(-)-MK 801 maleate

Name: (-)-MK 801 maleate
SKU: A13435

目录号: A13435

NMDA receptor 拮抗剂.

(-)-MK 801 maleate Chemical Structure

CAS NO. 121917-57-5

(-)-MK 801 maleate是一种有效的、选择性的、非竞争性的NMDA受体拮抗剂。它通过与NMDA相关离子通道内的一个位点结合而起作用。

库存：现货

规格	价格	数量
25 mg	￥ 1,000.00
50 mg	￥ 1,850.00
100 mg	￥ 3,200.00

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生物活性

(-)-MK 801 maleate是一种有效的、选择性的、非竞争性的NMDA受体拮抗剂。它通过与NMDA相关离子通道内的一个位点结合而起作用。

靶点信息

NMDA Receptor
30.5 nM(Ki)

溶解度 *

In vitro (25°C)	DMSO	63 mg/mL (186.73 mM)
	Water	Insoluble
	Ethanol	7 mg/mL (20.74 mM)
In vivo	2% DMSO+40% PEG 300+2% Tween 80+ddH2O	7 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	29.64 mL	148.21 mL	296.41 mL
0.5 mM	5.93 mL	29.64 mL	59.28 mL
1 mM	2.96 mL	14.82 mL	29.64 mL
5 mM	0.59 mL	2.96 mL	5.93 mL

*The above data is based on the productmolecular weight 337.37. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A13435
作用机制	Antagonist (拮抗剂)
M. Wt	337.37
Formula	C16H15NC4H4O4
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	121917-57-5
Synonyms	MK801, MK-801
SMILES	C[C@]12C3=CC=CC=C3C[C@H](N1)C4=CC=CC=C24.C(=C/C(=O)O)\C(=O)O