CCT129202

目录号: A10184

Aurora 抑制剂

CCT129202

CCT129202 Chemical Structure

CAS NO. 942947-93-5

CCT129202是一种ATP竞争性的pan-Aurora抑制剂,作用于Aurora A,Aurora B和Aurora C时,IC50分别为0.042 μM,0.198 μM和0.227 μM,对FGFR3, GSK3β, PDGFRβ等作用效果稍弱。

库存: 现货

规格 价格 数量
5 mg
¥ 950.00
10 mg
¥ 1,800.00
50 mg
¥ 5,200.00
100 mg
¥ 9,380.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

CCT129202是一种ATP竞争性的pan-Aurora抑制剂,作用于Aurora A,Aurora B和Aurora C时,IC50分别为0.042 μM,0.198 μM和0.227 μM,对FGFR3, GSK3β, PDGFRβ等作用效果稍弱。
靶点信息
Aurora A Aurora B Aurora C
42 nM198 nM227 nM
In vitro (25°C) DMSO 3 mg/mL (6.03 mM)
Water Insoluble
Ethanol Insoluble
In vivo 1% DMSO+30% polyethylene glycol+1% Tween 80 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.12 mL 100.6 mL 201.21 mL
0.5 mM 4.02 mL 20.12 mL 40.24 mL
1 mM 2.01 mL 10.06 mL 20.12 mL
5 mM 0.4 mL 2.01 mL 4.02 mL

*The above data is based on the productmolecular weight 497.0 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A10184
作用机制 Inhibitor (抑制剂)
M. Wt 497.0
Formula C23H25ClN8OS
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 942947-93-5
Synonyms CCT-129202
SMILES CN(C)C1=CC=C(C=C1)C2=NC3=NC=C(C(=C3N2)N4CCN(CC4)CC(=O)NC5=NC=CS5)Cl

产品标签

产品标签

其他人对该产品使用了下列标签:

使用空格分隔标签。使用单引号(')标注词组。

Product Questions

Product Questions

No Questions
Keywords:购买 CCT129202 | CCT129202 供应商 | 订购 CCT129202 | CCT129202 价格 | CCT129202 生产商 | 订单 CCT129202 | CCT129202 代理商 | 购买 942947-93-5| 942947-93-5 供应商 | 订购 942947-93-5 | 942947-93-5 价格 | 942947-93-5 生产商 | 订单 942947-93-5 | 942947-93-5 代理商|buy CCT129202 | CCT129202 Supplier | purchase CCT129202 | CCT129202 cost | CCT129202 manufacturer | order CCT129202 | CCT129202 distributor | buy 942947-93-5| 942947-93-5 Supplier | purchase 942947-93-5 | 942947-93-5 cost | 942947-93-5 manufacturer | order 942947-93-5 | 942947-93-5 distributor
Rewards