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搜索结果：“jwh 250”

“jwh 250”的搜索结果

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Cannabichromene

Catalog No. A15497
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TRPA1 activatior/TRPM8 blocker

Cannabichromene是一种主要的非精神植物大麻素，可抑制内源性大麻素失活并激活瞬时受体电位锚蛋白1（TRPA1）。内源性大麻素和TRPA1均可调节肠胃蠕动。了解更多

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Gap 26

Catalog No. A14865
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Gap junction blocker

Gap 26是连接蛋白模拟肽，对应于连接蛋白43的残基63-75，其是间隙连接阻断剂。了解更多

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GSK-2193874

Catalog No. A14201
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TRPV4 blocker

GSK2193874被确定为选择性的口服活性TRPV4阻滞剂，可通过重组TRPV4通道和天然内皮TRPV4电流抑制Ca(2+)流入。了解更多

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Encainide HCl

Catalog No. A13898
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Sodium channel blocker

Encainide hydrochloride是一种钠通道阻滞剂，具有Ic类抗心律不齐的作用。Encainide是一种非手性抗心律失常药和苯甲酰苯胺衍生物。了解更多

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Procainamide HCl

Catalog No. A14240
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Sodium channel blocker/DNMT 抑制剂

Procainamide HCl是钠通道阻滞剂，又是DNA甲基转移酶抑制剂。了解更多

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TRAM-34

Catalog No. A12783
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Potassium Channel Blocker

TRAM-34是中等电导Ca2+激活的K+通道（KCa3.1）（Kd = 20 nM）的高度选择性阻滞剂。在KV，BKCa，KCa2，Na+，CRAC和Cl-通道上具有200-1500倍的选择性。抑制有丝分裂刺激对淋巴细胞的激活。了解更多

Product Citations (2)

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- Samuel Drinkall, .et al. The two pore potassium channel THIK-1 regulates NLRP3 inflammasome activation, Glia, 2022, Jul;70(7):1301-1316 PMID: 35353387
- Cheong Hoon Seo, .et al. Altered K Ca 3.1 expression following burn injury and the therapeutic potential of TRAM-34 in post-burn hypertrophic scar formation, Transl Res, 2021, Apr 24 PMID: 33905948
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A 803467

Catalog No. A11234
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Sodium channel Blocker

A 803467是NaV1.8通道的选择性阻滞剂（hNaV1.8，hNaV1.3，hNaV1.7，hNaV1.5和hNaV1.2通道的IC50值分别为8、2450、6740、7340和7380 nM）。了解更多

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Cinnarizine

Catalog No. A16455
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calcium channel blocker

Cinnarizine是哌嗪的药物衍生物，其特征在于抗组胺药和钙通道阻滞剂。了解更多

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Phentolamine HCl

Catalog No. A13421
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α-Adrenergic blocker

Phentolamine HCl是一种AR(α肾上腺素能)阻滞剂。了解更多

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QX 314 chloride

Catalog No. A13760
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Sodium channel Blocker

QX 314 chloride是利多卡因的膜不可渗透的季衍生物，一种电压激活的Na+通道阻滞剂。了解更多

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Pindolol

Catalog No. A13422
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Beta adrenergic receptor blocker

Pindolol是一种非选择性β阻断剂，具有部分β肾上腺素能受体激动剂活性。了解更多

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Glyburide

Catalog No. A10433
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K+ channel and CFTR Cl- channel blocker

Glyburide (Glibenclamide) 是一种抗糖尿病化合物，是一类磺脲类药物。了解更多

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Cilnidipine

Catalog No. A10215
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Calcium channel blocker

Cilnidipine是提供血管平滑肌中L型电压门控钙通道和交感神经末梢N型钙通道的双重阻滞剂。了解更多

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