“jwh 370”的搜索结果

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  1. KN-92 phosphate

    Catalog No. A15139
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    CaMKII 抑制剂
    KN-92 phosphate是KN-93的非活性衍生物。KN-93是Ca2+/钙调蛋白依赖性激酶II(CaMKII)的选择性抑制剂,竞争性阻断CaM与激酶的结合(Ki = 370 nM)。 了解更多
  2. KN-92

    Catalog No. A15137
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    CaMK-II 抑制剂
    KN-92是KN-93的非活性衍生物。KN-93是Ca2+/钙调蛋白依赖性激酶II(CaMKII)的选择性抑制剂,竞争性阻断CaM与激酶的结合(Ki = 370 nM)。 了解更多
  3. Cangrelor Tetrasodium

    Catalog No. A17919
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    P2Y12 receptors inhibitor
    Cangrelor Tetrasodium is a high-affinity, reversible inhibitor of P2Y12 receptors that causes almost complete inhibition of ADP-induced platelet aggregate. It is a modified ATP derivative stable to enzymatic degradation. Unlike clopidogrel (Plavix), which is a prodrug, cangrelor is an active drug not requiring metabolic conversion. 了解更多
  4. CID 797718

    Catalog No. A13809
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    PKD1 抑制剂
    CID797718是CID755673(Adooq目录号A13804)的结构类似物。它是效力降低10倍的PKD1抑制剂,IC50值为7.0+/-0.8 uM。 了解更多

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