“jwh 370”的搜索结果

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  1. Pancopride

    Catalog No. A12967
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    5-HT3 receptor antagonist
    Pancopride is a new potent and selective 5-HT3 receptor antagonist. 了解更多
  2. ML303

    Catalog No. A13702
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    NS1 antagonist
    ML303 is a pyrazolopyridine influenza virus nonstructural protein 1 (NS1) antagonist (IC90 = 155 nM), with an EC50 of 0.7 μM for Influenza A virus H1N1. 了解更多
  3. Alprenolol hydrochloride

    Catalog No. A17781
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    5-HT1A receptor antagonist
    Alprenolol (hydrochloride) is a non-selective beta blocker as well as 5-HT1A receptor antagonist. 了解更多
  4. LY 334370 hydrochloride

    Catalog No. A17027
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    5-HT1F 激动剂
    LY 334370 hydrochloride是一种选择性的5-HT1F受体激动剂(Ki值为1.87、16.4,> 100 (IC50))。CAS:199673-74-0(LY 334370盐酸盐);182563-08-2(LY 334370游离碱) 了解更多
  5. Tradipitant

    Catalog No. A16918
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    NK1 receptor 拮抗剂
    Tradipitant,也称为VLY-686和LY686017,是第二代神经激肽1受体拮抗剂,在临床前焦虑模型中表现出活性。 了解更多
  6. Naloxegol Oxalate

    Catalog No. A15972
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    Opioid 拮抗剂
    Naloxegol Oxalate是用于治疗阿片类药物引起的便秘的外周选择性阿片类药物拮抗剂。 了解更多
  7. PF-3274167

    Catalog No. A13754
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    Oxytocin 拮抗剂
    PF-3274167是一种高亲和力非肽催产素受体(OTR)拮抗剂,Ki为9.5 nM。 了解更多
  8. SCH 563705

    Catalog No. A15234
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    CXCR2/CXCR1 拮抗剂
    SCH 563705是有效的双重CXCR2(IC50 = 1.3 nM)/CXCR1(IC50 = 7.3 nM)拮抗剂。 了解更多
  9. Cilliobrevin D

    Catalog No. A12913
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    cytoplasmic dynein 拮抗剂
    Ciliobrevin D是第一个特定的细胞质动力蛋白小分子拮抗剂。 了解更多
  10. OC 000459

    Catalog No. A11946
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    CRTH2 拮抗剂
    OC 000459是一种有效的口服和选择性CRTH2(也称为DP2)拮抗剂。 了解更多

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