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￥ 0.00 “MK 1775”的搜索结果
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MK-1775
Catalog No. A10599 -
Flavokawain B
Catalog No. A22437 apoptosis inducerFlavokawain B (Flavokavain B) is a chalcone isolated from the root extracts of kava-kava plant and a potent apoptosis inducer for inhibiting the growth of various cancer cell lines. 了解更多 -
Molnupiravir
Catalog No. A22165 broad-spectrum antiviral activityMolnupiravir (EIDD-2801, MK-4482) is an orally bioavailable prodrug of the ribonucleoside analog β-d-N4-hydroxycytidine (NHC; EIDD-1931) with broad-spectrum antiviral activity against SARS-CoV-2, MERS-CoV, SARS-CoV, and the causative agent of COVID-19. 了解更多 -
KN-93 phosphate
Catalog No. A22229 membrane-permeant synthetic inhibitorKN-93 phosphate is a novel membrane-permeant synthetic inhibitor of purified neuronal CaMK-II, with Ki of 370 nM. 了解更多 -
Emamectin Benzoate
Catalog No. A22417 nervoussystem toxicantEmamectin Benzoate (MK-244) is an orally active nervoussystem toxicant by binding g-aminobutyric (GABA) receptor in insects. 了解更多 -
MK-212 HCl
Catalog No. A22531 MK 212 hydrochloride is a 5-HT receptor agonist; displays selectivity for 5-HT2C over 5-HT2A (IC50 values are 0.028 and 0.42 μM for human 5-HT2C and 5-HT2A receptors expressed in HEK293 cells respectively). 了解更多 -
MK-8033 hydrochloride
Catalog No. A22011 dual c-Met/Ron inhibitorMK8033 Hcl is a novel and specific dual ATP competitive c-Met/Ron inhibitor (IC50=1 nM Wt c-Met) under investigation as a treatment for cancer. 了解更多 -
MK-0941
Catalog No. A20823 allosteric glucokinase activatorMK-0941 is a potent, orally active and allosteric glucokinase activator, with EC50s of 240 and 65 nM for recombinant human glucokinase in the presence of 2.5 and 10 mM glucose, respectively. MK-0941 has potential in the treatment of type 2 diabetes. 了解更多 -
Pumosetrag Hydrochloride
Catalog No. A20692 5-HT3 partial agonistPumosetrag Hydrochloride (MKC-733; DDP-733) is an orally available 5-HT3 partial agonist developed for the treatment of irritable bowel syndrome and gastroesophageal reflux disease. 了解更多 -
DFMTI
Catalog No. A20558 -
Biotin-VAD-FMK
Catalog No. A20384 caspase inhibitorBiotin-VAD-FMK is a cell permeable, irreversible biotin-labeled caspase inhibitor, used to identify active caspases in cell lysates. 了解更多 -
Paprotrain
Catalog No. A20346 MKLP-2 inhibitorPaprotrain is a cell-permeable inhibitor of the kinesin MKLP-2, inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM and shows a moderate inhibition activity on DYRK1A with an IC50 of 5.5 μM. 了解更多 -
VU591 hydrochloride
Catalog No. A20009 ROMK inhibitorVU591 hydrochloride is a potent, selective renal outer medullary potassium channel (ROMK or Kir1.1) inhibitor, with an IC50 of 0.24 μM. 了解更多 -
OT antagonist 3
Catalog No. A19949 oxytocin (OT) antagonistOT antagonist 3 is an oxytocin (OT) antagonist extracted from patent WO2007017752A1. 了解更多 -
Islatravir
Catalog No. A19638 Islatravir (MK-8591) is a potent anti-HIV-1 agent, acting as a nucleoside reverse transcriptase inhibitor, with EC50s of 0.068 nM, 3.1 nM and 0.15 nM for HIV-1 (WT), HIV-1 (M184V), HIV-1 (MDR), respectively. 了解更多 -
Calmidazolium chloride
Catalog No. A19306 CaMK antagonistCalmidazolium chloride (R 24571) is a calmodulin (CaMK) antagonist, antagonizing CaM-dependent phosphodiesterase and calmodulin-induced activation of erythrocyte Ca2+-transporting ATPase with IC50s of 0.15 and 0.35 μM, respectively. Also in anti-cancer research. Calmidazolium binds to CaMK with a Kd of 3 nM. 了解更多 -
Gefapixant
Catalog No. A19254 P2X3R antagonistGefapixant is an orally active P2X3 receptor (P2X3R) antagonist with IC50s of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors. 了解更多 -
Eprinomectin
Catalog No. A21657 Eprinomectin(MK-397) is an avermectin selected for development as a topical endectocide; has anthelmintic, insecticidal and miticidal activity. 了解更多 -
CaMKII-IN-1
Catalog No. A21034 CaMKII inhibitorCaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM. 了解更多 -
MK-7145
Catalog No. A21030 -
Raltegravir potassium
Catalog No. A21403 integrase (IN) inhibitorRaltegravir is a potent integrase (IN) inhibitor, used to treat HIV infection. 了解更多 -
Rislenemdaz
Catalog No. A21907 NMDA receptor GluN2B antagonistRislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively. 了解更多 -
Niraparib R-enantiomer
Catalog No. A21880 PARP1 inhibitorNiraparib R-enantiomer (MK-4827 R-enantiomer) is an excellent PARP1 inhibitor with IC50 of 2.4 nM. 了解更多 -
Etoricoxib D4
Catalog No. A21877 COX-2 inhibitorEtoricoxib D4 (MK-0663 D4) is a deuterium labeled Etoricoxib. Etoricoxib is a non steroidal anti-inflammatory agent, acting as a selective and orally active COX-2 inhibitor, with IC50s of 1.1 μM and 116 μM for COX-2 and COX-1 in human whole blood. 了解更多 -
1-Naphthyl PP1 hydrochloride
Catalog No. A21790 Src/c-Abl inhibitor1-Naphthyl PP1 hydrochloride is a selective inhibitor of src family kinases v-Src and c-Fyn as well as the tyrosine kinase c-Abl (IC50 values are 1.0, 0.6, 0.6, 18 and 22 μM for v-Src, c-Fyn, c-Abl, CDK2 and CAMK II respectively). 了解更多 -
SRI 31215 TFA
Catalog No. A21775 triplex matriptase inhibitorSRI 31215 (TFA), a triplex inhibitor of matriptase, hepsin and hepatocyte growth factor activator (HGFA) with IC50s of 0.69 μM, 0.65 μM, 0.3 μM, blocks pro-HGF activation and thus mimics the activity of HAI-1/2. 了解更多 -
LY 344864 hydrochloride
Catalog No. A21748 5-HT1F agonistLY 344864 hydrochloride is a selective 5-HT1F agonist with a Ki of 6 nM. 了解更多 -
Taranabant ((1R,2R)stereoisomer)
Catalog No. A21705 CB1 receptor inverse agonistTaranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多 -
Taranabant racemate
Catalog No. A21699 CB1 antagonist/inverse agonistTaranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor extracted from patent WO 2004048317 A1. 了解更多 -
Ubrogepant
Catalog No. A21670 CGRP antagonistUbrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine. 了解更多 -
MK2-IN-1 hydrochloride
Catalog No. A21662 MAPKAPK2(MK2) inhibitorMK2-IN-1 hydrochloride is a potent and selecitve MAPKAPK2(MK2) inhibitor(IC50=0.11 uM) with a non-ATP competitive binding mode. 了解更多 -
Serlopitant
Catalog No. A21582 Neurokinin-1 (NK-1) receptor antagonistSerlopitant is a selective Neurokinin-1 (NK-1) receptor antagonist. 了解更多 -
Finasteride acetate
Catalog No. A21537 testosterone 5-alpha-reductase inhibitorFinasteride (acetate) is an orally active testosterone 5-alpha-reductase inhibitor. 了解更多 -
Amicarbazone
Catalog No. A21294 photosynthetic electron transport inhibitorAmicarbazone(BAY-MKH3586; BAY314666) is a potent inhibitor of photosynthetic electron transport via binding to the Qb domain of photosystem II (PSII); herbicide with a broad spectrum of weed control. 了解更多
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- Epigenetics (10)
- Apoptosis (14)
- PI3K / Akt / mTOR (6)
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- Products On Sale (41)
- Recombinant Proteins (2)
- Enzymes (6)
- 作用机制
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- Inhibitor (抑制剂) (116)
- Agonist (激动剂) (10)
- Antagonist (拮抗剂) (28)
- Activator (激活剂) (3)
- Modulator (调节剂) (3)
- Blocker (阻断剂) (2)
- 靶点
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- AKT1 (1)
- AKT2 (1)
- AKT3 (1)
- Aurora A (3)
- Aurora B (2)
- Aurora C (1)
- Caspase-1 (4)
- Caspase-10 (3)
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- Caspase-4 (3)
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- Caspase-8 (3)
- Caspase-9 (3)
- CETP (1)
- COX (1)
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- ERK5 (1)
- HDAC (1)
- HDAC4 (1)
- HDAC5 (1)
- MEK1 (2)
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- MEK5 (1)
- Pan-Caspase (2)
- PARP1 (1)
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