Flupirtine maleate

Name: Flupirtine maleate
SKU: A10251

目录号: A10251

NMDA 拮抗剂

Flupirtine maleate Chemical Structure

CAS NO. 75507-68-5

Flupirtine maleate是Flupirine的盐形式，是一种非阿片类中枢性镇痛药，是一种选择性的神经元钾离子通道开放剂，也具有NMDA受体拮抗剂特性。

库存：现货

规格	价格	数量
10 mg	￥ 300.00
25 mg	￥ 400.00
100 mg	￥ 900.00
10mM * 1mL in DMSO	￥ 720.00

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生物活性

Flupirtine maleate是Flupirine的盐形式，是一种非阿片类中枢性镇痛药，是一种选择性的神经元钾离子通道开放剂，也具有NMDA受体拮抗剂特性。

靶点信息

NMDA receptor	Potassium channel

溶解度 *

In vitro (25°C)	DMSO	76 mg/mL (180.78 mM)
	Water	Insoluble
	Ethanol	Warmed: 2 mg/mL (4.75 mM)
In vivo	30% propylene glycol, 5% Tween 80, 65% D5W	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	23.79 mL	118.93 mL	237.87 mL
0.5 mM	4.76 mL	23.79 mL	47.57 mL
1 mM	2.38 mL	11.89 mL	23.79 mL
5 mM	0.48 mL	2.38 mL	4.76 mL

*The above data is based on the productmolecular weight 420.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A10251
作用机制	Antagonist (拮抗剂)
M. Wt	420.4
Formula	C15H17FN4O2.C4H4O4
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	75507-68-5
Synonyms	D 9998
SMILES	CCOC(=O)NC1=C(N=C(C=C1)NCC2=CC=C(C=C2)F)N.C(=C\C(=O)O)\C(=O)O