NMDA Receptors

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  1. Rislenemdaz

    Catalog No. A21907
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    NMDA receptor GluN2B antagonist
    Rislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively. 了解更多
  2. SDZ 220-581 hydrochloride, SDZ220-581, SDZ-220-581

    Catalog No. A21897
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    NMDA receptor antagonist
    SDZ 220-581 hydrochloride is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. 了解更多
  3. 7-Chlorokynurenic acid sodium salt

    Catalog No. A21879
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    NMDA receptor antagonist
    7-Chlorokynurenic acid sodium salt is a potent and selective antagonist of the glycine B coagonist site of the N-methyl-D-aspartate (NMDA) receptor (IC50=0.56 μM). 了解更多
  4. NMDA-IN-1

    Catalog No. A21419
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    NMDA antagonist
    NMDA-IN-1 is a potent and NR2B-selective NMDA antagonist with Ki of 0.85 nM. 了解更多
  5. Radiprodil

    Catalog No. A21193
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    NMDA NR2B antagonist
    Radiprodil (RGH-896) is an orally active and selective NMDA NR2B antagonist. A potential therapeutic agent in treatment of neuropathic pain and possibly other chronic pain conditions. 了解更多
  6. MDL 105519

    Catalog No. A21192
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    NMDA receptor antagonist
    MDL 105519 is a potent and selective antagonist of glycine binding to the NMDA receptor. 了解更多
  7. Transcrocetinate disodium

    Catalog No. A21051
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    NMDA receptor antagonist
    Transcrocetinate disodium, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity. 了解更多
  8. Ifenprodil tartrate

    Catalog No. A16583
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    NMDA receptor antagonist
    Ifenprodil tartrate is the atypical N-methyl-D-aspartate (NMDA) receptor antagonist, inhibits NMDA-induced currents at NR1A/NR2B receptors with high affinity (IC50 = 0.34 μM). 了解更多
  9. RPR104632

    Catalog No. A13385
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    NMDA receptor antagonist
    RPR104632 is a specific antagonist of NMDA receptor, with potent neuroprotective properties. 了解更多
  10. GV-196771A

    Catalog No. A13438
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    NMDA receptor antagonist
    GV-196771A is the sodium salt form of GV196771, is an NMDA receptor antagonist. 了解更多
  11. Sarcosine

    Catalog No. A16692
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    GlyT inhibitor/NMDA receptor
    Sarcosine is a glycine transporter type 1 (GlyT) inhibitor and an N-methyl-D-aspartate (NMDA) receptor co-agonist at the glycine binding site. 了解更多
  12. Eliprodil

    Catalog No. A12946
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    NMDA 拮抗剂
    Eliprodil是一种非竞争性NR2B-NMDA受体拮抗剂(IC50 = 1 uM),对含NR2A和NR2C的受体效力较低(IC50> 100 uM)。 了解更多
  13. CGS19755

    Catalog No. A15791
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    NMDA 拮抗剂
    CGS 19755(顺式-4-膦酰基甲基-2-哌啶羧酸)是一种有效的立体定向抑制剂,由N-甲基-D-天冬氨酸(NMDA)诱发,但不是由KCl诱发的[3H]乙酰胆碱释放大鼠纹状体的切片。 了解更多
  14. (+)-MK 801 Maleate

    Catalog No. A12761
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    NMDA receptor 拮抗剂
    (+)-MK 801 Maleate是NMDA的有效拮抗剂,Ki值为30.5nM。 了解更多
  15. L-701324

    Catalog No. A15522
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    NMDA/glycine receptor 拮抗剂
    L-701324是一种活性且长效的抗惊厥药,对NMDA受体上的甘氨酸位点具有高亲和力和选择性。 了解更多
  16. Flupirtine maleate

    Catalog No. A10251
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    NMDA 拮抗剂
    Flupirtine maleate是Flupirine的盐形式,是一种非阿片类中枢性镇痛药,是一种选择性的神经元钾离子通道开放剂,也具有NMDA受体拮抗剂特性。 了解更多
  17. TCN 201

    Catalog No. A11947
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    NMDA Receptor 拮抗剂
    TCN 201是对NR1/NR2A相对于含NR1/NR2B的受体具有选择性的NMDA受体拮抗剂。 了解更多
  18. SDZ 220-581

    Catalog No. A12426
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    NMDA receptor 拮抗剂
    SDZ 220-581是一种竞争性NMDA受体拮抗剂(pKi = 7.7)。 了解更多
  19. NMDA

    Catalog No. A12751
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    NMDA receptor 激动剂
    NMDA是一种原型NMDA受体激动剂。 了解更多
  20. DNQX

    Catalog No. A13882
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    NMDA receptor 拮抗剂
    DNQX是一种非N-甲基-D-天冬氨酸(非NMDA)受体复合物拮抗剂。 了解更多
  21. SDZ 220-581 Ammonium salt

    Catalog No. A15235
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    NMDA receptor 拮抗剂
    SDZ 220-581 Ammonium salt是NMDA谷氨酸受体亚型(pKi = 7.7)的有效竞争性拮抗剂。 了解更多
  22. (-)-MK 801 maleate

    Catalog No. A13435
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    NMDA receptor 拮抗剂.
    (-)-MK 801 maleate是一种有效的、选择性的、非竞争性的NMDA受体拮抗剂。它通过与NMDA相关离子通道内的一个位点结合而起作用。 了解更多
  23. Memantine hydrochloride

    Catalog No. A11708
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    NMDA receptor 拮抗剂
    Memantine hydrochloride是nmda受体的拮抗剂,与离子通道位点结合。它还是CYP2B6和CYP2D6抑制剂,作用于重组CYP2B6和CYP2D6,Ki分别为0.51 nM和94.9 μM。它被用于治疗帕金森综合征。 了解更多
  24. Orphenadrine citrate

    Catalog No. A11712
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    NMDA receptor 拮抗剂
    Orphenadrine柠檬酸盐是NMDA受体拮抗剂,Ki为6.0μM,还是HERG钾离子通道阻断剂。 了解更多
  25. CIQ

    Catalog No. A15523
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    NMDA receptors Potentiator
    CIQ是包含NR2C或NR2D亚基的NMDA受体的亚基选择性增强剂。 了解更多
  26. Felbamate

    Catalog No. A11862
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    Felbamate是NMDA相关甘氨酸结合位点的拮抗剂。 了解更多
  27. Ibotenic Acid

    Catalog No. A14006
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    NMDA& mGlu receptor 激动剂
    Ibotenic Acid是最初从鹅膏菌属物种中分离出来的一种神经兴奋性氨基酸,它起着NMDA和代谢型谷氨酸受体激动剂的作用。 了解更多
  28. MDL 29951

    Catalog No. A13729
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    NMDA receptor 拮抗剂
    MDL-29951是在体外和体内均能激活NMDA受体的新型甘氨酸拮抗剂(Ki = 0.14 mM,[3H]甘氨酸结合)。 了解更多
  29. GLYX-13 (Rapastinel)

    Catalog No. A13576
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    NMDAR modulator
    GLYX-13 (Rapastinel)是NMDA受体甘氨酸位点的选择性弱部分激动剂。 了解更多
  30. NVP-AAM077 Tetrasodium Hydrate (PEAQX)

    Catalog No. A14071
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    NMDA receptors 拮抗剂
    NVP-AAM077抑制成年小鼠在脑室下区域和齿状回中的祖细胞增殖,并降低了齿状回中的新生细胞的存活。 了解更多
  31. ARL-15896

    Catalog No. A13858
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    NMDA receptor ion channel 拮抗剂
    ARL-15896是新型的N-甲基-D-天冬氨酸受体离子通道拮抗剂。 了解更多
  32. GNE 0723

    Catalog No. A12757
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    NMDAR modulator
    GNE 0723 is a brain permeable positive allosteric modulator of NMDAR, with an EC50 of 21 nM for GluN2A, 7.4 and 6.2 μM for GluN2C and GluN2D, respectively. 了解更多
  33. Glycine

    Catalog No. A17936
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    NMDA antagonist
    AZD-4282, also known as aminoacetic acid and glycine, is a N-methyl-D-aspartate (NMDA) receptor antagonist potentially for the treatment of neuropathic pain. 了解更多
  34. Mephenesin

    Catalog No. A17493
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    NMDA receptor antagonist
    Mephenesin is an NMDA receptor antagonist, is a centrally acting muscle relaxant. 了解更多
  35. Neu-2000

    Catalog No. A17033
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    NMDA receptor 拮抗剂
    Neu-2000是可能用于治疗中风的NMDA受体拮抗剂。 了解更多
  36. D-AP5

    Catalog No. A17044
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    NMDA 拮抗剂
    D-AP5是一种选择性的N-甲基-D-天冬氨酸(NMDA)受体拮抗剂,可竞争性抑制NMDA受体的谷氨酸结合位点。 了解更多
  37. 7CKA

    Catalog No. A17070
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    NMDA receptor 拮抗剂
    7CKA是在甘氨酸位点起作用的NMDA受体拮抗剂。 了解更多
  38. Ro 25-6981 maleate

    Catalog No. A13144
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    NMDA receptors Blocker
    Ro 25-6981是N-甲基-D-天冬氨酸(NMDA)受体的高亲和力,强效选择性阻断剂。 了解更多
  39. CNQX

    Catalog No. A16109
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    AMPA/kainate 拮抗剂
    CNQX是一种竞争性的非NMDA谷氨酸受体拮抗剂(AMPA和海藻酸酯受体的IC50分别为0.3和1.5 uM,而NMDA受体的IC50 = 25 uM)。 了解更多
  40. RO 25-6981 maleate

    Catalog No. A16083
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    NMDA receptors blocker
    RO 25-6981 maleate是含有NR2B亚基的NMDA受体的强效和选择性活性依赖性阻断剂。克隆的受体亚基组合NR1C/NR2B和NR1C/NR2A的IC50值分别为0.009和52 uM。 了解更多

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