“ab fubinaca”的搜索结果

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  1. YF-2

    Catalog No. A21018
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    histone acetyltransferase activator
    YF-2 is a highly selective, blood-brain-barrier permeable histone acetyltransferase activator, acetylates H3 in the hippocampus, with EC50s of 2.75 μM, 29.04 μM and 49.31 μM for CBP, PCAF, and GCN5, respectively, shows no effect on HDAC. Anti-cancer and anti-Alzheimer's disease. 了解更多
  2. (1S,2S,3R)-DT-061

    Catalog No. A21701
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    PP2A activator
    (1S,2S,3R)-DT-061 is an enantiomer of DT-061. DT-061 is an orally bioavailable activator of protein phosphatase 2A (PP2A) and could be applied in the therapy of KRAS-mutant and MYC-driven tumorigenesis. 了解更多
  3. GPR40 Activator 1

    Catalog No. A21154
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    GPR40 activator
    GPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes. 了解更多
  4. Y-26763

    Catalog No. A12271
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    K+ (KATP) channel activator
    Y-26763 is a K+ channel opener and active metabolite of Y-27152. Y-26763 is an ATP-sensitive K+ (KATP) channel activator. 了解更多
  5. PF-04937319

    Catalog No. A13154
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    glucokinase activator
    PF-04937319 is a glucokinase activator (GKA) with EC50 value of 154.4 ?μM, one of the most promising strategies for the treatment of type 2 diabetes mellitus. 了解更多
  6. SMAP-2 (DT-1154)

    Catalog No. A18776
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    PP2A activator
    SMAP-2 (DT-1154) is an orally bioavailable phosphatase 2A (PP2A) activator which binds to the PP2A Aα scaffold subunit to drive conformational changes in PP2A. 了解更多
  7. ML-098

    Catalog No. A15925
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    Rab7 activator
    ML-098是GTP结合蛋白Rab7的激活剂(EC50 = 77.6 nM)。 了解更多
  8. Cannabichromene

    Catalog No. A15497
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    TRPA1 activatior/TRPM8 blocker
    Cannabichromene是一种主要的非精神植物大麻素,可抑制内源性大麻素失活并激活瞬时受体电位锚蛋白1(TRPA1)。内源性大麻素和TRPA1均可调节肠胃蠕动。 了解更多
  9. Mirabegron

    Catalog No. A12861
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    β3 adrenergic receptor activator
    Mirabegron是一种选择性的beta3-adrenoceptor(β3肾上腺素受体)激动剂,EC50为22.4 nM。是有效的膀胱松弛药和糖尿病药物。 了解更多

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