“2c i hcl”的搜索结果

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  1. P005672 HCl (Sarecycline HCl)

    Catalog No. A11283
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    P005672 HCl (Sarecycline HCl)是用于抗菌/消炎痤疮治疗的II期药物。 了解更多
  2. AMG-073 HCl (Cinacalcet HCl)

    Catalog No. A10219
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    CaSR activator
    AMG-073 HCl(Cinacalcet HCl)是一种用于治疗甲状旁腺功能亢进的化合物,称为拟钙剂,通过增加甲状旁腺钙敏感受体(CaR)对细胞外钙的敏感性来减少甲状旁腺激素(PTH)的合成和分泌 。 了解更多
  3. TP0427736 HCl

    Catalog No. A22382
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    ALK5 kinase activity inhibitor
    TP0427736 is a potent inhibitor of ALK5 kinase activity with an IC50 of 2.72 nM and this effect is 300-fold higher than the inhibitory effect on ALK3 (IC50 = 836 nM for ALK3). It also inhibits Smad2/3 phosphorylation in A549 cells induced by TGF-β1 with an IC50 value of 8.68 nM. 了解更多
  4. SB203186 HCl

    Catalog No. A22523
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    5-HT4 receptor antagonist
    SB203186 is potent 5-HT4 receptor antagonist. 了解更多
  5. Anlotinib HCl

    Catalog No. A17076
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    RTK 抑制剂
    Anlotinib HCl,也称为AL3818,是一种受体酪氨酸激酶(RTK)抑制剂,具有潜在的抗肿瘤和抗血管生成活性。 了解更多
  6. MLN4924 (HCL Salt)

    Catalog No. A11499
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    NAE 抑制剂
    MLN4924 (HCL Salt)是一种有效,选择性的 NEDD8 活化酶 (NEDD8-activating enzyme) 抑制剂。 了解更多
  7. 17-DMAG HCl (Alvespimycin)

    Catalog No. A10011
    Hsp90 抑制剂
    17-DMAG HCl (Alvespimycin)是17-AAG和格尔德霉素的水溶性类似物,与Hsp90的ATP结合位点结合并抑制其伴侣活性。显示出比17-AAG更有效的抗肿瘤活性。 了解更多
  8. CFI-400437 HCl

    Catalog No. A22463
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    CFI-400437 is a potent and selective inhibitor of polo-like kinase 4 (PLK4). 了解更多
  9. Sisunatovir HCl

    Catalog No. A22476
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    Sisunatovir, also known as RV521, is a highly potent fusion inhibitor with efficacy against a panel of clinical isolates of RSV-A and RSV-B viruses. 了解更多
  10. Caroverine HCl

    Catalog No. A22495
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    Caroverine hydrochloride is a potent, competitive and reversible antagonist of NMDA and AMPA glutamate receptor. Caroverine hydrochloride is also an antioxidant and calcium-blocking agent that exhibits vasorelaxant action. Caroverine hydrochloride can be used for the research of inner ear tinnitus. 了解更多
  11. ML095 HCl

    Catalog No. A22545
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    PLAP inhibitor
    ML-095 is an inhibitor of PLAP (IC50 = 3.7 μM) that demonstrates high selectivity against the related alkaline phosphatases, TNAP and IAP (IC50s > 100 μM). 了解更多
  12. SEP-363856 HCl

    Catalog No. A22555
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    SEP-363856, also known as SEP-856, is an orally active and CNS active psychotropic agent. 了解更多
  13. LM11A-31 HCl

    Catalog No. A22564
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    p75NTR ligand
    LM11A-31 is a small-molecule p75NTR modulator and proNGF antagonist. 了解更多
  14. SEL120-34A HCl

    Catalog No. A21485
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    CDK8 inhibitor
    SEL120-34A HCl is a potent, selective, orally available, ATP-competitive CDK8 inhibitor, with IC50s of 4.4 nM and 10.4 nM for CDK8/CycC and CDK19/CycC, respectively, with antitumor activity. 了解更多
  15. Glucagon HCl

    Catalog No. A17906
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    Glucagon is a peptide hormone, produced by alpha cells of the pancreas. It works to raise the concentration of glucose in the bloodstream. Its effect is opposite that of insulin, which lowers the glucose. 了解更多
  16. Methoxamine HCl

    Catalog No. A17365
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    alpha-1 adrenergic agonist
    Methoxamine Hydrochloride is an alpha-1 adrenergic agonist that causes prolonged peripheral vasoconstriction. 了解更多
  17. ICEC0942 HCl

    Catalog No. A16903
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    CDK7 抑制剂
    ICEC0942 HCl,也称为CT7001,是CDK7的口服生物利用选择性抑制剂。它选择性抑制CDK7,IC50为40nM。CDK1,CDK2,CDK5和CDK9的IC50值分别高45倍,15倍,230倍和30倍。 了解更多
  18. SB399885 HCl

    Catalog No. A16971
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    SR-6 拮抗剂
    SB 399885 hydrochloride是一种有效的,脑渗透剂和口服活性的SR-6拮抗剂。它对SR-6的选择性比其他血清素受体高200倍(对于人类重组,天然大鼠和天然人类SR-6受体,pKi值分别为9.11、8.81和9.02)。 了解更多
  19. MC 70 HCl

    Catalog No. A16080
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    P-gp 抑制剂
    MC 70 HCl是有效的P-gp抑制剂(EC50 = 0.69 uM)。 了解更多
  20. L-778123 HCl

    Catalog No. A15796
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    FPTase 抑制剂
    L-778123 hydrochloride是FPTase和GGPTase-I双重抑制剂,在酶抑制测定中IC50为2 nM和98 nM。 了解更多
  21. Medetomidine HCl

    Catalog No. A13775
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    adrenergic alpha-2 receptor 激动剂
    Medetomidine Hydrochloride是一种肾上腺素α2-受体激动剂,Ki为1.08 nM,比作用于α1-adrenoceptor选择性高1620倍。由于其镇痛和镇静作用而被用于兽医学。 了解更多
  22. Blasticidin S HCl

    Catalog No. A14212
    Blasticidin S HCl是一种分离自gistreochromogenes链霉菌的核苷抗生素,并充当DNA和蛋白质合成抑制剂。 了解更多
  23. Deltarasin HCl

    Catalog No. A13722
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    PDE-KRAS 抑制剂
    Deltarasin HCl是一种新型的抑制KRASPDEδ相互作用从而破坏致癌性KRAS信号的小分子。 了解更多
  24. PRT062607 HCL

    Catalog No. A12731
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    Syk 抑制剂
    PRT2607,也称为PRT062607,P505-15和BIIB057,是一种新型,高度选择性且口服可生物利用的小分子SYK抑制剂(SYK IC(50)= 1 nM),具有至少80倍的抗SYK活性 大于对其他激酶的亲和力。 了解更多
  25. Ondansetron HCl (GR 38032F)

    Catalog No. A10674
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    5-HT Receptors 拮抗剂
    Ondansetron HCl (GR 38032F)是5-羟色胺5-HT3受体拮抗剂,主要用作止吐药,通常在化疗后用于治疗恶心和呕吐。 了解更多
  26. Articaine HCl

    Catalog No. A11808
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    Articaine HCl是一种牙科局部麻醉剂,含有一个附加的酯基,该酯基可以被血液和组织中的酯酶代谢掉。 了解更多
  27. Fexofenadine HCl

    Catalog No. A11859
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    COX 抑制剂/histamine H1 receptor 激动剂
    Fexofenadine Hydrochloride是一种抗组胺药,可抑制Cox-1,Cox-2,并且是组胺H1受体激动剂,IC50为246 nM。 了解更多
  28. Ivabradine HCl (Procoralan)

    Catalog No. A11868
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    Ivabradine Hydrochloride,也称为S-16257,是缓动剂伊伐布雷定的盐酸盐制剂。 了解更多
  29. Adrenalone HCl

    Catalog No. A11807
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    adrenergic 激动剂
    Adrenalone HCl是一种肾上腺素能激动剂,用作局部血管收缩药和止血药,主要作用于α-1肾上腺素能受体。 了解更多
  30. Nebivolol HCl

    Catalog No. A10630
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    Nebivolol hydrochloride是β1-肾上腺素受体的高度选择性拮抗剂(Ki = 0.88 nM,β2-肾上腺素受体Ki = 48 nM)。 了解更多
  31. Anamorelin HCl

    Catalog No. A12345
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    Anamorelin HCl目前正在开发中,是口服活性的饥饿素受体(ghrelin receptor)激动剂。用于治疗与恶病质/厌食症相关的非小肺癌。 了解更多
  32. Paroxetine HCl

    Catalog No. A11904
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    Paroxetine HCl是SSRI类型的抗抑郁药。 了解更多
  33. CGS 21680 HCl Hydrate

    Catalog No. A11619
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    Adenosine A2A Receptor 激动剂
    CGS 21680 HCl是一种特定的腺苷A2A亚型受体激动剂。 了解更多
  34. AT7519 HCl

    Catalog No. A11313
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    CDK 抑制剂
    AT7519是多种细胞周期蛋白依赖性激酶(CDK)的抑制剂,可导致细胞周期停滞,诱导细胞凋亡和抑制肿瘤细胞增殖。 了解更多
  35. Alfuzosin HCl

    Catalog No. A10052
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    Alfuzosin HCl是用于治疗良性前列腺增生(BPH)的α1受体拮抗剂。 它通过放松前列腺和膀胱颈的肌肉来起作用,使其更容易排尿。 了解更多
  36. Idarubicin HCl

    Catalog No. A10465
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    Topoisomerase 抑制剂
    Idarubicin HCl是蒽环类抗生素,是一种比柔红霉素具有更高DNA结合能力和更大细胞毒性的抗白血病药物。 了解更多
  37. GW3965 HCl

    Catalog No. A11204
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    LXR-like receptors 激动剂
    GW3965 HCl是一种选择性的口服活性肝X受体(LXR)完全激动剂。 了解更多
  38. Cerubidine (Daunorubicin HCl, Rubidomycin HCl)

    Catalog No. A10194
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    Topoisomerase 抑制剂
    Cerubidine (Daunorubicin HCl,Rubidomycin HCl)通过插入和抑制大分子生物合成与DNA相互作用。这抑制了拓扑异构酶II的进程,该酶使DNA中的超螺旋松弛以进行转录。 了解更多
  39. ADL5859 HCl

    Catalog No. A11072
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    Opioid Receptor 激动剂
    ADL5859 HCl是高效的选择性δ阿片受体激动剂,Ki值为0.84 nM,ED50值为20 nM。 了解更多
  40. Topotecan HCl (Hycamtin)

    Catalog No. A10939
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    DNA topoisomerase I 抑制剂
    Topotecan HCl (Hycamtin)是一种化学治疗剂,是拓扑异构酶抑制剂。 了解更多
  41. Flavopiridol HCl

    Catalog No. A11045
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    CDK 抑制剂
    Flavopiridol HCl是细胞周期蛋白依赖性激酶的抑制剂。(-)-顺式形式诱导特定肿瘤细胞的凋亡。 了解更多
  42. Gemcitabine HCl (Gemzar)

    Catalog No. A10423
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    DNA/RNA Synthesis 抑制剂
    Gemcitabine HCl (Gemzar)是一种DNA synthesis抑制剂,作用于PANC1,MIAPaCa2,BxPC3和Capan2细胞,通过在癌细胞dna复制过程中取代核酸的一个组成部分,防止肿瘤生长。 了解更多
  43. PD 0332991 HCl (Palbociclib)

    Catalog No. A10701
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    CDK 4/6 抑制剂
    PD 0332991 HCl (Palbociclib)是一种高度选择性的CDK4/6抑制剂,它对CDK1/2/5,EGFR,FGFR,PDGFR,InsR等没有抑制活性,具有潜在的抗肿瘤活性。 了解更多
  44. Prexasertib HCl

    Catalog No. A22156
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    ATP-competitive CHK1 inhibitor
    Prexasertib (LY2606368) is an ATP-competitive CHK1 inhibitor with a Ki value of 0.9 nmol/L. For CHK2 and RSK, its IC50 values are 8 nM and 9 nM respectively in cell-free assay. 了解更多
  45. SEL24-B489 HCl

    Catalog No. A22203
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    pan-PIM/FLT3 inhibitor
    SEL24-B489 HCl is a potent, dual pan-PIM/FLT3 inhibitor. 了解更多
  46. UK-371804 HCl

    Catalog No. A22379
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    uPA inhibitor
    UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin). 了解更多
  47. AVN-101 HCl

    Catalog No. A22498
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    5-HT7 receptor antagonist
    AVN-101 is a very potent 5-HT7 receptor antagonist, with slightly lesser potency toward 5-HT6, 5-HT2A, and 5HT-2C receptors. It is a milti-target drug candidate for the treatment of CNS disorders. 了解更多
  48. Varenicline HCl

    Catalog No. A22519
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    Varenicline is a nicotinic receptor partial agonist. 了解更多
  49. MK-212 HCl

    Catalog No. A22531
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    MK 212 hydrochloride is a 5-HT receptor agonist; displays selectivity for 5-HT2C over 5-HT2A (IC50 values are 0.028 and 0.42 μM for human 5-HT2C and 5-HT2A receptors expressed in HEK293 cells respectively). 了解更多
  50. Acecainide HCl

    Catalog No. A22660
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    Class III antiarrhythmic agent
    Acecainide, also known as N-acetylprocainamide and ASL 601, is the N-acetylated metabolite of procainamide. Acecainide is a Class III antiarrhythmic agent. It can be given either intravenously or orally, and is eliminated primarily by renal excretion. 了解更多

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