“jwh 307”的搜索结果

产品 1 到 50 共 107个

每页
页面:
  1. 1
  2. 2
  3. 3

设置降序顺序
  1. Flumatinib

    Catalog No. A16258
    Quick View
    multi-kinase 抑制剂
    Flumatinib是一种多激酶抑制剂,对c-Abl,PDGFRbeta和c-Kit的IC50值分别为1.2 nM,307.6 nM和2662 nM。 了解更多
  2. RY785

    Catalog No. A22104
    Quick View
    inhibitor of Kv2.1 and Kv2.2
    RY785 (Kv2-IN-A1) is an inhibitor of Kv2.1 and Kv2.2. 了解更多
  3. LDN-193189 2HCl

    Catalog No. A22307
    Quick View
    BMP signaling inhibitor
    LDN193189 HCl (DM-3189) is the hydrochloride salt of LDN193189, which is a selective BMP signaling inhibitor, and inhibits the transcriptional activity of the BMP type I receptors ALK2 and ALK3 with IC50 of 5 nM and 30 nM in C2C12 cell lines, respectively, 200-fold selectivity for BMP versus TGF-β. 了解更多
  4. Higenamine

    Catalog No. A22315
    Quick View
    β2-AR agonist
    Higenamine (Norcoclaurine), a β2-AR agonist, is a key component of the Chinese herb aconite root that prescribes for treating symptoms of heart failure in the oriental Asian countries. 了解更多
  5. BIO-013077-01

    Catalog No. A22185
    Quick View
    antagonist of the TGFbeta family type I receptors, Alk5 and/or Alk4
    BIO-013077-01, Novel potent antagonist of the TGFbeta family type I receptors, Alk5 and/or Alk4. 了解更多
  6. (R)-Propranolol hydrochloride

    Catalog No. A22258
    Quick View
    β-adrenergic receptor (βAR) antagonist
    (R)-Propranolol hydrochloride is a less active enantiomer of the β-adrenoceptor antagonist propranolol (HY-B0573). Propranolol is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively. 了解更多
  7. BTK inhibitor 1 (Compound 27)

    Catalog No. A22445
    Quick View
    BTK inhibitor
    BTK inhibitor 1 (compound 27) is an inhibitor of BTK with an IC50 of 0.11 nM for Btk and inhibits B cell activation in hWB with an IC50 of 2 nM. 了解更多
  8. GRA Ex-25

    Catalog No. A20625
    Quick View
    glucagon receptor inhibitor
    GRA Ex-25 is an inhibitor of glucagon receptor, with IC50 of 56 and 55 nM for rat and human glucagon receptors, respectively. 了解更多
  9. ST034307

    Catalog No. A20414
    Quick View
    AC1 inhibitor
    ST034307 is a potent and selective adenylyl cyclase 1 (AC1) inhibitor, with IC50 of 2.3 μM. 了解更多
  10. Simurosertib

    Catalog No. A20392
    Quick View
    CDC7 inhibitor
    Simurosertib (TAK-931) is a selective cycle 7 (CDC7) kinase inhibitor, with an IC50<0.3 nM. 了解更多
  11. Antifungal agent 1

    Catalog No. A20307
    Quick View
    Antifungal agent 1 is a potent antifungal agent. 了解更多
  12. N6-Cyclopentyladenosine

    Catalog No. A19595
    Quick View
    Adenosine A1 receptor agonist
    N6-Cyclopentyladenosine (CPA) is a selective Adenosine A1 receptor agonist, with Ki values of 2.3 nM, 790 nM and 43 nM for human A1, A2A and A3 receptors, respectively. 了解更多
  13. Ds-HAPP

    Catalog No. A19307
    Quick View
    Ds-HAPP is an anthrancenyl and dansyl fluorophore ligand. 了解更多
  14. PLpro inhibitor

    Catalog No. A21044
    Quick View
    Plpro inhibitor
    PLpro inhibitor is a potent inhibitor of papain-like protease (PLpro) with IC50 of 2.6 uM. 了解更多
  15. (R)-Simurosertib

    Catalog No. A21894
    Quick View
    CDC7 kinase inhibitor
    (R)-Simurosertib ((R)-TAK-931) is the (R)-enantiomer of Simurosertib, Simurosertib (TAK-931) is a selective cycle 7 (CDC7) kinase inhibitor, with an IC50<0.3 nM. 了解更多
  16. ATN-161

    Catalog No. A21307
    Quick View
    integrin α5β1 antagonist
    ATN-161 is a novel integrin α5β1 antagonist, which inhibits angiogenesis and growth of liver metastases in a murine model. 了解更多
  17. Emiglitate

    Catalog No. A20917
    Quick View
    α-glucoside hydrolase inhibitor
    Emiglitate (BAY o 1248) is a potent, selective and competitive inhibitor of α-glucoside hydrolase. 了解更多
  18. Diclofenac

    Catalog No. A17814
    Quick View
    COX inhibitor
    Diclofenac is a potent and nonselective anti-inflammatory agent, acts as a COX inhibitor, with IC50s of 4 nM, 1.3 nM for human COX-1 and COX-2 in CHO cells, and 5.1, 0.84 μM for ovine COX-1 and COX-2, respectively. 了解更多
  19. (4-Acetamidocyclohexyl) nitrate

    Catalog No. A13355
    Quick View
    guanylate cyclase activator
    (4-Acetamidocyclohexyl) nitrate (BM121307) is a guanylate cyclase activator that was in phase I development for the treatment of ischaemic heart disorders. The research has been discontinued. 了解更多
  20. Y-33075 dihydrochloride

    Catalog No. A11611
    Quick View
    ROCK inhibitor
    Y-33075 dihydrochloride is a selective ROCK inhibitor with an IC50 of 3.6 nM. 了解更多
  21. NMDI14

    Catalog No. A12958
    Quick View
    NMD inhibitor
    NMDI14 is a nonsense mediated RNA decay (NMD) inhibitor. 了解更多
  22. Ipenoxazone

    Catalog No. A12307
    Quick View
    Ipenoxazone is a potent and centrally acting muscle relaxant. 了解更多
  23. GSK2593074A

    Catalog No. A13600
    Quick View
    necroptosis inhibitor
    GSK2593074A (GSK??074) is a necroptosis inhibitor with dual targeting ability to both RIP1 and RIP3. 了解更多
  24. BAY885

    Catalog No. A13765
    Quick View
    ERK5 inhibitor
    BAY885 is a novel ERK5 inhibitor. 了解更多
  25. STF-083010

    Catalog No. A16720
    Quick View
    IRE1α inhibitor
    STF-083010 is a specific IRE1α inhibitor. STF-083010 inhibits Ire1 endonuclease activity, without affecting its kinase activity, after endoplasmic reticulum stress. 了解更多
  26. Levoleucovorin Calcium

    Catalog No. A11626
    Quick View
    Levoleucovorin calcium is the calcium salt of Levoleucovorin, which is the enantiomerically active form of folinic acid. 了解更多
  27. Enzaplatovir

    Catalog No. A20830
    Quick View
    RSV fusion protein inhibitor
    Enzaplatovir is an inhibitor of Respiratory Syncytial Virus (RSV). It can be used as a viral fusion protein inhibitor. 了解更多
  28. RTC-30

    Catalog No. A18865
    Quick View
    RTC-30 is an optimized phenothiazine with anti-cancer potency. RTC-30 contains a hydroxylated linker (N) that confers increased oral bioavailability. 了解更多
  29. NNC0640

    Catalog No. A18900
    Quick View
    GLP-1R modulator
    NNC0640 is a negative allosteric modulator of glucagon-like peptide-1 receptor (GLP-1R). 了解更多
  30. RTC-5

    Catalog No. A19067
    Quick View
    RTC-5 is an optimized phenothiazine with anti-cancer potency. RTC-5 demonstrates efficacy against a xenograft model of an EGFR driven cancer, its effects is attributed to concomitant negative regulation of PI3K-AKT and RAS-ERK signaling. 了解更多
  31. ODM-203

    Catalog No. A19098
    Quick View
    FGFR/VEGFR 抑制剂
    ODM-203 is a potent FGFR and VEGFR families inhibitor with IC50s of 11, 16, 6, 35 nM towards recombinant FGFR1, FGFR2, FGFR3 and FGFR4 as well as 26, 9, 5 nM towards VEGFR1, VEGFR2 and VEGFR3, respectively. 了解更多
  32. LY-2940094

    Catalog No. A19125
    Quick View
    NOP receptor antagonist
    LY-2940094 is a potent, selective and orally available nociceptin receptor (NOP receptor) antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY-2940094 reduces ethanol self-administration in animal models. 了解更多
  33. AN11251

    Catalog No. A19475
    Quick View
    AN11251 is a potent and oral active anti-Wolbachia agent with potential for treatment of onchocerciasis and lymphatic filariasis, with EC50 values of 1.5 nM in LDW1 cell lines and 15 nM in C6/36 cell lines. 了解更多
  34. ZXH-3-26

    Catalog No. A18399
    Quick View
    PROTAC BRD4 degrader
    ZXH-3-26 is a selective PROTAC BRD4 degrader with a DC50/5h (DC50/5h referring to half-maximal degradation after 5 hours of treatment) of ~ 5 nM. 了解更多
  35. GRL0617

    Catalog No. A18780
    Quick View
    SARS PLPro inhibitor
    GRL0617 is a potent, selective and competitive noncovalent inhibitor of SARS PLPro, with an IC50 of 0.6 μM, and with a Ki of 0.49 μM. 了解更多
  36. Metoclopramide hydrochloride hydrate

    Catalog No. A18072
    Quick View
    Dopamine D2 antagonist
    Metoclopramide hydrochloride hydrate is a dopamine D2 antagonist that is used as an antiemetic. 了解更多
  37. o-Cresol

    Catalog No. A17823
    Quick View
    o-Cresol is a compound used as a disinfectant and have also been used as antiseptic in surgery. 了解更多
  38. Revaprazan Hydrochloride

    Catalog No. A17506
    Quick View
    Acid pump antagonist
    Revaprazan hydrochloride is a novel acid pump antagonist (APA). Revaprazan hydrochloride reduces COX-2 expression and has significant anti-inflammatory actions activities in H. pylori infection. 了解更多
  39. Benznidazole

    Catalog No. A17307
    Quick View
    Benznidazol (Ro 07-1051) is an antiparasitic medication, with an IC50 of 20.35 μM for Colombian T. cruzi strains, and has been used in the treatment of Chagas disease. 了解更多
  40. Treponema TmpA 45kDa

    Catalog No. AP6307
    Quick View
    Treponema pallidum TmpA, 45kDa Recombinant 了解更多
  41. IL 16 Human, (121 a.a.)

    Catalog No. AP5307
    Quick View
    Interleukin-16 Human Recombinant, (121 a.a.) 了解更多
  42. GSTT1 Human

    Catalog No. AP4904
    Quick View
    Glutathione S-Transferase Theta-1 Human Recombinant 了解更多
  43. NAE1 Human

    Catalog No. AP4307
    Quick View
    NEDD8 Activating Enzyme E1 Subunit 1 Human Recombinant 了解更多
  44. Procalcitonin Mouse

    Catalog No. AP3307
    Quick View
    Procalcitonin Mouse Recombinant 了解更多
  45. CRABP2 Antibody

    Catalog No. AP3079
    Quick View
    Cellular Retinoic Acid binding Protein 2, Mouse Anti Human 了解更多
  46. FABP7 Antibody

    Catalog No. AP3078
    Quick View
    Fatty Acid Binding Protein-7, Mouse Anti Human 了解更多
  47. CFL1 Antibody

    Catalog No. AP3077
    Quick View
    Cofilin-1, Mouse Anti Human 了解更多
  48. BID Antibody

    Catalog No. AP3076
    Quick View
    BH3 Interacting Domain Death Agonist , Mouse Anti Human 了解更多
  49. VAMP3 Antibody

    Catalog No. AP3075
    Quick View
    Synaptobrevin-3, Mouse Anti Human 了解更多
  50. CHGA Antibody

    Catalog No. AP3074
    Quick View
    Chromogranin-A, Mouse Anti Human 了解更多

产品 1 到 50 共 107个

每页
页面:
  1. 1
  2. 2
  3. 3

设置降序顺序
Rewards