RQ-00203078

目录号: A15830

TRPM8 拮抗剂

RQ-00203078

RQ-00203078 Chemical Structure

CAS NO. 1254205-52-1

RQ-00203078是一种高度选择性,有效且可口服的TRPM8拮抗剂(大鼠和人类通道的IC50值分别为5.3和8.3 nM),对TRPM8的选择性是TRPV4,TRPV1和TRPA1的> 350倍。

库存: 现货

规格 价格 数量
10 mg
¥ 1,200.00
25 mg
¥ 2,500.00
50 mg
¥ 4,500.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

RQ-00203078是一种高度选择性,有效且可口服的TRPM8拮抗剂(大鼠和人类通道的IC50值分别为5.3和8.3 nM),对TRPM8的选择性是TRPV4,TRPV1和TRPA1的> 350倍。
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.02 mL 90.11 mL 180.23 mL
0.5 mM 3.6 mL 18.02 mL 36.05 mL
1 mM 1.8 mL 9.01 mL 18.02 mL
5 mM 0.36 mL 1.8 mL 3.6 mL

*The above data is based on the productmolecular weight 554.85. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A15830
作用机制 Antagonist (拮抗剂)
M. Wt 554.85
Formula C21H13ClF6N2O5S
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 1254205-52-1
Synonyms RQ 00203078, RQ00203078
SMILES ClC1=C(N(CC2=CC=C(OC(F)(F)F)C=C2)S(C3=CC=C(C(O)=O)C=C3)(=O)=O)N=CC(C(F)(F)F)=C1

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