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Tubastatin A HCl是一种有效的选择性HDAC6抑制剂，在无细胞试验中IC50为15 nM。它对除HDAC8（57倍）以外的所有其他同工酶（1000倍）具有选择性。
Targets
| Target | Value |
|---|---|
| HDAC6 | IC50: 15nM |
| HDAC8 | IC50: 854nM |
| HDAC1 | IC50: 16.4μM |
| HDAC2 | IC50: >30μM |
| HDAC3 | IC50: >30μM |
| HDAC4 | IC50: >30μM |
| HDAC5 | IC50: >30μM |
| HDAC7 | IC50: >30μM |
| HDAC9 | IC50: >30μM |
| HDAC10 | IC50: >30μM |
| HDAC11 | IC50: >30μM |
| In vitro (25°C) | DMSO | 67 mg/mL (180.17 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
| In vivo | 5%DMSO+40%PEG300+5%Tween80+50%ddH2O | 5.2 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 26.89 mL | 134.44 mL | 268.89 mL |
| 0.5 mM | 5.38 mL | 26.89 mL | 53.78 mL |
| 1 mM | 2.69 mL | 13.44 mL | 26.89 mL |
| 5 mM | 0.54 mL | 2.69 mL | 5.38 mL |
*The above data is based on the productmolecular weight 371.9 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| 目录号 | A11042 |
|---|---|
| 作用机制 | Inhibitor (抑制剂) |
| M. Wt | 371.9 |
| Formula | C20H21N3O2.HCl |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
| CAS No. | 1310693-92-5, 1239262-52-2 |
| SMILES | CN1CCC2=C(C1)C3=CC=CC=C3N2CC4=CC=C(C=C4)C(=O)NO.Cl |
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