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￥ 0.00 c-Kit
| Catalog No. | Inhibitor Name | c-Kit | Other |
|---|---|---|---|
| A10290 | Dasatinib | *** | Abl,Src |
| A10468 | Imatinib Mesylate | ** | PDGFR,v-Abl |
| A10996 | Cabozantinib | *** | VEGFR2/KDR,c-Met,VEGFR3/FLT4 |
| A10103 | Axitinib | **** | VEGFR1/FLT1,VEGFR2/Flk1,VEGFR2/KDR |
| A10699 | Pazopanib HCl | * | VEGFR1,VEGFR2,VEGFR3 |
| A11411 | Dovitinib | **** | FLT3,FGFR1,VEGFR3/FLT4 |
| A10967 | Vatalanib 2HCl | * | VEGFR2/KDR,VEGFR1/FLT1,VEGFR2/Flk1 |
| A10558 | Masitinib | * | Lyn B,PDGFRα,PDGFRβ |
| A10101 | Tivozanib | ** | VEGFR2,VEGFR3,EphB2 |
| A10610 | Amuvatinib | *** | PDGFRα (V561D),FLT3 (D835Y) |
| A10608 | Motesanib Diphosphate | *** | VEGFR1,VEGFR2,VEGFR2/Flk1 |
| A10679 | OSI-930 | ** | FLT1,KDR,CSF-1R |
| A10502 | Ki8751 | ** | VEGFR2,PDGFRα,FGFR2 |
| A10903 | Telatinib | **** | VEGFR3,VEGFR2,PDGFRα |
| A11518 | Pazopanib | * | VEGFR1,VEGFR2,VEGFR3 |
| A10198 | Dovitinib Dilactic Acid | **** | FLT3,FGFR1,VEGFR3/FLT4 |
| A16320 | Dasatinib Monohydrate | *** | Abl ,Src |
| A14156 | AZD2932 | *** | PDGFRβ,Flt3,VEGFR-2 |
| A10880 | Sunitinib Malate | FLT3,PDGFRβ,VEGFR2 | |
| A15062 | DCC-2618 | *** | PDGFRα, PDGFRβ |
| A15519 | PLX647 | *** | Fms |
| A15520 | Pexidartinib (PLX3397) | *** | CSF-1R, Flt-3 |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
5 个项目
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Pazopanib (GW-786034)
Catalog No. A11518 VEGFR 抑制剂Pazopanib (GW-786034)是VEGFR-1，VEGFR-2，VEGFR-3，PDGFR-a/β和c-kit的有效且选择性的多靶点酪氨酸激酶抑制剂，可阻止肿瘤生长并抑制血管生成。 了解更多 -
Dovitinib (TKI-258)
Catalog No. A11411 RTK 抑制剂Dovitinib是一种小分子多靶点酪氨酸激酶抑制剂，可抑制通过ZNF198-FGFR1或BCR-FGFR1转化为IL3独立性的Ba / F3细胞，IC50值分别为150 nM和90 nM。 了解更多 -
N-Desethyl Sunitinib
Catalog No. A15182 VEGFR/PDGFRβ/KIT 抑制剂N-Desethyl Sunitinib是舒尼替尼的主要药理活性代谢产物，是有效的，ATP竞争性VEGFR，PDGFRβ和KIT抑制剂（VEGFR -1，-2，-3的Ki值为2、9、17、8和4 nM。分别为PDGFRβ和KIT）。 了解更多 -
Dovitinib Dilactic acid (TKI258 Dilactic acid)
Catalog No. A10198 RTK 抑制剂Dovitinib是一种小分子多靶点酪氨酸激酶抑制剂，可抑制通过ZNF198-FGFR1或BCR-FGFR1转化为IL3独立性的Ba / F3细胞，IC50值分别为150 nM和90 nM。 了解更多 -
Regorafenib monohydrate
Catalog No. A15218 Tyrosine kinase 抑制剂Regorafenib monohydrate是VEGFR1/VEGFR2/VEGFR3/PDGFRβ/Kit/RET和Raf-1的多靶点抑制剂，IC50分别为13 nM/4.2 nM/46 nM/22 nM/7 nM/1.5 nM和2.5 nM。 了解更多
5 个项目
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