PI-103 Hydrochloride

目录号: A15212

PI3K 抑制剂

PI-103 Hydrochloride

PI-103 Hydrochloride Chemical Structure

CAS NO. 371935-79-4

PI-103 Hydrochloride是对重组PI3K亚型p110alpha(IC50 = 2 nM),p110beta(IC50 = 3 nM),p110delta(IC50 = 3 nM)和p110gamma(IC50 = 15 nM)具有低IC50值的有效抑制剂,对mTOR的效力较低/DNA-PK,IC50为30 nM/23 nM。

库存: 现货

规格 价格 数量
10 mg
¥ 650.00
50 mg
¥ 2,000.00
100 mg
¥ 3,600.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

PI-103 Hydrochloride是对重组PI3K亚型p110alpha(IC50 = 2 nM),p110beta(IC50 = 3 nM),p110delta(IC50 = 3 nM)和p110gamma(IC50 = 15 nM)具有低IC50值的有效抑制剂,对mTOR的效力较低/DNA-PK,IC50为30 nM/23 nM。
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.99 mL 129.93 mL 259.86 mL
0.5 mM 5.2 mL 25.99 mL 51.97 mL
1 mM 2.6 mL 12.99 mL 25.99 mL
5 mM 0.52 mL 2.6 mL 5.2 mL

*The above data is based on the productmolecular weight 384.82. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A15212
作用机制 Inhibitor (抑制剂)
M. Wt 384.82
Formula C19H17ClN4O3
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 371935-79-4
Synonyms PI 103 hydrochloride, PI103 hydrochloride
SMILES C1COCCN1C2=NC(=NC3=C2OC4=C3C=CC=N4)C5=CC(=CC=C5)O.Cl

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