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SU9516

促销

CDK2 抑制剂

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产品目录号: A14318

库存状态:中国现货中国现货

产品名 目录号 价格 数量
SU9516 10mg A14318-10
¥ 900.00
SU9516 25mg A14318-25
¥ 2,000.00
SU9516 50mg A14318-50
¥ 3,200.00
SU9516 10mM * 1mL in DMSO A14318-10mM-D
¥ 750.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

SU9516 is a potent, selective cdk2 inhibitor. It inhibits pRb phosphorylation causing enhanced pRB/E2F complex formation and induces G1 and G2-M cell cycle arrest.

SU9516

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Chemical Information

目录号 A14318
Mechanism of action Inhibitor
分子量 241.25
化学分子式 C13H11N3O2
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 377090-84-1
Synonyms SU 9516, SU-9516
SMILES code COC1=CC\2=C(C=C1)NC(=O)/C2=C\C3=CN=CN3
化学名称 (Z)-1,3-Dihydro-3-(1H-imidazol-4-ylmethylene)-5-methoxy-2H-indol-2-one

Biological Activity

Description
SU9516 is a potent, selective cdk2 inhibitor. It inhibits pRb phosphorylation causing enhanced pRB/E2F complex formation and induces G1 and G2-M cell cycle arrest.
Targets
Target Value
CDK2IC50: 22nM
CDK1IC50: 40nM
CDK4IC50: 200nM
PKCIC50: >10μM
p38IC50: >10μM
PDGFRIC50: 18μM
EGFRIC50: >100μM

Solubility

Solubility (25°C)* In vitro DMSO 48 mg/mL (198.96 mM)
Water <1 mg/mL (<1 mM)
Ethanol 12 mg/mL heating (49.74 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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