PD 151746

目录号: A14245

Calpain 抑制剂

PD 151746

PD 151746 Chemical Structure

CAS NO. 179461-52-0

PD 151746是一种选择性的,细胞可渗透的钙蛋白酶抑制剂,对μ-钙蛋白酶的Ki值为0.26 uM,选择性是m-钙蛋白酶的20倍。

库存: 现货

规格 价格 数量
10 mg
¥ 900.00
25 mg
¥ 1,800.00
50 mg
¥ 3,000.00
10mM * 1mL in DMSO
¥ 950.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

PD 151746是一种选择性的,细胞可渗透的钙蛋白酶抑制剂,对μ-钙蛋白酶的Ki值为0.26 uM,选择性是m-钙蛋白酶的20倍。
靶点信息
μ-Calpain m-calpain
260 nM5.33 μM
In vitro DMSO 40 mg/mL (168.6 mM)
Water Insoluble
Ethanol 40 mg/mL (168.6 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 42.15 mL 210.75 mL 421.5 mL
0.5 mM 8.43 mL 42.15 mL 84.3 mL
1 mM 4.21 mL 21.07 mL 42.15 mL
5 mM 0.84 mL 4.21 mL 8.43 mL

*The above data is based on the productmolecular weight 237.25. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A14245
作用机制 Inhibitor (抑制剂)
M. Wt 237.25
Formula C11H8FNO2S
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 179461-52-0
Synonyms PD-151746,PD151746
SMILES C1=CC2=C(C=C1F)C(=CN2)/C=C(/C(=O)O)\S

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