“ehop 016”的搜索结果

37 个项目

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  1. EHop-016

    Catalog No. A12740
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    Rac GTPase Inhibitor
    EHop-016 is a potent and specific inhibitor of Rac1 and Rac3 GTPase activity that inhibits Vav2 interaction with Rac, Rac-activated PAK1, lamellipodia formation, and cell migration. 了解更多
  2. NMS-P515

    Catalog No. A18449
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    PARP-1 抑制剂
    NMS-P515 is a potent inhibitor of PARP-1 both in biochemical (Kd: 0.016 μM) and cellular (IC50: 0.027 μM) assays. 了解更多
  3. MethADP sodium salt

    Catalog No. A21603
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    CD73 inhibitor
    MethADP (sodium salt) is a specific CD73 inhibitor. 了解更多
  4. CRA-026440

    Catalog No. A12179
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    HDAC inhibitor
    CRA-026440 is a potent, broad-spectrum HDAC inhibitor. 了解更多
  5. Glycolic acid oxidase inhibitor 1

    Catalog No. A13016
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    glycolate oxidase inhibitor
    Glycolic acid oxidase inhibitor 1 is a glycolate oxidase inhibitor, extracted from patent EP0021228A1, in Table IV. 了解更多
  6. T56-LIMKi

    Catalog No. A12266
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    LIMK2 inhibitor
    T56-LIMKi is a selective inhibitor of LIMK2; inhibits the growth of Panc-1 cells with an IC50 of 35.2 μM. 了解更多
  7. EC330

    Catalog No. A13799
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    leukemia inhibitory factor (LIF) inhibitor
    EC330 is a leukemia inhibitory factor (LIF) inhibitor. 了解更多
  8. HPGDS inhibitor 2

    Catalog No. A18390
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    H-PGDS 抑制剂
    HPGDS inhibitor 2 is a highly potent and selective hematopoietic prostaglandin D synthase (H-PGDS) inhibitor with an IC50 of 9.9 nM. 了解更多
  9. Bromodomain IN-1

    Catalog No. A18845
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    Bromodomain inhibitor
    Bromodomain IN-1 is a Bromodomain inhibitor extracted from patent WO2016069578A1, compound 4 . 了解更多
  10. UPGL00004

    Catalog No. A19047
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    GAC inhibitor
    UPGL00004 is a potent allosteric glutaminase C (GAC) inhibitor (IC50=29 nM; Kd=27 nM). UPGL00004 strongly inhibits the proliferation of highly aggressive triple-negative breast cancer cell lines. 了解更多
  11. RV01

    Catalog No. A19104
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    ALDH2 inhibitor
    RV01 is an analogue of resveratrol, inhibits DNA damage, reduces acetaldehyde dehydrogenase 2 (ALDH2) mRNA expression induced by ethanol, and exhibits hydroxyl radical scavenging activity. RV01 decreases iNOS expression, with anti-neuroinflammatory activity. 了解更多
  12. Fosfomycin calcium

    Catalog No. A18154
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    MurA and isopentenyl mevalonate kinase inhibitor
    Fosfomycin calcium is a MurA and isopentenyl mevalonate kinase inhibitor that prevents synthesis of bacterial cell walls. 了解更多
  13. MIK665

    Catalog No. A18362
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    Mcl-1 inhibitor
    MIK665 (S-64315) is a special Mcl-1 inhibitor extracted from patent WO2016207225A1, compound Preparation 13, has an IC50 of 1.81 nM. 了解更多
  14. Vadadustat

    Catalog No. A16794
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    HIF prolyl-hydroxylase 抑制剂
    Vadadustat,也称为AKB-6548和PG-1016548,是一种有效的缺氧诱导因子脯氨酸双加氧酶抑制剂。 了解更多
  15. Sivelestat sodium hydrate (ONO-5046 sodium hydrate)

    Catalog No. A16137
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    Neutrophil elastase 抑制剂
    Sivelestat sodium hydrate (ONO-5046 sodium hydrate)是人嗜中性粒细胞弹性蛋白酶的竞争性抑制剂,还抑制从兔,大鼠,仓鼠和小鼠获得的白细胞弹性蛋白酶。 了解更多
  16. LY2801653 (Merestinib)

    Catalog No. A12557
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    c-MET 抑制剂
    LY2801653 (Merestinib)是一种有效的,口服生物利用的小分子c-MET激酶抑制剂(Ki = 2 nM)。 了解更多
  17. KT 5720

    Catalog No. A16016
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    PKA 抑制剂
    KT5720 是一种能透过细胞的、有效的、特异性的、可逆的、ATP 竞争性的蛋白酶 K (PKA) 的抑制剂,其 Ki 值为 60 nM。 了解更多
  18. PD0166285

    Catalog No. A15863
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    Wee1 抑制剂
    PD0166285是一种有效的Wee1和Chk1抑制剂,在纳摩尔浓度下具有活性。PD0166285是一种新型的G2检查点消除剂。 了解更多
  19. ORY-1001 (RG-6016)

    Catalog No. A15893
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    LSD1 抑制剂
    ORY-1001 (RG-6016)是一种活性的选择性赖氨酸脱甲基酶LSD1/KDM1A抑制剂,IC50 <20 nM,对相关FAD依赖性氨氧化酶具有高选择性。 了解更多
  20. ETC-1002

    Catalog No. A15815
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    ACL 抑制剂 and AMPK 激活剂
    ETC-1002是一种新颖的,一流的可以降低LDL-C的小分子;肝AMP激活的蛋白激酶(AMPK)的激活剂;对肝ATP-柠檬酸裂解酶也具有有效的抑制活性(IC50 = 29 uM)。 了解更多
  21. JH-II-127

    Catalog No. A15777
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    LRRK2 抑制剂
    JH-II-127是一种高效,选择性和脑渗透性的LRRK2抑制剂,对于LRRK2野生型,LRRK2-G2019S和LRRK2-A2016T,IC50为6.6 nM,2.2 nM和47.7 nM。 了解更多
  22. SU6656

    Catalog No. A15518
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    SRC 抑制剂
    SU6656是Src激酶的选择性抑制剂,包括Src,Yes,Lyn和Fyn(分别为IC50 = 280、20、130、170 nM)。 了解更多
  23. NVP DPP 728 dihydrochloride

    Catalog No. A15320
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    DPP-4 抑制剂
    NVP DPP 728 dihydrochloride是一种有效的活性二肽基肽酶(DPP)-IV抑制剂,Ki和IC50值分别为11 nM和14 nM。 了解更多
  24. LY2801653 dihydrochloride

    Catalog No. A15150
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    MET 抑制剂
    LY2801653 dihydrochloride是一种有效的,口服可生物利用的c-MET激酶小分子抑制剂(Ki = 2 nM)。 了解更多
  25. SR 11302

    Catalog No. A14950
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    AP-1 transcription factor 抑制剂
    SR 11302,活化蛋白1(AP-1)转录因子活性的抑制剂,在体内表现出抗肿瘤作用。 了解更多
  26. Deoxygalactonojirimycin HCl

    Catalog No. A14016
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    Alpha-galactosidase 抑制剂
    Deoxygalactonojirimycin Hydrochloride是一种有效且选择性的Alpha-gal A(Alpha-半乳糖苷酶)抑制剂。 了解更多
  27. BV-6

    Catalog No. A14231
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    dual cIAP and XIAP 抑制剂
    BV-6是一种SMAC模拟,双重cIAP和XIAP抑制剂。 了解更多
  28. KX2-391

    Catalog No. A11177
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    Src 抑制剂
    KX2-391是新型的非ATP竞争底物口袋定向SRC抑制剂。 了解更多
  29. SB939 ( Pracinostat )

    Catalog No. A10830
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    HDAC 抑制剂
    SB939 (Pracinostat)是HDAC的口服抑制剂,对I,II和IV类HDAC具有选择性,在体外HDAC1活性测定中显示IC50值为77 nM。 了解更多
  30. BS-181

    Catalog No. A10163
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    CDK 抑制剂
    BS-181 是作为CDK7抑制剂的潜在抗肿瘤剂。 了解更多
  31. Bosutinib (SKI-606)

    Catalog No. A10161
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    Src 抑制剂
    Bosutinib (SKI-606)是一种酪氨酸激酶抑制剂。 了解更多
  32. Brivanib alaninate (BMS-582664)

    Catalog No. A10162
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    VEGFR 抑制剂
    Brivanib alaninate (BMS-582664)是VEGFR和FGFR信号转导的双重酪氨酸激酶抑制剂。 了解更多
  33. YM201636

    Catalog No. A11064
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    PI3K 抑制剂
    YM201636是PIKfyve的细胞渗透性和选择性抑制剂(IC50 = 33 nM)。 了解更多
  34. BSI-201 (Iniparib)

    Catalog No. A10164
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    PARP 抑制剂
    BSI-201 (Iniparib)是一种有效的PARP-1抑制剂,已被证明可以穿越血脑屏障。 了解更多
  35. BTZ043 (BTZ038, BTZ044) Racemate

    Catalog No. A10165
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    DprE1 抑制剂
    BTZ043 (BTZ038,BTZ044) Racemate 抑制癸二烯基磷酸基-β-d-核糖2α-表异构酶,它是一种产生致病细菌结核分枝杆菌细胞壁的酶。 了解更多
  36. Bortezomib (Velcade)

    Catalog No. A10160
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    Proteasome 抑制剂
    Bortezomib (Velcade)是26S蛋白酶体的高度选择性,可逆抑制剂。 了解更多
  37. BKM120 (NVP-BKM120, Buparlisib)

    Catalog No. A11016
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    PI3K 抑制剂?
    BKM120 (NVP-BKM120,Buparlisib)是生物可利用的口服泛I类磷脂酰肌醇3激酶(PI3K)激酶抑制剂,在无细胞试验中作用于p110α/β/δ/γ的。对VPS34,mTOR,DNAPK的作用效果下降,而对 PI4Kβ几乎没有活性。 了解更多

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