MK-3207

Name: MK-3207
SKU: A15165

目录号: A15165

CGRP Receptor 拮抗剂

MK-3207 Chemical Structure

CAS NO. 957118-49-9

MK-3207是一种有效且口服可生物利用的CGRP受体拮抗剂（IC50 = 0.12 nM；Ki = 0.024 nM）；对人类AM1，AM2，CTR和AMY3具有高度选择性。

库存：现货

规格	价格	数量
10 mg	￥ 2,000.00
25 mg	￥ 3,800.00
50 mg	￥ 6,500.00

大包装询价

或

添加到收藏

产品仅用于科学研究，不针对患者销售，望谅解.

产品详情

生物活性

MK-3207是一种有效且口服可生物利用的CGRP受体拮抗剂（IC50 = 0.12 nM；Ki = 0.024 nM）；对人类AM1，AM2，CTR和AMY3具有高度选择性。

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	17.93 mL	89.67 mL	179.34 mL
0.5 mM	3.59 mL	17.93 mL	35.87 mL
1 mM	1.79 mL	8.97 mL	17.93 mL
5 mM	0.36 mL	1.79 mL	3.59 mL

*The above data is based on the productmolecular weight 557.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15165
作用机制	Antagonist (拮抗剂)
M. Wt	557.59
Formula	C31H29F2N5O3
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	957118-49-9
Synonyms	MK3207, MK 3207
SMILES	C1CCC2(C1)C(=O)N(C(CN2)C3=CC(=CC(=C3)F)F)CC(=O)NC4=CC5=C(CC6(C5)C7=C(NC6=O)N=CC=C7)C=C4