DYRK

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  1. NU 6102

    Catalog No. A12438
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    CDK 抑制剂
    NU 6102与CDK4/D1(IC50 = 1.6μM),DYRK1A(IC50 = 0.9μM),PDK1(IC50 = 0.8μM)和ROCKII(IC50 = 0.6μM)相比,NU6102对CDK1和CDK2具有选择性。 了解更多
  2. ID 8

    Catalog No. A12922
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    DYRK 抑制剂
    ID-8是DYRK抑制剂。ID 8还以稳定的速率刺激增殖(在30天的补充有10 μM的无血清培养基中观察到)。 了解更多
  3. AZ191

    Catalog No. A14314
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    DYRK 抑制剂
    AZ191是一种有效的选择性DYRK1B抑制剂,IC50为17 nM,选择性比DYRK1A和DYRK2高5到110倍。 了解更多
  4. Mirk-IN-1

    Catalog No. A16255
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    Dyrk1B 抑制剂
    Mirk-IN-1是有效的Dyrk1B(Mirk kianse)和Dyrk1A抑制剂,IC50分别为68±48 nM和22±8 nM。 了解更多
  5. 10058-F4

    Catalog No. A13725
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    c-Myc-Max 抑制剂
    10058-F4是c-Myc抑制剂,可防止c-Myc/Max二聚化。 了解更多
  6. KJ Pyr 9

    Catalog No. A16324
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    MYC 抑制剂
    KJ Pyr 9是来自Krhnke吡啶库的MYC的新型小分子抑制剂KJ-Pyr-9。 了解更多
  7. ML327

    Catalog No. A17009
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    MYC 抑制剂
    ML327是MYC的阻止者。ML327介导E-钙黏着蛋白的转录去阻遏和上皮到间充质转化的抑制。 了解更多
  8. 10074-G5

    Catalog No. A17169
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    c-Myc 抑制剂
    10074-G5是c-Myc抑制剂,可抑制c-Myc/Max异二聚体形成并抑制其转录活性,IC50值为146μM。 了解更多
  9. sAJM589

    Catalog No. A18429
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    Myc 抑制剂
    sAJM589 is a Myc inhibitor which potently disrupts the Myc-Max heterodimer with an IC50 of 1.8 μM. 了解更多
  10. EHT 5372

    Catalog No. A12586
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    DYRK inhibitor
    EHT 5372 is a strong inhibitor of DYRK??s family kinases, with IC50s of 0.22, 0.28 nM for DYRK1A and DYRK1B, respectively. 了解更多
  11. LDN-192960 hydrochloride

    Catalog No. A21390
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    DYRK2 inhibitor
    LDN-192960 hydrochloride is an inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50s of 10 nM and 48 nM, respectively. 了解更多

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