“jwh 250”的搜索结果

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  1. AZD8797

    Catalog No. A21230
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    human CX3CR1 receptor modulator
    AZD8797 is an allosteric non-competitive and orally active modulator of the human CX3CR1 receptor; antagonizes CX3CR1 and CXCR2 with Kis of 3.9 and 2800 nM, respectively. 了解更多
  2. GLP-26

    Catalog No. A18914
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    HBV capsid assembly modulator
    GLP-26 is a HBV capsid assembly modulators (CAM), inhibits HBV DNA replication in Hep AD38 system (IC50=3 nM), and reduces cccDNA by >90% at 1 μM. GLP-26 disrupts the encapsidation of pre-genomic RNA, causes nucleocapsid disassembly and reduces cccDNA pools. 了解更多
  3. TD-106

    Catalog No. A18595
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    CRBN modulator
    TD-106 is a cereblon (CRBN) modulator, which can be used for targeted protein degradation. BRD4 PROTACs with TD-106 induce BRD4 degradation. 了解更多
  4. (-)-(S)-B-973B

    Catalog No. A18761
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    α7 nAChR modulator
    -)-(S)-B-973B is a potent allosteric agonist and positive allosteric modulator of α7 nAChR, with antinociceptive activity. 了解更多
  5. Lorediplon

    Catalog No. A13449
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    GABAA receptor modulator
    Lorediplon 是一种新型的非苯二氮卓类催眠药,作为GABAA受体调节剂。 了解更多
  6. CBiPES HCl

    Catalog No. A15811
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    mGlu2 receptor modulator
    CBiPES HCl是mGluR-2的选择性正变构调节剂,IC50值为98.2 nM。 了解更多
  7. Cyclosporin B

    Catalog No. A15433
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    Immunomodulators
    Cyclosporin B是一种免疫抑制剂,已通过预防器官移植排斥反应而彻底改变了器官移植。 了解更多
  8. ISX-9

    Catalog No. A15774
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    Neurogenic Modulator
    ISX-9是成人神经干细胞分化的小分子诱导剂。 了解更多
  9. Toremifene

    Catalog No. A15265
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    Estrogen receptor modulator
    Toremifene是正在开发中的第二代选择性雌激素受体调节剂(SERM),用于预防骨质疏松症。 了解更多
  10. A-867744

    Catalog No. A11290
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    modulator of α7 nAChRs
    A-867744是α7烟碱乙酰胆碱受体的新型正变构调节剂。 了解更多
  11. BINA

    Catalog No. A11126
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    mGluR2 modulator
    BINA是mGlu2的选择性正构构调节剂(在表达人mGlu2的CHO细胞中EC50 = 33.2 nM)。 了解更多
  12. Plumbagin

    Catalog No. A15334
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    Immunomodulators
    Plumbagin在致癌和癌的啮齿动物模型中显示出细胞毒性;具有抗真菌,抗病毒和抗菌作用。 了解更多
  13. Compound W

    Catalog No. A15296
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    Gamma-secretase modulator
    Compound W是一种γ-分泌酶抑制剂,已被证明可以降低分泌的Aβ42和Nβ25的水平。 了解更多
  14. Flurizan

    Catalog No. A12433
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    gamma-secretase modulator
    Flurizan是一种非甾体抗炎药(NSAID),可抑制γ-分泌酶的活性。 了解更多

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