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PD153035 (HCl salt)是EGFR酪氨酸激酶活性的极其有效和特异的抑制剂。
靶点信息
| EGFR (Cell-free assay) | EGFR (Cell-free assay) | |||
| 5.2 pM(Ki) | 5.2 pM(Ki) |
| In vitro (25°C) | DMSO | 0.46 mg/mL (1.16 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
| In vivo | 30% propylene glycol, 5% Tween 80, 65% D5W | 28 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 25.21 mL | 126.04 mL | 252.08 mL |
| 0.5 mM | 5.04 mL | 25.21 mL | 50.42 mL |
| 1 mM | 2.52 mL | 12.6 mL | 25.21 mL |
| 5 mM | 0.5 mL | 2.52 mL | 5.04 mL |
*The above data is based on the productmolecular weight 396.7 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| 目录号 | A10702 |
|---|---|
| 作用机制 | Inhibitor (抑制剂) |
| M. Wt | 396.7 |
| Formula | C16H14BrN3O2.HCl |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
| CAS No. | 183322-45-4 |
| Synonyms | ZM 252868, AG 1517, Tyrphostin AG 1517, SU 5271, PD-153035 |
| SMILES | COC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC(=CC=C3)Br)OC.Cl |
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