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Linagliptin (BI-1356)

Linagliptin (BI-1356)

Name: Linagliptin (BI-1356)
SKU: A11224

目录号: A11224

DPP-4 抑制剂

Linagliptin (BI-1356) Chemical Structure

CAS NO. 668270-12-0

Linagliptin (BI-1356)是DPP-4抑制剂，是一种降解肠降血糖素激素胰高血糖素样肽1（GLP-1）和葡萄糖依赖性促胰岛素多肽（GIP）的酶。

库存：现货

规格	价格	数量
100 mg	￥ 400.00
500 mg	￥ 700.00
10mM * 1mL in DMSO	￥ 500.00

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生物活性

Linagliptin (BI-1356)是DPP-4抑制剂，是一种降解肠降血糖素激素胰高血糖素样肽1（GLP-1）和葡萄糖依赖性促胰岛素多肽（GIP）的酶。

靶点信息

DPP-4
1 nM

溶解度 *

In vitro (25°C)	DMSO	16 mg/mL (33.85 mM)
	Water	Insoluble
	Ethanol	1 mg/mL (2.11 mM)
In vivo	0.5% hydroxyethyl cellulose	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	21.16 mL	105.82 mL	211.64 mL
0.5 mM	4.23 mL	21.16 mL	42.33 mL
1 mM	2.12 mL	10.58 mL	21.16 mL
5 mM	0.42 mL	2.12 mL	4.23 mL

*The above data is based on the productmolecular weight 472.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11224
作用机制	Inhibitor (抑制剂)
M. Wt	472.5
Formula	C25H28N8O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	668270-12-0
Synonyms	BI-1356,Tradjenta,Trajenta
SMILES	CC#CCN1C2=C(N=C1N3CCC[C@H](C3)N)N(C(=O)N(C2=O)CC4=NC5=CC=CC=C5C(=N4)C)C