“neurotransmitter transporters”的搜索结果

19 个项目

每页

设置降序顺序
  1. GET73

    Catalog No. A22683
    Quick View
    neurotransmitter
    GET73 is a γ-hydroxybutyric acid (GHB) analog, a naturally occurring neurotransmitter. GET73 has anti-alcohol and anxiolytic properties. GET73 significantly affects glutamate transmission in the hippocampus. 了解更多
  2. L-aspartic Acid

    Catalog No. A17965
    Quick View
    neurotransmitter
    Aspartic acid is one of the non-essential amino acids commonly occurring in the L-form. It is found in animals and plants, especially in sugar cane and sugar beets. It may be a neurotransmitter. 了解更多
  3. Agmatine sulfate

    Catalog No. A20485
    Quick View
    NO synthase inhibitor
    Agmatine sulfate exerts modulatory action at multiple molecular targets, such as neurotransmitter systems, ion channels and nitric oxide synthesis. It is an endogenous agonist at imidazoline receptor and a NO synthase inhibitor. 了解更多
  4. DMP-543

    Catalog No. A19991
    Quick View
    KV7 channel blocker
    DMP-543 (XR-543) is a KV7 channel blocker, also acts as a potent neurotransmitter release enhancer. 了解更多
  5. (R)-Serine

    Catalog No. A17978
    Quick View
    NMDA glutamate receptor co-agonist
    (R)-Serine, an endogenous amino acid involved in glia-synapse interactions that has unique neurotransmitter characteristics, is a potent co-agonist at the NMDA glutamate receptor. 了解更多
  6. NMI 8739

    Catalog No. A12334
    Quick View
    dopamine D2 autoreceptor agonist
    NMI 8739 is a dopamine D2 autoreceptor agonist, which is an amine conjugate of the DHA carrier and the neurotransmitter dopamine. 了解更多
  7. Lonidamine

    Catalog No. A11633
    Quick View
    antitumor agent
    Lonidamine (AF-1890), an antitumor agent, is a hexokinase, mitochondrial pyruvate carrier (Ki 2.5 μM in isolated rat liver mitochondria) and plasma membrane monocarboxylate transporters inhibitor, which also inhibits mitochondrial complex II. 了解更多
  8. Radafaxine hydrochloride

    Catalog No. A20951
    Quick View
    dopamine transporter/norepinephrine transportertransporters inhibitor
    Radafaxine hydrochloride (GW-353162A) is a DAT (dopamine transporter) and NET(norepinephrine transporter) transporters inhibitor, and nAChR family modulator. 了解更多
  9. ITI214 free base

    Catalog No. A21947
    Quick View
    picomolar PDE1 inhibitor
    ITI-214 (free base) is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and against a panel of enzymes, receptors, transporters, and ion channels, exhibits potent PDE1 inhibitory activity (Ki = 58 pM). 了解更多
  10. Dasotraline hydrochloride

    Catalog No. A21684
    Quick View
    triple reuptake inhibitor
    Dasotraline hydrochloride (SEP-225289 hydrochloride) is a triple reuptake inhibitor that blocks dopamine, norepinephrine, and serotonin transporters with IC50 values of 4, 6, and 11 nM, respectively. 了解更多
  11. Dasotraline

    Catalog No. A21618
    Quick View
    triple reuptake inhibitor
    Dasotraline is a triple reuptake inhibitor that blocks dopamine, norepinephrine, and serotonin transporters with IC50 values of 4, 6, and 11 nM, respectively. 了解更多
  12. ITI214

    Catalog No. A21422
    Quick View
    PDE1 inhibitor
    ITI-214 is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and against a panel of enzymes, receptors, transporters, and ion channels, exhibits potent PDE1 inhibitory activity (Ki = 58 pM). 了解更多
  13. Uridine triphosphate

    Catalog No. A13317
    Quick View
    nucleotide
    Uridine triphosphate (UTP;Uridine 5'-triphosphate) is a nucleotide that regulates the functions of the pancreas in endocrine and exocrine secretion, proliferation, channels, transporters, and intracellular signaling under normal and disease states. 了解更多
  14. N-Dodecyl-β-D-maltoside

    Catalog No. A19128
    Quick View
    N-Dodecyl-β-D-maltoside (Lauryl Maltoside) is a derivatives of pyrene (Py), and it is a alkyl maltopyranoside detergent, especially in transporters and respiratory complexes. 了解更多
  15. BI01383298

    Catalog No. A18831
    Quick View
    SLC13A5 inhibitor
    BI01383298 is a potent inhibitor of SLC13A5, being selective over other family members and other transporters. 了解更多
  16. Bretylium tosylate

    Catalog No. A21798
    Quick View
    Bretylium (tosylate) is an inhibitor of the presynaptic release of vasoconstrictor neurotransmitters. 了解更多
  17. Droxidopa

    Catalog No. A21541
    Quick View
    Droxidopa(L-DOPS), the mixture of Droxidopa (w/w80%) and Pharmaceutical starch (w/w20%), acts as a prodrug to the neurotransmitters norepinephrine (noradrenaline) and epinephrine (adrenaline). 了解更多
  18. Ertugliflozin L-pyroglutamic acid

    Catalog No. A18054
    Quick View
    SGLT inhibitor
    Ertugliflozin pidolate belongs to the class of potent and selective inhibitors of the sodium-dependent glucose cotransporters (SGLT), more specifically the type 2 which is responsible for about 90% of the glucose reabsorption from glomerulus. 了解更多
  19. Harmaline

    Catalog No. A17416
    Quick View
    Harmaline is a psychoactive indole found naturally in certain plants. Its stimulating activities are achieved, in part, through inhibition of monoamine oxidases, thus increasing the levels of monoamine neurotransmitters (e.g., at 7-70 μM/kg in rats). Harmaline (30 mg/kg) induces tremor in mice through the N-methyl-D-aspartate (NMDA) receptor, at which harmaline may act as an inverse agonist. 了解更多

19 个项目

每页

设置降序顺序
Rewards