Endocrinology / Hormones

产品 1 到 50 共 236个

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  1. (Glp1)-Apelin-13

    Catalog No. A13215
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    Apelin Receptor activator
    (Glp1)-Apelin-13是Apelin受体的激活剂。 了解更多
  2. SR-2211

    Catalog No. A13568
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    RORr 激动剂
    SR-2211选择性结合RORr(Ki = 105 nM),充当体外本构RORr活性的反向激动剂(IC50 = 320 nM)。 了解更多
  3. AGN-242428

    Catalog No. A16935
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    RORγt 抑制剂
    AGN-242428,也称为VTP-43742,是一种有效的,选择性的和口服活性的RORγ抑制剂,Ki值为<100 nM。用于治疗自身免疫性疾病,包括多发性硬化症和牛皮癣。 了解更多
  4. Cintirorgon (LYC-55716)

    Catalog No. A16863
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    RORγ 激动剂
    Cintirorgon (LYC-55716)是新型口服RAR相关孤儿受体γ(RORγ)激动剂。 了解更多
  5. AZD-0284

    Catalog No. A18766
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    RORγ 激动剂
    AZD-0284 is a potent, selective, inverse agonist of the nuclear receptor RORγ for the potential treatment of Plaque psoriasis. 了解更多
  6. XY101

    Catalog No. A18437
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    RORγ inverse 激动剂
    XY101 is a potent, selective, metabolically stable and orally available RORγ inverse agonist with an IC50 of 30 nM and a Kd of 380 nM. 了解更多
  7. S18-000003

    Catalog No. A19105
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    RORγt 抑制剂
    S18-000003 is a potent orally bioavailable retinoic acid receptor-related orphan receptor-gamma-t (RORγt) inhibitor with an IC50 of 29 nM. S18-000003 inhibits IL-17 production. 了解更多
  8. A-9758

    Catalog No. A19078
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    RORγt inverse 激动剂
    A-9758 is a RORγ ligand and a potent, selective RORγt inverse agonist (IC50=5 nM), and exhibits robust potency against IL-17A release. 了解更多
  9. ROR agonist-1

    Catalog No. A18569
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    ROR 激动剂
    ROR agonist-1 is a potent and orally bioavailable inverse agonist of the retinoic acid receptor-related orphan receptor C2 (RORC2), inhibition of IL-17A production from human primary TH 17 cells with a pIC50 of 7.5. 了解更多
  10. SR1078

    Catalog No. A15245
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    ROR 激动剂
    SR1078是视黄酸受体相关的孤儿受体(ROR)RORα/γ的激动剂;增加RORα靶基因的转录;认为可以增加p53的稳定性。 了解更多
  11. SR3335

    Catalog No. A15246
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    RORα 激动剂
    SR3335是一种选择性RORα合成配体,直接与RORα结合,但不与其他ROR结合,并且在基于细胞的测定中用作RORα的选择性部分反向激动剂。 了解更多
  12. SR1001

    Catalog No. A13193
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    ROR 激动剂
    SR1001是选择性的ROR-α和ROR-γ反向激动剂;抑制TH17细胞分化并抑制自身免疫。 了解更多
  13. ROR gamma modulator 1

    Catalog No. A16291
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    RORγ modulator
    ROR gamma modulator 1 是类维生素A相关的孤儿受体γ(RORy)调节剂 了解更多
  14. Ozarelix

    Catalog No. A12350
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    GnRH 拮抗剂
    Ozarelix是第四代GnRH拮抗剂,诱导激素难治性雄激素受体阴性前列腺癌细胞凋亡,调节死亡受体的表达和活性。 了解更多
  15. Abarelix Acetate

    Catalog No. A12613
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    GnRH 拮抗剂
    Abarelix acetate是一种合成的肽促性腺激素释放激素受体(GnRH)拮抗剂。 了解更多
  16. NBI-42902

    Catalog No. A12375
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    GnRH receptor 抑制剂
    NBI-42902是人促性腺激素释放激素受体的新型非肽拮抗剂。 了解更多
  17. SR 144528

    Catalog No. A12376
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    CB2 inverse 激动剂
    SR 144528是一种选择性的外周大麻素受体反向激动剂,对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM,对大鼠脑和人重组CB1受体的Ki值为400 nM。 了解更多
  18. Ganirelix

    Catalog No. A12862
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    Ganirelix是一种可注射的竞争性促性腺激素释放激素拮抗剂(GnRH拮抗剂)。 了解更多
  19. Degarelix acetate

    Catalog No. A12840
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    GnRH 拮抗剂
    Degarelix acetate是促性腺激素释放激素(GnRH)受体拮抗剂。 了解更多
  20. GHRP-6 Acetate

    Catalog No. A13464
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    GHRP-6 Acetate是一种生长激素释放肽。 了解更多
  21. Elagolix sodium

    Catalog No. A13893
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    GnRH 拮抗剂
    Elagolix sodium是促性腺激素释放激素(GnRH)拮抗剂。Elagolix sodium抑制垂体腺中的促性腺激素释放激素(GnRH)受体,并最终降低循环性激素水平。 了解更多
  22. AEZS-108

    Catalog No. A13536
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    GnRH-1 激动剂
    AEZS-108是促性腺激素释放激素1受体(GnRH-1R)的肽激动剂,其与蒽环类抗生素阿霉素结合,具有潜在的抗肿瘤活性。 了解更多
  23. Leuprolide Acetate

    Catalog No. A15143
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    GnRH 激动剂
    Leuprolide Acetate是GnRH类似物;醋酸亮丙瑞林在垂体GnRH受体上起激动剂的作用。 了解更多
  24. Triptorelin Acetate

    Catalog No. A15997
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    GnRH 激动剂
    Triptorelin Acetate是一种促性腺激素释放激素激动剂(GnRH激动剂),用作乙酸盐或pamoate盐。 了解更多
  25. Goserelin Acetate

    Catalog No. A15959
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    GnRH 激动剂
    Goserelin Acetate是具有抗肿瘤活性的促黄体激素释放激素(LHRH)的合成十肽类似物。 了解更多
  26. Relugolix

    Catalog No. A17783
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    GnRH antagonist
    Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013. 了解更多
  27. Leuprorelin Acetate

    Catalog No. A17986
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    GnRH/LHRH receptor agonist
    Leuprorelin is a Gonadotropin-releasing hormone (GnRH, luteinizing hormone-releasing hormone, LHRH) receptor agonist. Suppresses estradiol, LH and FSH serum levels and represses the growth of experimental rat endometriosis. 了解更多
  28. Nafarelin Acetate

    Catalog No. A17992
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    GnRH agonist
    Nafarelin is a gonadotropin-releasing hormone agonist (GnRH agonist) which acts as an analog of GnRH. 了解更多
  29. Cetrorelix Acetate

    Catalog No. A18282
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    GnRH antagonist
    Cetrorelix acetate is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity used in infertility treatment. The IC50 of 1.21 nM. 了解更多
  30. Goserelin

    Catalog No. A21197
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    GnRH agonist
    Goserelin(ICI 118630) is an injectable gonadotropin releasing hormone superagonist (GnRH agonist). 了解更多
  31. (R)-Elagolix

    Catalog No. A21184
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    GnRHR antagonist
    Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). 了解更多
  32. Alarelin Acetate

    Catalog No. A20968
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    synthetic GnRH agonist
    Alarelin acetate is a synthetic GnRH agonist. 了解更多
  33. Ercalcidiol

    Catalog No. A11413
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    VD/VDR 抑制剂
    Ercalcidiol是D2的代谢物。 了解更多
  34. Betamethasone dipropionate

    Catalog No. A10130
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    Glucocorticoid Receptor 激动剂
    Betamethasone Dipropionate是糖皮质激素类固醇,具有抗炎和免疫抑制特性。 了解更多
  35. Betamethasone valerate (Betnovate, Celestone)

    Catalog No. A10131
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    Betamethasone valerate是一种有效的糖皮质激素类固醇,具有抗炎和免疫抑制作用 了解更多
  36. Budesonide

    Catalog No. A10166
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    Budesonide是一种糖皮质激素类固醇,可用于治疗哮喘,非感染性鼻炎 了解更多
  37. Prednisolone acetate (Omnipred)

    Catalog No. A11687
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    Prednisolone是合成的糖皮质激素,是皮质醇的衍生物,用于治疗各种炎症和自身免疫性疾病。 了解更多
  38. Deflazacort

    Catalog No. A10294
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    Deflazacort是一种糖皮质激素,用作抗炎和免疫抑制剂。 了解更多
  39. Hydrocortisone(Cortisol)

    Catalog No. A10457
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    Hydrocortisone是肾上腺产生的类固醇激素或糖皮质激素。 了解更多
  40. Meprednisone (Betapar)

    Catalog No. A10567
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    Meprednisone是糖皮质激素和泼尼松的甲基化衍生物。 了解更多
  41. Methylprednisolone

    Catalog No. A10582
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    Methylprednisolone是一种凋亡诱导剂,并且在体外也能抑制人小细胞肺癌细胞的生长。 了解更多
  42. Prednisone (Adasone)

    Catalog No. A10752
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    Glucocorticoid Receptor 激动剂
    Prednisone (Adasone)可降低粘膜TNF-a的产生,肠道通透性和NF-kB表达水平。 了解更多
  43. Fluticasone propionate

    Catalog No. A11860
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    Fluticasone propionate是一种高亲和力的选择性糖皮质激素受体激动剂(Kd = 0.5 nM)。 了解更多
  44. RU43044

    Catalog No. A14340
    Glucocorticoid receptor 拮抗剂
    RU43044在骨肉瘤细胞而非人乳腺癌细胞中发挥显着的激动剂活性并激活MMTV-Luc转录。 了解更多
  45. GW-870086

    Catalog No. A18343
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    Glucocorticoid receptor agonist
    GW-870086 is a potent anti-inflammatory agent, acting as a glucocorticoid receptor agonist, with a pIC50 of 10.1 in A549 cells expressing NF-κB. 了解更多
  46. Beclometasone

    Catalog No. A18177
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    glucocorticoid receptor agonist
    Beclometasone, also known as Beclomethasone, is an anti-inflammatory, synthetic glucocorticoid. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma. 了解更多
  47. AZD9567

    Catalog No. A18850
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    selective glucocorticoid receptor modulator
    AZD9567 is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. 了解更多
  48. OP-3633

    Catalog No. A18468
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    Glucocorticoid Receptor Antagonist
    OP-3633 is a Potent Steroidal Glucocorticoid Receptor Antagonist with Enhanced Selectivity against the Progesterone and Androgen Receptors (IC50 = 29 nM). 了解更多
  49. AZD5423

    Catalog No. A13249
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    nonsteroidal glucocorticoid receptor 激动剂
    AZD5423是新型的非甾体类糖皮质激素受体激动剂。 了解更多
  50. Fluorometholone

    Catalog No. A17651
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    glucocorticoid
    Fluorometholone is a glucocorticoid employed, usually as eye drops, in the treatment of allergic and inflammatory conditions of the eye. It has also been used topically in the treatment of various skin disorders. 了解更多

产品 1 到 50 共 236个

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