“jwh 370”的搜索结果

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  1. KN-92 phosphate

    Catalog No. A15139
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    CaMKII 抑制剂
    KN-92 phosphate是KN-93的非活性衍生物。KN-93是Ca2+/钙调蛋白依赖性激酶II(CaMKII)的选择性抑制剂,竞争性阻断CaM与激酶的结合(Ki = 370 nM)。 了解更多
  2. KN-92

    Catalog No. A15137
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    CaMK-II 抑制剂
    KN-92是KN-93的非活性衍生物。KN-93是Ca2+/钙调蛋白依赖性激酶II(CaMKII)的选择性抑制剂,竞争性阻断CaM与激酶的结合(Ki = 370 nM)。 了解更多
  3. CG-806

    Catalog No. A19814
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    FLT3/BTK inhibitor
    CG-806 is an orally active, potent and non-covalent pan-FLT3/pan-BTK inhibitor with an IC50 of 0.08 μM for FLT3. CG-806 has an IC50 of 11 nM against FLT3 wild type (WT)-transfected Ba/F3 cells. 了解更多
  4. MSI-1436 lactate

    Catalog No. A21929
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    PTB1B inhibitor
    MSI-1436 lactate is a selective, non-competitive inhibitor of the enzyme protein-tyrosine phosphatase 1B (PTB1B), with an IC50 of 1 μM, 200-fold preference over TCPTP (IC50 of 224 μM). 了解更多
  5. Liarozole dihydrochloride

    Catalog No. A21853
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    CYP450 dependent inhibitor
    Liarozole dihydrochloride (R75251; R85246) is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase). 了解更多
  6. Ensartinib hydrochloride

    Catalog No. A21719
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    ALK/MET inhibitor
    Ensartinib hydrochloride (X-396 hydrochloride) is a potent and dual ALK/MET inhibitor with IC50s of <0.4 nM and 0.74 nM, respectively. 了解更多
  7. Solenopsin

    Catalog No. A21087
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    ATP-competitive AKT inhibitor
    Solenopsin is an ATP-competitive AKT inhibitor with IC50 value of 10 μM . 了解更多
  8. LDN-27219

    Catalog No. A20844
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    hTGase inhibitor
    LDN-27219 is a potent inhibitor of hTGase(Tissue transglutaminase) with an IC50 of 0.6 uM. 了解更多
  9. RIPA-56

    Catalog No. A12473
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    RIP1 inhibitor
    RIPA-56 is a highly potent, selective, and metabolically stable inhibitor of receptor-interacting protein 1 (RIP1) with an IC50 of 13 nM. 了解更多
  10. JNJ4796

    Catalog No. A13707
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    Influenza virus inhibitor
    JNJ4796 is an oral active fusion inhibitor of influenza virus, neutralizing influenza A group 1 viruses by inhibiting hemagglutinin (HA)-mediated fusion. 了解更多
  11. ZT-12-037-01

    Catalog No. A18395
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    ATP-competitive STK19 inhibitor
    ZT-12-037-01 is a potent, selective, ATP-competitive STK19 inhibitor. ZT-12-037-01 effectively blocks oncogenic NRAS-driven melanocyte malignant transformation and melanoma growth in vitro and in vivo. 了解更多
  12. DW14800

    Catalog No. A18491
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    PRMT5 inhibitor
    DW14800 is a protein arginine methyltransferase 5 (PRMT5) inhibitor, with an IC50 of 17 nM. DW14800 reduces H4R3me2s levels and enhances the transcription of HNF4α, but does not alter PRMT5 expression. Anti-cancer activity. 了解更多
  13. BC-1215

    Catalog No. A18605
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    FBXO3 inhibitor
    BC-1215 is an inhibitor of F-box protein 3 (FBXO3, a ubiquitin E3 ligase component, IC50=0.9 μg/mL for IL-1β release). BC-1215 decreases Fbxo3-Fbxl2 interaction and prevents SCFFbxo3 catalyzed Fbxl2 ubiquitination. 了解更多
  14. Cangrelor Tetrasodium

    Catalog No. A17919
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    P2Y12 receptors inhibitor
    Cangrelor Tetrasodium is a high-affinity, reversible inhibitor of P2Y12 receptors that causes almost complete inhibition of ADP-induced platelet aggregate. It is a modified ATP derivative stable to enzymatic degradation. Unlike clopidogrel (Plavix), which is a prodrug, cangrelor is an active drug not requiring metabolic conversion. 了解更多
  15. SSE15206

    Catalog No. A18350
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    Microtubule/Tubulin Inhibitor
    SSE15206 is a pyrazolinethioamide derivative that has potent antiproliferative activities in cancer cell lines of different origins and overcomes resistance to microtubule-targeting agents. 了解更多
  16. PF-06737007

    Catalog No. A17179
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    Trk 抑制剂
    PF-06737007是泛原肌球蛋白相关激酶(Trk)抑制剂。 了解更多
  17. SR-4370

    Catalog No. A16899
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    HDAC 抑制剂
    SR-4370是HDAC抑制剂。SR-4370对HDAC1,HDAC2和HDAC3的IC50值分别为0.5 uM,0.1 uM和0.06 uM。 了解更多
  18. Elbasvir (MK-8742)

    Catalog No. A16855
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    NS5A 抑制剂
    Elbasvir (MK-8742)是一种NS5A抑制剂,可预防丙型肝炎病毒RNA复制和病毒体组装。根据基因型,EC50的中值范围为0.2至3600 pmol/L。 了解更多
  19. AX-024

    Catalog No. A16926
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    T cell receptor 抑制剂
    AX-024是一种细胞因子释放抑制剂,可以强烈抑制白介素6(IL-6),肿瘤坏死因子-α(TNFα),干扰素-γ(IFN-γ),IL-10和IL-17A的产生。 了解更多
  20. CI 976

    Catalog No. A16370
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    ACAT/SOAT 抑制剂
    CI 976是肝和肠酰基辅酶A胆固醇酰基转移酶(ACAT)和固醇O-酰基转移酶(SOAT)的三甲氧基脂肪酸苯胺抑制剂。Cl 976降低非高密度脂蛋白(non-HDL)胆固醇并增加HDL-胆固醇浓度。 了解更多
  21. FLT3-IN-1

    Catalog No. A16249
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    FLT3 抑制剂
    FLT3-IN-1是一种新型的有效选择性Flt3抑制剂,IC50为10 nM。抗表达FLT3-ITD的MV4-11细胞,IC50为6 nM。 了解更多
  22. BML-210

    Catalog No. A15935
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    HDAC 抑制剂?
    BML-210是HDAC抑制剂。BML-210诱导宫颈癌细胞中的生长抑制和凋亡并调节HDAC和DAPC复合物的表达水平。 了解更多
  23. CL-387785 (EKI-785)

    Catalog No. A13146
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    EGFR 抑制剂
    CL-387785是EGFR的不可逆抑制剂,IC50为370+/-120 pM;能够在功能水平上克服由T790M突变引起的抗药性。 了解更多
  24. CID 797718

    Catalog No. A13809
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    PKD1 抑制剂
    CID797718是CID755673(Adooq目录号A13804)的结构类似物。它是效力降低10倍的PKD1抑制剂,IC50值为7.0+/-0.8 uM。 了解更多
  25. AZ-33

    Catalog No. A13341
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    LDHA 抑制剂
    AZ33是LDHA抑制剂。 了解更多
  26. E7820

    Catalog No. A15456
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    lpha-2-integrin 抑制剂
    E7820是一种小分子芳香族磺酰胺衍生物,具有潜在的抗血管生成和抗肿瘤活性。E7820通过抑制整合素α2(一种在内皮细胞上表达的细胞粘附分子)来抑制血管生成。 了解更多
  27. GSK2879552

    Catalog No. A15547
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    LSD1 抑制剂
    GSK2879552是一种可逆的赖氨酸特异性脱甲基酶1(LSD1)抑制剂,具有潜在的抗肿瘤活性。 了解更多
  28. 4-HQN

    Catalog No. A15370
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    PARP 抑制剂
    4-HQN已显示抑制PARP(聚(ADP-核糖)合成酶),该酶催化NAD+的ADP-核糖部分与各种蛋白质的共价结合。 了解更多
  29. TC-H 106

    Catalog No. A15357
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    HDAC 抑制剂
    TC-H 106是一种慢速,紧密结合的I类HDAC(组蛋白脱乙酰基酶)抑制剂。 了解更多
  30. UK 370106

    Catalog No. A15316
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    MMP-3/MMP-12 Inhiibitor
    UK 370106是一种高度选择性的MMP-3和MMP-12抑制剂。 了解更多
  31. O6-Benzylguanine

    Catalog No. A13706
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    MGMT 抑制剂
    O6-Benzylguanine是DNA烷基转移酶的有效底物和有效灭活剂。O6-苄基鸟嘌呤是MGMT的抑制剂。 了解更多
  32. NBMPR

    Catalog No. A13701
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    ENT1 抑制剂
    NBMPR是一种核苷类似物,可竞争性抑制平衡的核苷转运蛋白1(大鼠和人的Kd = 0.1-1.0 nM,IC50s = 4.6和3.6 nM)。 了解更多
  33. Cyclothiazide

    Catalog No. A13700
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    AMPA desensitization 抑制剂
    Cyclothiazide是苯并噻二叠氮,可作为AMPA受体的增效剂,正向调节其对谷氨酸的响应(EC50 = 3.8 M)。 了解更多
  34. RG108

    Catalog No. A13054
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    DNA methyltransferase 抑制剂
    RG108是DNA甲基转移酶的非核苷抑制剂,IC50为115 nM。 了解更多
  35. AK-1

    Catalog No. A14370
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    SIRT2 抑制剂
    AK-1比SIRT1和SIRT3选择性抑制SIRT2。 了解更多
  36. CAY10650

    Catalog No. A14355
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    cPLA2α 抑制剂
    CAY10650是一种高效(IC50 = 12 nM)cPLA2α抑制剂。 了解更多
  37. DTP348

    Catalog No. A14410
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    CAIX 抑制剂/ radiosensitizer
    DTP348是双重CAIX抑制剂/放射增敏剂。 了解更多
  38. 1-Azakenpaullone

    Catalog No. A14303
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    GSK-3β 抑制剂
    1-Azakenpaullone是一种有效的选择性GSK-3β抑制剂,IC50为18 nM,选择性比CDK1/cyclin B和CDK5/p25高100倍。 了解更多
  39. ESI-09

    Catalog No. A14233
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    EPAC1/EPAC2 抑制剂
    ESI-09是一种直接由cAMP(EPAC)抑制剂激活的特异性交换蛋白,对于EPAC1和EPAC2,IC50为3.2 uM和1.4 uM。 了解更多
  40. Mevastatin

    Catalog No. A13709
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    HMG-CoA reductase 抑制剂
    Mevastatin是HMG-CoA还原酶的抑制剂。 了解更多
  41. UNC1215

    Catalog No. A12948
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    L3MBTL3 抑制剂
    UNC1215是具有细胞活性的L3MBTL3的强效选择性拮抗剂。 了解更多
  42. PRT062607 HCL

    Catalog No. A12731
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    Syk 抑制剂
    PRT2607,也称为PRT062607,P505-15和BIIB057,是一种新型,高度选择性且口服可生物利用的小分子SYK抑制剂(SYK IC(50)= 1 nM),具有至少80倍的抗SYK活性 大于对其他激酶的亲和力。 了解更多
  43. Batimastat (BB-94)

    Catalog No. A12985
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    MMP 抑制剂
    Batimastat (BB-94)是多种基质金属蛋白酶(MMP)的强效合成抑制剂,包括间质胶原酶(IC50 = 3 nM),溶血素(IC50 = 20 nM),Mr 72,000型IV胶原酶(IC50 = 4) nM),92,000型IV胶原酶先生(IC50 = 4 nM)和基质溶素(IC50 = 6 nM)。它是一种低分子量(MW = 478)的肽样胶原蛋白底物类似物,由类似物结合而成,分别与MMP和催化活性锌原子结合在一起。 了解更多
  44. BCH

    Catalog No. A13370
    LAT1 抑制剂
    BCH是L型氨基酸转运蛋白LAT1的抑制剂。通过激活KB,Saos2和C6癌细胞系中的半胱氨酸蛋白酶抑制生长并诱导凋亡。 了解更多
  45. JNK-IN-8

    Catalog No. A12749
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    JNK 抑制剂
    JNK-IN-8是第一种JNK1,JNK2和JNK4不可逆JNK抑制剂,IC50分别为4.7 nM,18.7 nM和1 nM。 了解更多
  46. P505-15 (PRT062607, BIIB057)

    Catalog No. A11952
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    Syk 抑制剂
    P505-15 (PRT062607,BIIB057)是一种新型的,高度选择性的,Syk抑制剂(SYK IC(50)= 1 nM),具有比SYK活性至少高80倍的抗SYK活性。 了解更多
  47. MK-2461

    Catalog No. A11753
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    c-Met 抑制剂
    MK-2461是一种新型的多靶点激酶抑制剂,优先抑制活化的c-Met受体。 了解更多
  48. KRN 633

    Catalog No. A10504
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    VEGFR 抑制剂
    KRN 633是一种细胞可渗透、可逆、ATP竞争性VEGFR激酶抑制剂,仅在较高浓度下(IC50 = 0.97 μM和4.33 μM)抑制PDGFR-α和C-Kit,对其他17种激酶无活性(IC50 ≥ 10 μM)。 了解更多
  49. Tubacin

    Catalog No. A10954
    HDAC6 抑制剂
    Tubacin (tubulin acetylation inducer)是一种高效且选择性强,可逆,可透过细胞的HDAC6抑制剂,IC50为4 nM。 了解更多
  50. BTZ043 (BTZ038, BTZ044) Racemate

    Catalog No. A10165
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    DprE1 抑制剂
    BTZ043 (BTZ038,BTZ044) Racemate 抑制癸二烯基磷酸基-β-d-核糖2α-表异构酶,它是一种产生致病细菌结核分枝杆菌细胞壁的酶。 了解更多

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