MAO

Catalog No.Inhibitor Name MAO-AMAO-BMAOOther
A10818Safinamide Mesylate
*
****
A11722Rasagiline Mesylate
***
****
A11885Moclobemide
***
A10690Paeonol
*
**
A13358Tranylcypromine HCl
CYP2A6

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

30 个项目

每页

设置升序顺序
  1. Brofaromine

    Catalog No. A21777
    Quick View
    MAO inhibitor
    Brofaromine (CGP 11305A) is a monoamine oxidase (MAO) inhibitor with IC50 of 0.2?μM for MAO-A. 了解更多
  2. Ro 41-1049 hydrochloride

    Catalog No. A21672
    Quick View
    inhibitor of monoamine oxidase-A (MAO-A)
    Ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine oxidase-A (MAO-A). 了解更多
  3. Lazabemide

    Catalog No. A21270
    Quick View
    MAO-B inhibitor
    Lazabemide(Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively). 了解更多
  4. RS 8359

    Catalog No. A21240
    Quick View
    MAO-A inhibitor
    RS 8359 is a selective and reversible MAO-A inhibitor, with antidepressant activity. 了解更多
  5. Salsolidine

    Catalog No. A12969
    Quick View
    MAO-A inhibitor
    Salsolidine is a tetrahydroisoquinoline alkaloid, acts as a stereoselective competitive MAO A inhibitor. 了解更多
  6. CX-157

    Catalog No. A12200
    Quick View
    MAO-A inhibitor
    CX-157 is a reversible inhibitor of monoamine oxidase-A (MAO-A) with an EC50 of 19.3?ng/mL. 了解更多
  7. TB5

    Catalog No. A13170
    Quick View
    hMAO-B inhibitor
    TB5 is a potent, selective and reversible inhibitor of hMAO-B with a Ki value of 0.11??0.01 μM. 了解更多
  8. Iproniazid phosphate

    Catalog No. A18135
    Quick View
    MAO inhibitor
    Iproniazid phosphate is an irreversible inhibitor of monoamine oxidase types A and B that is used as an antidepressive agent. It has also been used as an antitubercular agent, but its use is limited by its toxicity. 了解更多
  9. Toloxatone

    Catalog No. A18043
    Quick View
    MAO-A inhibitor
    Toloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor. Antidepressant. 了解更多
  10. Minaprine dihydrochloride

    Catalog No. A17722
    Quick View
    MAO-A inhibitor
    Minaprine is a reversible inhibitor of MAO-A; weakly inhibit acetylcholinesterase; an antidepressant for treatment of depression. 了解更多
  11. Molindone hydrochloride

    Catalog No. A17647
    Quick View
    MAO inhibitor
    Molindone HCl is a D2 dopamine receptor antagonist. It also acts as a MAO inhibitor. 了解更多
  12. Iproniazid

    Catalog No. A17445
    Quick View
    MAO inhibitor
    Iproniazid is a non-selective, irreversible monoamine oxidase (MAO) inhibitor (MAOI) that is used as an antidepressive agent. 了解更多
  13. Pargyline hydrochloride

    Catalog No. A17288
    Quick View
    MAO inhibitor
    Pargyline hydrochloride is an irreversible inhibitor of monoamine oxidase (MAO) that is used clinically to treat moderate hypertension. 了解更多
  14. Olodaterol

    Catalog No. A15761
    Quick View
    MAO 抑制剂
    Olodaterol是一种长效的β肾上腺素受体激动剂,由Boehringer-Ingelheim生产,用于吸入治疗慢性阻塞性肺疾病(COPD)患者。 了解更多
  15. Rasagiline

    Catalog No. A11111
    Quick View
    MAO B 抑制剂
    Rasagiline是MAO-B(单胺氧化酶-B)的选择性不可逆抑制剂。 了解更多
  16. Hordenine

    Catalog No. A10454
    Quick View
    MAO-B 抑制剂
    Hordenine是一种苯乙胺生物碱,具有抗菌和抗生素特性。 了解更多
  17. Quercetin (Sophoretin)

    Catalog No. A10766
    Quick View
    MAO-B 抑制剂
    Quercetin (Sophoretin)抑制许多酶系统,包括酪氨酸蛋白激酶,磷脂酶A2,磷酸二酯酶,线粒体ATPase,PI 3-激酶和蛋白激酶C。 了解更多
  18. Quercetin dihydrate (Sophoretin)

    Catalog No. A10765
    Quick View
    MAO-B 抑制剂
    Quercetin dihydrate (Sophoretin)抑制许多酶系统,包括酪氨酸蛋白激酶,磷脂酶A2,磷酸二酯酶,线粒体ATPase,PI 3-激酶和蛋白激酶C。 了解更多
  19. PAT-1251 Hydrochloride

    Catalog No. A21969
    Quick View
    LOXL2 inhibitor
    PAT-1251 Hydrochloride is a potent, selective and oral lysyl oxidase-like 2 (LOXL2) inhibitor, with IC50s of 0.71 and 1.17 μM for hLOXL2 and hLOXL3, respectively, and also potently inhibits mouse, rat, and dog LOXL2 (IC50s, 0.10, 0.12, and 0.16 μM, respectively). 了解更多
  20. Rasagiline 13C3 mesylate racemic

    Catalog No. A21350
    Quick View
    Monoamine oxidase inhibitor
    Rasagiline 13C3 mesylate racemic is the deuterium labeled Rasagiline, which is an irreversible inhibitor of monoamine oxidase. 了解更多
  21. Isocarboxazid

    Catalog No. A17887
    Quick View
    monoamine oxidase inhibitor
    Isocarboxazid is a non-selective and irreversible inhibitor of monoamine oxidase, with an IC50 of 4.8 μM for rat brain monoamine oxidase in vitro. 了解更多
  22. Clorgyline hydrochloride

    Catalog No. A17357
    Quick View
    monoamine oxidase A inhibitor
    Clorgyline hydrochloride is an irreversible and selective inhibitor of monoamine oxidase A (MAO-A) that is used in scientific research; structurally related to Pargyline. 了解更多
  23. Safinamide Mesylate (FCE28073)

    Catalog No. A10818
    Quick View
    MAO 抑制剂
    Safinamide Mesylate是沙芬酰胺的甲磺酸盐,可选择性和可逆地抑制MAO-B,IC50为0.45μM。 了解更多
  24. Rasagiline mesylate

    Catalog No. A11722
    Quick View
    Monoamine oxidase 抑制剂
    Rasagiline mesylate是一种不可逆的单胺氧化酶抑制剂,在早期帕金森氏病中用作单一疗法,在较晚期的病例中用作辅助疗法。对于B型MAO,它对A型的选择性是14倍。 了解更多
  25. SL251188

    Catalog No. A11777
    Quick View
    MAO-B 抑制剂
    SL-251188是恶唑烷酮衍生物,在狒狒中被表征为放射性配体,可使用正电子发射断层扫描(PET)在体内可视化MAO-B。 了解更多
  26. Moclobemide

    Catalog No. A11885
    Quick View
    MAO 抑制剂
    Moclobemide是单胺氧化酶A(MAO-A)的可逆和选择性抑制剂。 了解更多
  27. Bifemelane HCl

    Catalog No. A13353
    Quick View
    MAO 抑制剂
    Bifemelane hydrochloride是抗抑郁的MAO抑制剂。逆转丁苯那嗪在小鼠中引起的僵直,并增加MPTP处理的mar猴的自发活动。 了解更多
  28. Tranylcypromine hydrochloride

    Catalog No. A13358
    Quick View
    LSD1/BHC110 & MAO 抑制剂
    Tranylcypromine hydrochloride是一种非选择性的MAO-A/B抑制剂。 了解更多
  29. Safinamide

    Catalog No. A13294
    Quick View
    MAO-B 抑制剂
    Safinamide是一种高度选择性和可逆的B型单胺氧化酶(MAO-B)抑制剂,可增加新纹状体多巴胺的浓度。 了解更多
  30. RN-1 2HCl

    Catalog No. A14344
    Quick View
    MAO 抑制剂
    RN-1 2HCl对LSD1的选择性优于单胺氧化酶(MAO)-A和MAO-B(在辣根过氧化物酶偶联测定中,IC50值分别为70 nM,0.51和2.79 μM)。 了解更多

30 个项目

每页

设置升序顺序
Rewards