Adrenergic Receptors

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  1. Norepinephrine

    Catalog No. A11306
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    β1-selective adrenergic receptor agonist
    Norepinephrine (Levarterenol; L-Noradrenaline) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多
  2. AGN 192836

    Catalog No. A13013
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    α2 adrenergic agonist
    AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. 了解更多
  3. β3-AR agonist 1

    Catalog No. A12777
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    β3-adrenergic receptor agonist
    β3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). 了解更多
  4. Norepinephrine hydrochloride

    Catalog No. A21605
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    β1-selective adrenergic receptor agonist
    Norepinephrine hydrochloride (Levarterenol hydrochloride; L-Noradrenaline hydrochloride) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多
  5. Synephrine (Oxedrine)

    Catalog No. A10882
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    Adrenergic Receptor 激动剂
    Synephrine (Oxedrine)是一种通常用于减肥的胺化合物。 了解更多
  6. Salbutamol sulfate (Albuterol)

    Catalog No. A10819
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    Adrenergic Receptor 激动剂
    Salbutamol sulfate (Albuterol)是一种短效β2肾上腺素能受体激动剂。 了解更多
  7. Phenylephrine HCl

    Catalog No. A11666
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    α1-adrenergic receptor 激动剂
    Phenylephrine HCl是一种选择性的α1肾上腺素能受体激动剂,主要用作减充血剂,扩张瞳孔和增加血压的药物。 了解更多
  8. Isoprenaline HCl

    Catalog No. A10484
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    β adrenoceptor 激动剂
    Isoprenaline HCl或isoproterenol是非选择性β肾上腺素能激动剂,在结构上类似于肾上腺素。 了解更多
  9. Detomidine hydrochloride

    Catalog No. A10298
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    Adrenergic Receptor 激动剂
    Detomidine hydrochloride是具有镇痛作用的镇静剂。α2-肾上腺素能激动剂产生剂量依赖性的镇静和镇痛作用,并通过激活α2儿茶酚胺受体介导,从而引起负反馈反应,从而减少兴奋性神经递质的产生。 了解更多
  10. Clonidine hydrochloride

    Catalog No. A10232
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    Alpha adrenergic 激动剂
    Clonidine hydrochloride被归类为中枢作用的α肾上腺素能激动剂。Clonidine主要作为咪唑啉受体激动剂。 了解更多
  11. Dobutamine hydrochloride

    Catalog No. A10325
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    Adrenoceptors 激动剂
    Dobutamine hydrochloride是一种直接作用剂,其主要活性来自刺激心脏的β1肾上腺素能受体,增加收缩力和心输出量。 了解更多
  12. Rilmenidine

    Catalog No. A10794
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    α2 adrenergic 激动剂
    Rilmenidine是第二代咪唑啉-α2肾上腺素能激动剂。 了解更多
  13. Carvedilol

    Catalog No. A11843
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    β2-adrenergic receptor
    Carvedilol是具有抗氧化特性的β1和β2肾上腺素能受体(AR)激动剂。 了解更多
  14. Salmeterol

    Catalog No. A11788
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    beta2-adrenergic receptor 激动剂
    Salmeterol是一种长效β2-肾上腺素能受体激动剂。 了解更多
  15. Adrenalone HCl

    Catalog No. A11807
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    adrenergic 激动剂
    Adrenalone HCl是一种肾上腺素能激动剂,用作局部血管收缩药和止血药,主要作用于α-1肾上腺素能受体。 了解更多
  16. Arformoterol tartrate

    Catalog No. A12795
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    beta2-adrenergic 激动剂
    Arformoterol tartrate是β2-肾上腺素能激动剂。 了解更多
  17. Oxymetazoline hydrochloride

    Catalog No. A10686
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    alpha-1 adrenergic 激动剂
    Oxymetazoline是一种选择性的α-1激动剂和部分α-2激动剂局部减充血剂,以盐酸羟甲唑啉的形式使用。 了解更多
  18. Tetrahydrozoline Hydrochloride

    Catalog No. A13080
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    Adrenergic Receptor 激动剂
    Tetrahydrozoline Hydrochloride是一种引起结膜血管收缩的α激动剂。 了解更多
  19. Salmeterol Xinafoate

    Catalog No. A14223
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    β2-adrenoceptor 激动剂
    Salmeterol Xinafoate是一种长效的β2-肾上腺素能受体激动剂,具有抗炎作用。 了解更多
  20. Bambuterol HCl

    Catalog No. A14251
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    β-adrenoceptor 激动剂
    Bambuterol HCl是一种有效的β-肾上腺素受体激动剂,用于治疗哮喘。 了解更多
  21. Dexmedetomidine HCl

    Catalog No. A11846
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    alpha2-adrenoceptor 激动剂
    Dexmedetomidine hydrochloride是美托咪啶的活性异构体,它充当有效的,高度选择性的α2-AR(α2-肾上腺素受体)激动剂。 了解更多
  22. Medetomidine HCl

    Catalog No. A13775
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    adrenergic alpha-2 receptor 激动剂
    Medetomidine Hydrochloride是一种肾上腺素α2-受体激动剂,Ki为1.08 nM,比作用于α1-adrenoceptor选择性高1620倍。由于其镇痛和镇静作用而被用于兽医学。 了解更多
  23. CL 316243 disodium salt

    Catalog No. A13657
    β3 adrenergic 激动剂
    CL 316243 disodium salt是一种3β-肾上腺素能激动剂,被开发为一种抗肥胖和糖尿病的药物,并使小鼠的血糖水平迅速下降。 了解更多
  24. BRL 37344 Na Salt

    Catalog No. A13676
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    β3-adrenergic receptors 激动剂
    BRL 37344 Na Salt是具有脂解活性的β3-AR(β3-肾上腺素能受体)选择性激动剂。 了解更多
  25. Guanabenz acetate

    Catalog No. A13635
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    2A-AR adrenergic 激动剂
    Guanabenz acetate是a2A-AR肾上腺素能激动剂和IGRS(咪唑啉I2结合位点)选择性配体。 了解更多
  26. Cimaterol

    Catalog No. A13401
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    β-adrenergic receptors 激动剂
    Cimaterol是β的有效激动剂;肾上腺素能受体(人β的pEC50 = 8.13、8.78和6.62;1β,2β和3β)。 了解更多
  27. Idazoxan Hydrochloride

    Catalog No. A13409
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    α2- adrenoceptor 拮抗剂 / I2 imidazoline receptor 激动剂
    Idazoxan hydrochloride 是α2-AR肾上腺素受体拮抗剂和潜在I2咪唑啉受体激动剂。还显示I1咪唑啉受体拮抗剂活性。(I1、I2和α的公钥基础设施值分别为5.90、7.22、8.01、7.43和7.7)。 了解更多
  28. Tulobuterol

    Catalog No. A13432
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    Adrenergic Receptor 激动剂
    Tulobuterol是β-肾上腺素能受体激动剂,在结构上与特布他林有关。 了解更多
  29. UK 14,304 tartrate

    Catalog No. A13433
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    Adrenoceptors 激动剂
    UK 14,304 tartrate是一种全α2肾上腺素能激动剂。 了解更多
  30. Xylazine HCl

    Catalog No. A13434
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    Adrenergic Receptor 激动剂
    Xylazine hydrochloride是α2A-AR、α2B-AR和α2C-AR的活化剂。 了解更多
  31. (R,R)-Formoterol

    Catalog No. A14964
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    β2-adrenoceptor 激动剂
    (R,R)-Formoterol是一种长效β2激动剂,用于哮喘和慢性阻塞性疾病的治疗。 了解更多
  32. Guanfacine hydrochloride

    Catalog No. A15098
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    α2A-adrenoceptor 激动剂
    Guanfacine hydrochloride是一种抗高血压药,是一种选择性的α2A肾上腺素受体激动剂,Kd为31 nM,选择性是α2B肾上腺素受体的60倍。 了解更多
  33. Vilanterol trifenatate

    Catalog No. A15998
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    β2-adrenergic receptor 激动剂
    Vilanterol trifenatate是一种长效的β-2激动剂药物,于2013年5月与葛兰素氟替卡松合用,获葛兰素史克(Brax Elmitta)出售为Breo Ellipta,用于治疗慢性阻塞性肺疾病(COPD)。 了解更多
  34. Brimonidine Tartrate

    Catalog No. A15033
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    α-adrenergic receptor 激动剂
    Brimonidine Tartrate是一种高度选择性的α-肾上腺素能受体激动剂,对α2A肾上腺素能受体的EC50为0.45 nM。 了解更多
  35. Clorprenaline HCl

    Catalog No. A16465
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    β2-adrenergic receptor 激动剂
    Clorprenaline HCl是一种β2受体激动剂,具有显着的支气管扩张作用。 了解更多
  36. Vilanterol

    Catalog No. A13125
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    ultra-long-acting β? adrenoreceptor 激动剂
    Vilanterol是一种新的选择性β2-AR激动剂,PEC50值为10.37±0.05。 了解更多
  37. Methoxamine HCl

    Catalog No. A17365
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    alpha-1 adrenergic agonist
    Methoxamine Hydrochloride is an alpha-1 adrenergic agonist that causes prolonged peripheral vasoconstriction. 了解更多
  38. Ractopamine HCl

    Catalog No. A17372
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    beta-Adrenergic agonist
    Ractopamine HCl is a beta-Adrenergic agonist. It acts by being a full agonist at the TAAR1. 了解更多
  39. Midodrine hydrochloride

    Catalog No. A17757
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    Adrenergic alpha-1 agonist
    Midodrine hydrochloride is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of hypotension. It improves clinical outcome of chronic hypotension. 了解更多
  40. Midodrine

    Catalog No. A17758
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    adrenergic alpha-1 agonist
    Midodrine is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of HYPOTENSION. 了解更多
  41. Fenoterol

    Catalog No. A17774
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    Beta 2 adrenergic agonist
    Fenoterol is a Beta 2 adrenergic agonist designed to open up the airways to the lungs. It is classed as sympathomimetic beta agonist and asthma medication. 了解更多
  42. Brimonidine

    Catalog No. A17899
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    α2-adrenergic receptor agonist
    Brimonidine (UK 14304) is a full α2-adrenergic receptor (α2-AR) agonist. 了解更多
  43. Nylidrin Hydrochloride

    Catalog No. A17947
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    beta-adrenergic agonist
    Nylidrin hydrochloride is a beta-adrenergic agonist. Nylidrin hydrochloride is shown to be an effective inhibitor of IgE-mediated release of histamine from human basophils, and thus can be used as antiallergic agent. 了解更多
  44. Tulobuterol hydrochloride

    Catalog No. A18226
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    β2-adrenergic receptor agonist
    Tulobuterol Hydrochloride is a long-acting beta2-adrenergic receptor agonist. 了解更多
  45. BI-167107

    Catalog No. A18687
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    β2 adrenergic receptor agonist
    BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM. 了解更多

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