Cathepsin Inhibitor 1

Name: Cathepsin Inhibitor 1
SKU: A11466

目录号: A11466

Cathepsin 抑制剂

Cathepsin Inhibitor 1 Chemical Structure

CAS NO. 225120-65-0

Cathepsin Inhibitor 1抑制剂1 是一种Cathepsin (L, L2, S, K, B)的抑制剂，pIC50分别为7.9、6.7、6.0、5.5和5.2。

库存：现货

规格	价格	数量
5 mg	￥ 1,100.00
10 mg	￥ 2,000.00
50 mg	￥ 6,000.00

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产品仅用于科学研究，不针对患者销售，望谅解.

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生物活性

Cathepsin Inhibitor 1抑制剂1 是一种Cathepsin (L, L2, S, K, B)的抑制剂，pIC50分别为7.9、6.7、6.0、5.5和5.2。

靶点信息

Cathepsin L	Cathepsin L2	Cathepsin S	Cathepsin K	Cathepsin S
7.9(pIC50)	6.7(pIC50)	6(pIC50)	5.5(pIC50)	5.2(pIC50)

溶解度 *

In vitro	DMSO	70 mg/mL (174.17 mM)
	Water	Insoluble
	Ethanol	44 mg/mL (109.48 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	24.88 mL	124.41 mL	248.82 mL
0.5 mM	4.98 mL	24.88 mL	49.76 mL
1 mM	2.49 mL	12.44 mL	24.88 mL
5 mM	0.5 mL	2.49 mL	4.98 mL

*The above data is based on the productmolecular weight 401.89. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11466
作用机制	Inhibitor (抑制剂)
M. Wt	401.89
Formula	C20H24ClN5O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	225120-65-0
SMILES	CC(C)(C)C1=NN(C(=C1)C(=O)NC(CC2=CC(=CC=C2)Cl)C(=O)NCC#N)C