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Santacruzamate A

Santacruzamate A

Name: Santacruzamate A
SKU: A14236

目录号: A14236

HDAC 抑制剂

Santacruzamate A Chemical Structure

CAS NO. 1477949-42-0

Santacruzamate A (CAY10683)是一种有效的选择性HDAC抑制剂，对HDAC2的IC50为119 pM，选择性是其他HDAC的3600倍以上。

库存：现货

规格	价格	数量
25 mg	￥ 1,500.00
50 mg	￥ 2,500.00
100 mg	￥ 4,000.00
10mM * 1mL in DMSO	￥ 550.00

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生物活性

Santacruzamate A (CAY10683)是一种有效的选择性HDAC抑制剂，对HDAC2的IC50为119 pM，选择性是其他HDAC的3600倍以上。

靶点信息

HDAC2	HDAC6	HDAC4
119 pM	434 nM	>1000 nM

溶解度 *

In vitro (25°C)	DMSO	47 mg/mL (168.85 mM)
	Water	Insoluble
	Ethanol	47 mg/mL (168.85 mM)
In vivo	5%DMSO+30%PEG300+5%TW80+H2O	9 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	35.93 mL	179.63 mL	359.26 mL
0.5 mM	7.19 mL	35.93 mL	71.85 mL
1 mM	3.59 mL	17.96 mL	35.93 mL
5 mM	0.72 mL	3.59 mL	7.19 mL

*The above data is based on the productmolecular weight 278.35. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A14236
作用机制	Inhibitor (抑制剂)
M. Wt	278.35
Formula	C15H22N2O3
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1477949-42-0
Synonyms	CAY10683
SMILES	CCOC(=O)NCCCC(=O)NCCC1=CC=CC=C1