Sigma receptor

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  1. E1R

    Catalog No. A18825
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    sigma-1 receptors modulator
    E1R is a novel positive allosteric modulator of sigma-1 receptors. 了解更多
  2. Sigma-1 receptor antagonist 2

    Catalog No. A18504
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    sigma 1 receptor antagonist
    Sigma-1 receptor antagonist 2 is a potent and selective sigma 1 receptor (??1 R) antagonist with Kis of 3.88 and 1288 nM for ??1 and ??2 receptor, respectively. 了解更多
  3. Sigma-1 receptor antagonist 3

    Catalog No. A18501
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    Sigma-1 receptor antagonist
    Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (??1) receptor antagonist with a Ki of 1.14 nM. 了解更多
  4. Cutamesine

    Catalog No. A21152
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    sigma 1 receptor agonist
    Cutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(??1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4??1.9 nM); 100-fold less affinity for the sigma 2 receptor. 了解更多
  5. Ditolylguanidine

    Catalog No. A21268
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    Sigma receptor agonist
    Ditolylguanidine (1,3-Di-o-tolylguanidine) is an agonist of sigma receptor (??1/??2 receptor). 了解更多
  6. Siramesine Hydrochloride

    Catalog No. A12479
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    Sigma-2 receptor 激动剂
    Siramesine Hydrochloride是一种选择性sigma-2受体激动剂,已被证明可触发癌细胞的细胞死亡并在体内表现出强大的抗癌活性。 了解更多
  7. S1RA (E-52862)

    Catalog No. A12504
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    sigma-1 receptor 拮抗剂
    S1RA是一种选择性sigma-1受体拮抗剂,据报道其结合亲和力为Ki = 17.0±7.0 nM,对sigma-2受体具有选择性,并且对其他170种受体,酶,转运蛋白和离子通道具有选择性。 了解更多
  8. Siramesine

    Catalog No. A13036
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    Sigma-2 receptor 激动剂
    Siramesine是一种溶酶体去污剂,诱导细胞保护性自噬体积累。 了解更多
  9. UMB24

    Catalog No. A13513
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    Sigma2 拮抗剂
    UMB24是推定的sigma2优选拮抗剂。 了解更多
  10. BD-1047 2HBr

    Catalog No. A13196
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    Sigma-1 拮抗剂
    BD-1047 2HBr是sigma受体的选择性功能拮抗剂,在动物模型中显示出抗精神病活性,可预测精神分裂症的疗效。 了解更多
  11. SA-4503

    Catalog No. A12984
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    sigma 1 receptor(σ1R) 激动剂
    SA4503是选择性sigma 1受体(σ1R)激动剂;对(+)-[3H]喷他佐辛标记的sigma 1受体亚型具有高亲和力(IC50 = 17.4+/-1.9 nM);对sigma 2受体的亲和力低100倍。 了解更多
  12. Glycerol phenylbutyrate

    Catalog No. A18201
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    sigma-2 (σ2) receptor ligand
    Glycerol phenylbutyrate is a sigma-2 (σ2) receptor ligand, with a pKi of 8.02. 了解更多
  13. 4-IBP

    Catalog No. A12314
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    σ1 激动剂
    4-IBP is a selective ??1 agonist with a high level of affinity for the ??1 receptor (Ki = 1.7 nM) and a moderate affinity for the ??2 receptor (Ki = 25.2 nM) . 了解更多

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