴胺激动剂,适用于治疗早期帕金森氏病(PD)和不安腿综合征(RLS)。 了解更多
  50. 3AC

    Catalog No. A12817
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    SHIP1 抑制剂
    3AC是SHIP1多磷酸酶对PIP3的活性的细胞渗透性选择性抑制剂(IC50 = 10μM),但对SHIP2或PIP3的PTEN活性没有影响。 了解更多

产品 1 到 50 共 117个

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