Epigenetic Reader Domain

Catalog No.Inhibitor Name Epigenetic Reader Domain
A12729(*)-JQ1
***
A11783I-BET151
*
A12545PFI-1
**
A11440I-BET-762
***
A13956RVX-208
*
A13227SGC-CBP30
****
A13163Bromosporine
****
A13890OTX015
****
A12948UNC1215
**
A13717UNC669
*
A14133GSK1324726A
***
A13749MS436
**
A13068CPI-203
***
A13957PFI-3

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. OF-1

    Catalog No. A16000
    Quick View
    BRPF1B/BRPF2 bromodomain 抑制剂
    OF-1是BRPF溴结构域的化学探针。OF-1已显示以100 nM的KD(ITC)结合到BRPF1B,以500 nM的KD(ITC)结合到BRPF2和以2.4 uM的KD(ITC)结合到BRPF3。 了解更多

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