购物车 0 ￥ 0.00
微信关注
申请试用装
  • 主页 /
  • 搜索结果：“jwh 250”

“jwh 250”的搜索结果

产品 1 到 50 共 93个

每页
页面：
  1. 1
  2. 2

设置降序顺序
  1. Tonapofylline
    Quick View

    Tonapofylline

    Catalog No. A21328
    Quick View
    adenosine A1 receptor antagonist
    Tonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure. 了解更多
  2. Pavinetant
    Quick View

    Pavinetant

    Catalog No. A21174
    Quick View
    NK3R antagonist
    Pavinetant (MLE-4901) is a neurokinin-3 receptor (NK3R) antagonist. 了解更多
  3. AMG 487
    Quick View

    AMG 487

    Catalog No. A21162
    Quick View
    CXCR3 antagonist
    AMG 487 is an orally active and selective antagonist of CXC chemokine receptor 3 (CXCR3) which inhibits the binding of CXCL10 and CXCL11 to CXCR3 with IC50s of 8.0 and 8.2 nM, respectively. 了解更多
  4. RS102895 hydrochloride
    Quick View

    RS102895 hydrochloride

    Catalog No. A20918
    Quick View
    CCR2 antagonist
    RS102895 hydrochloride is a potent CCR2 antagonist, with an IC50 of 360 nM, and shows no effect on CCR1. 了解更多
  5. DW-1350
    Quick View

    DW-1350

    Catalog No. A12250
    Quick View
    LTB4 receptor antagonist
    DW-1350 is a LTB4 receptor antagonist. 了解更多
  6. I-191
    Quick View

    I-191

    Catalog No. A18629
    Quick View
    PAR2 antagonist
    I-191 is a potent, selective protease-activated receptor 2 (PAR2) antagonist. 了解更多
  7. BI-671800
    Quick View

    BI-671800

    Catalog No. A18902
    Quick View
    CRTH2 antagonist
    BI-671800 is a CRTH2 antagonist that treats patients with asthma. 了解更多
  8. AS-35
    Quick View

    AS-35

    Catalog No. A19409
    Quick View
    LTR antagonist
    AS-35 is an orally effective, potent and selective antagonist of leukotrienes, antagonizes LTC4-, LTD4 and LTE4-induced contractions of the ileum with IC50 values of 8 nM, 4 nM and 3 nM, respectively, and has antiallergic activities. 了解更多
  9. IAXO-102
    Quick View

    IAXO-102

    Catalog No. A18543
    Quick View
    TLR4 antagonist
    IAXO-102 is a TLR4 antagonist which negatively regulates TLR4 signalling. It inhibits MAPK and p65 NF-κB phosphorylation and expression of TLR4 dependent proinflammatory protein. 了解更多
  10. Icatibant
    Quick View

    Icatibant

    Catalog No. A18074
    Quick View
    Bradykinin B2 receptors antagonist
    Icatibant (HOE-140) is a selective and specific antagonist of bradykinin B2 receptor with IC50 and Ki of 1.07 nM and 0.798 nM respectively. 了解更多
  11. Revaprazan Hydrochloride
    Quick View

    Revaprazan Hydrochloride

    Catalog No. A17506
    Quick View
    Acid pump antagonist
    Revaprazan hydrochloride is a novel acid pump antagonist (APA). Revaprazan hydrochloride reduces COX-2 expression and has significant anti-inflammatory actions activities in H. pylori infection. 了解更多
  12. Fevipiprant
    Quick View
    • 最新产品

    Fevipiprant

    Catalog No. A17244
    Quick View
    CRTh2 receptor antagonist
    Fevipiprant, also known as NVP-QAW039 or QAW039, is an oral active and potent CRTh2 receptor antagonist and potentially useful for asthma treatment. 了解更多
  13. Procyclidine HCl
    Quick View

    Procyclidine HCl

    Catalog No. A17371
    Quick View
    Muscarinic antagonist
    Procyclidine hydrochloride is a muscarinic antagonist that crosses the blood-brain barrier and is used in the treatment of drug-induced extrapyramidal disorders and in Parkinsonism. 了解更多
  14. AF 12198
    Quick View

    AF 12198

    Catalog No. A17213
    Quick View
    IL-1 receptor 拮抗剂
    AF 12198是人I型白介素1（IL-1）受体的有效选择性拮抗剂。 了解更多
  15. TR-14035
    Quick View
    • 最新产品

    TR-14035

    Catalog No. A17118
    Quick View
    Integrin 拮抗剂
    TR-14035是α4β7和α4β1整联蛋白的双重拮抗剂。 了解更多
  16. AMG-333
    Quick View

    AMG-333

    Catalog No. A17182
    Quick View
    TRPM8 拮抗剂
    AMG-333是有效的选择性TRPM8拮抗剂，IC50为13 nM。 了解更多
  17. GYKI53655 Hydrochloride
    Quick View

    GYKI53655 Hydrochloride

    Catalog No. A17032
    Quick View
    AMPA 拮抗剂
    GYKI53655 Hydrochloride是一种非竞争性AMPA和海藻酸酯受体拮抗剂。 了解更多
  18. PHTPP
    Quick View

    PHTPP

    Catalog No. A17035
    Quick View
    ERβ receptor 拮抗剂
    PHTPP是基于吡唑并[1,5-α]嘧啶的配体，其作为雌激素ERβ受体的完全拮抗剂，其选择性是ERα的36倍。 了解更多
  19. Flavoxate
    Quick View

    Flavoxate

    Catalog No. A12900
    Quick View
    muscarinic AChR antagonist
    Flavoxate结合并抑制毒蕈碱受体，从而通过改变脑干的排尿中心来抑制排尿反射并增加膀胱容量。 了解更多
  20. RQ-00203078
    Quick View

    RQ-00203078

    Catalog No. A15830
    Quick View
    TRPM8 拮抗剂
    RQ-00203078是一种高度选择性，有效且可口服的TRPM8拮抗剂（大鼠和人类通道的IC50值分别为5.3和8.3 nM），对TRPM8的选择性是TRPV4，TRPV1和TRPA1的> 350倍。 了解更多
  21. UNBS5162
    Quick View

    UNBS5162

    Catalog No. A15439
    Quick View
    CXCL chemokines 拮抗剂
    UNBS5162是一种新型萘二甲酰亚胺，可降低实验性前列腺癌中CXCL趋化因子的表达。9种癌细胞系的平均抗增殖活性IC50值为17.9 uM；UNBS3157的水解产物。 了解更多
  22. SB271046
    Quick View

    SB271046

    Catalog No. A15438
    Quick View
    5-HT Receptor 拮抗剂
    SB271046 是一种有效的，选择性的5-HT6受体拮抗剂，pKi为8.9，与其他5-HT受体亚型相比，选择性高200倍。 了解更多
  23. CGS19755
    Quick View

    CGS19755

    Catalog No. A15791
    Quick View
    NMDA 拮抗剂
    CGS 19755（顺式-4-膦酰基甲基-2-哌啶羧酸）是一种有效的立体定向抑制剂，由N-甲基-D-天冬氨酸（NMDA）诱发，但不是由KCl诱发的[3H]乙酰胆碱释放大鼠纹状体的切片。 了解更多
  24. OPC21268
    Quick View

    OPC21268

    Catalog No. A15784
    Quick View
    vasopressin V1 拮抗剂
    OPC21268是一种非肽AVP受体V（Vasopressin Receptor）拮抗剂，对V1受体的选择性是V2受体的1000倍。 了解更多
  25. NIBR189
    Quick View

    NIBR189

    Catalog No. A15775
    Quick View
    EBI2 (GPR183) receptor 拮抗剂
    NIBR189是爱泼斯坦-巴尔病毒诱导的基因2（EBI2；GPR183）受体的小分子拮抗剂，IC50为16 nM（结合）和11 nM（功能性）。 了解更多
  26. SBC-115076
    Quick View

    SBC-115076

    Catalog No. A15769
    Quick View
    PCSK9 拮抗剂
    SBC-115076是抗蛋白原转化酶枯草杆菌蛋白酶kexin 9型（抗PCSK9）化合物，用于治疗和/或预防心血管疾病。 了解更多
  27. Talampanel
    Quick View

    Talampanel

    Catalog No. A15515
    Quick View
    AMPA/kainate receptor 拮抗剂
    Talampanel是AMPA受体的非竞争性拮抗剂，具有抗癫痫活性。 了解更多
  28. R18
    Quick View

    R18

    Catalog No. A15329
    Quick View
    14.3.3 proteins 拮抗剂
    R18是14.3.3蛋白的拮抗剂（KD≈80 nM）。竞争性地抑制14.3.3-配体相互作用，而无需磷酸化。 了解更多
  29. Ebrotidine
    Quick View

    Ebrotidine

    Catalog No. A15075
    Quick View
    H2-receptor 拮抗剂
    Ebrotidine是一种竞争性的H2受体拮抗剂（Ki = 127.5 nM），具有有效的抗分泌活性和胃保护作用。 了解更多
  30. SR 59230A HCl
    Quick View

    SR 59230A HCl

    Catalog No. A13430
    Quick View
    Adrenoceptors 拮抗剂
    SR 59230A HCl是3β-肾上腺素受体拮抗剂。 了解更多
  31. S-(-)-Atenolol
    Quick View

    S-(-)-Atenolol

    Catalog No. A13427
    Quick View
    Adrenoceptors 拮抗剂
    S-(-)-Atenolol是阿替洛尔的活性对映体，阿替洛尔是心脏选择性β肾上腺素能阻滞剂。 了解更多
  32. JP 1302 2HCl
    Quick View

    JP 1302 2HCl

    Catalog No. A13412
    Quick View
    α2C 拮抗剂
    JP 1302 2HCl是一种强效和选择性α2C拮抗剂。 了解更多
  33. HEAT hydrochloride (BE 2254)
    Quick View

    HEAT hydrochloride (BE 2254)

    Catalog No. A13408
    Quick View
    Adrenergic α1 Receptor 拮抗剂
    HEAT hydrochloride (BE 2254)是一种选择性很强的α1-肾上腺素受体拮抗剂，是3-[125I]-衍生物的前体。肾上腺素受体或肾上腺素能受体是参与多种交感神经系统过程的G蛋白偶联受体。 了解更多
  34. A 943931 2HCl
    Quick View

    A 943931 2HCl

    Catalog No. A13442
    Quick View
    Histamine H4 receptor 拮抗剂
    943931 2HCl是一种有效的选择性组胺H4受体拮抗剂（人和大鼠受体的pKi值分别为7.15和8.12）。 了解更多
  35. SB 258585 HCl
    Quick View

    SB 258585 HCl

    Catalog No. A14026
    Quick View
    5-HT6 serotonin receptor 拮抗剂
    SB 258585 hydrochloride是一种选择性和有效的SR-6拮抗剂。该化合物显示出比其他5-羟色胺受体亚型高160倍的选择性。 了解更多
  36. KU14R
    Quick View

    KU14R

    Catalog No. A13987
    Quick View
    I3 receptor 拮抗剂
    KU14R是胰腺β细胞非典型咪唑啉结合位点（可能的I3受体）的拮抗剂。KU14R也已显示出选择性阻断依法氧烷诱导的胰岛素分泌。 了解更多
  37. PF-3635659
    Quick View

    PF-3635659

    Catalog No. A13548
    Quick View
    muscarinic M(3) receptor 拮抗剂
    PF-3635659是有效的毒蕈碱M3受体拮抗剂。 了解更多
  38. IRL-2500
    Quick View

    IRL-2500

    Catalog No. A13638
    Quick View
    ETBR 拮抗剂
    IRL-2500是一种有效的选择性ETBR拮抗剂。它显示了对ETB受体的一些选择性（对于ETB和ETA受体，IC50值分别为1.3和94 nM）。 了解更多
  39. CYN-154806
    Quick View

    CYN-154806

    Catalog No. A13714
    Quick View
    somatostatin receptor 2 拮抗剂
    CYN-154806是一种有效的选择性生长抑素受体2（sst2）拮抗剂。 了解更多
  40. Atrasentan
    Quick View

    Atrasentan

    Catalog No. A13779
    Quick View
    ETA 拮抗剂
    Atrasentan是一种实验药物，正在研究中，用于治疗各种类型的癌症，包括非小细胞肺癌。它是对A型亚型（ETA）有选择性的内皮素受体拮抗剂,对ETA的IC50为0.0551 nM。 了解更多
  41. A-841720
    Quick View

    A-841720

    Catalog No. A13854
    Quick View
    mGluR-1 拮抗剂
    841720是一种有效的非竞争性mGluR-1拮抗剂，相对于mGluR-5具有34倍的选择性（IC50值分别为10和342 nM）。 了解更多
  42. BX471
    Quick View

    BX471

    Catalog No. A14409
    Quick View
    CCR1 拮抗剂
    BX471是一种有效的选择性非肽CCR1拮抗剂（对于人CCR1，Ki = 1 nM），对CCR1的选择性是CCR2，CCR5和CXCR4的250倍。 了解更多
  43. AM095
    Quick View

    AM095

    Catalog No. A13981
    LPA1 receptor 拮抗剂
    AM095是一种有效的LPA1受体拮抗剂，因为它抑制GTPβS与过量表达重组人或小鼠LPA1的中国仓鼠卵巢（CHO）细胞膜结合，IC50值分别为0.98和0.73μM，并且没有LPA1激动作用。 了解更多
  44. N-desMethyl EnzalutaMide
    Quick View

    N-desMethyl EnzalutaMide

    Catalog No. A13964
    Quick View
    androgen-receptor (AR) 拮抗剂
    N-desMethyl EnzalutaMide用于治疗涉及雄激素，雌激素和孕激素受体的疾病。 了解更多
  45. SB225002
    Quick View

    SB225002

    Catalog No. A14209
    Quick View
    CXCR2 拮抗剂
    SB225002是一种有效的选择性CXCR2拮抗剂，IC50为22 nM，可抑制白介素IL-8与CXCR2的结合，选择性是其他测试的7-TMR的150倍以上。 了解更多
  46. SB 399885 HCl
    Quick View

    SB 399885 HCl

    Catalog No. A14102
    Quick View
    5-HT6 拮抗剂
    SB 399885 hydrochloride是一种有效的，脑渗透剂和口服活性的SR-6拮抗剂。它对SR-6的选择性比其他血清素受体高200倍（对于人类重组，天然大鼠和天然人类SR-6受体，pKi值分别为9.11、8.81和9.02）。 了解更多
  47. Almorexant
    Quick View

    Almorexant

    Catalog No. A12503
    Quick View
    OX 拮抗剂
    Almorexant (ACT078573)是一种有效的竞争性双重食欲素1受体(OX1)/orexin 2受体（OX2）拮抗剂，对于OX1和OX2的Ki值分别为1.3和0.17 nM。 了解更多
  48. AM251
    Quick View

    AM251

    Catalog No. A12914
    Quick View
    CB1 receptor 拮抗剂
    AM251是有效的CB1受体拮抗剂（IC50 = 8 nM，Ki = 7.49 nM），其选择性是CB2受体的306倍。 了解更多
  49. S1RA (E-52862)
    Quick View

    S1RA (E-52862)

    Catalog No. A12504
    Quick View
    sigma-1 receptor 拮抗剂
    S1RA是一种选择性sigma-1受体拮抗剂，据报道其结合亲和力为Ki = 17.0±7.0 nM，对sigma-2受体具有选择性，并且对其他170种受体，酶，转运蛋白和离子通道具有选择性。 了解更多
  50. Reversine
    Quick View

    Reversine

    Catalog No. A13250
    Quick View
    human A3 adenosine receptor 拮抗剂 /Aurora 抑制剂
    Reversine是一种有效的人A3腺苷受体拮抗剂，Ki为0.66μM，是一种泛光A/B/C激酶抑制剂，IC50分别为12 nM/13 nM/20 nM。也用于干细胞去分化。 了解更多

产品 1 到 50 共 93个

每页
页面：
  1. 1
  2. 2

设置降序顺序
联系我们
ChinaChina

Adooq 中国 (南京百鑫德诺生物科技有限公司)

免费电话: 400-025-6535

企业QQ: 400-025-6535

www.adooq.cn

sales@adooq.cn

United StatesUnited States

Adooq Bioscience

Toll Free: (866) 930-6790

Fax: +1-323-606-8156

Email: sales@adooq.com

Not your Region? View all Distributors

FILTER BY:

Filtering:

  1. 作用机制: Antagonist (拮抗剂) 删除该内容
清除全部

购物选项

分类
  1. Epigenetics (1)
  2. Protein Tyrosine Kinases (1)
  3. Angiogenesis (1)
  4. Cell Cycle (1)
  5. Cytoskeleton (1)
  6. Cell Metabolism (2)
  7. Autophagy Signaling (5)
  8. Immunology & Inflammation (13)
  9. GPCR / G Protein (52)
  10. Neuronal Signaling (11)
  11. Microbiology (3)
  12. Membrane Transporters/Ion Channels (5)
  13. Endocrinology / Hormones (5)
  14. Others (1)
  15. Ready to Use Solution (13)
  16. Products On Sale (26)
  17. COVID-19 Related Products (1)
靶点
  1. A3 adenosine receptor (1)
  2. Aurora A (1)
  3. Aurora B (1)
  4. Aurora C (1)
  5. CXCR2 (1)
  6. CXCR4 (1)
ADOOQ 产品质量保证
Guaranteed product quality, 365 days Unconditional Return & Replacement

We promise all products to perform as described.

立即申请
Get Code
联系我们
查看FAQs

Adooq 公司

产品订购

技术资源

地址

© 2006-2019 AdooQ BioScience （南京百鑫德诺生物科技有限公司）. All Rights Reserved.
苏ICP备14027875号
Accept Payment
Rewards