“jwh 249”的搜索结果

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  1. L-APB

    Catalog No. A21872
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    mGluRs M3 agonist
    L-APB is a potent and specific agonist for the group III mGluRs, with EC50s of 0.13, 0.29, 1.0, 249 μM for mGlu4, mGlu8, mGlu6 and mGlu7 receptors, respectively. 了解更多
  2. Methoxy-PEPy

    Catalog No. A21899
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    mGlu5 receptor antagonist
    Methoxy-PEPy is a potent and highly selective mGlu5 receptor antagonist with IC50 of 1 nM. 了解更多
  3. Toreforant

    Catalog No. A21058
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    histamine H4 receptor (H4R) antagonist
    Toreforant is a potent and selective histamine H4 receptor (H4R) antagonist, with a Ki at the human receptor of 8.4 nM. 了解更多
  4. RU 24969

    Catalog No. A20857
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    5-HT1A/5-HT1B receptors agonist
    RU 24969 is a selective agonist at the 5-HT1A and 5-HT1B receptors. 了解更多
  5. ST-836 hydrochloride

    Catalog No. A15249
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    ST-836 hydrochloride是多巴胺受体配体;反帕金森氏剂。 了解更多
  6. SB225002

    Catalog No. A14209
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    CXCR2 拮抗剂
    SB225002是一种有效的选择性CXCR2拮抗剂,IC50为22 nM,可抑制白介素IL-8与CXCR2的结合,选择性是其他测试的7-TMR的150倍以上。 了解更多
  7. RU 24969 hemisuccinate

    Catalog No. A13833
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    5-HT1A/1B and 5-HT2C 激动剂
    RU 24969 hemisuccinate是有效的5-HT1A/1B和中度5-HT2C激动剂,也可能释放5-HT。 了解更多
  8. SB 334867

    Catalog No. A12786
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    OX1 receptor 拮抗剂
    SB 334867是一种选择性的非肽orexin OX1受体拮抗剂。对于分别表达人OX1和OX2受体的CHO细胞中的细胞内Ca2 +释放抑制,pKb值为7.2和<5。体内全身给药后,阻断orexin-A诱导的美容和进食。 了解更多
  9. Anamorelin

    Catalog No. A12346
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    Anamorelin是一种新型 ghrelin receptor激动剂,FLIPR 检测中,EC50 为 0.74 nM,用于治疗与恶病质/厌食症相关的非小肺癌。 了解更多

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