“No”的搜索结果

产品 1 到 50 共 2783个

每页
页面:
  1. 1
  2. 2
  3. 3
  4. 4
  5. 5

设置降序顺序
  1. Guanosine 5'-triphosphate trisodium salt

    Catalog No. A18283
    Quick View
    Guanosine 5'-triphosphate trisodium salt (5'-GTP trisodium salt) is an activator of signal transduction of G proteins. 了解更多
  2. 6-Diazo-5-oxo-L-nor-Leucine

    Catalog No. A20846
    Quick View
    6-Diazo-5-oxo-L-norleucine 是一种从链霉菌中分离出来的抗生素,一种 glutaminase 的拮抗剂对cKGA(肾脏型谷氨酰胺酶)的IC50值约为1 mM。 了解更多
  3. Docosahexaenoic Acid

    Catalog No. A18205
    Quick View
    Docosahexaenoic Acid (DHA) is an omega-3 fatty acid abundantly present brain and retina. It can be obtained directly from fish oil and maternal milk. 了解更多
  4. Auranofin

    Catalog No. A18996
    Quick View
    Auranofin is a gold salt classified by the World Health Organization as an antirheumatic agent. It is a gold-thiol complex with anti-inflammatory and immunosuppressive actions. 了解更多
  5. Enocyanin

    Catalog No. A18660
    Quick View
    anthocyanin extracted from grapes
    Enocyanin is an anthocyanin extracted from grapes. Enocyanin shows inhibitory effect on the leucine aminopeptidase, acid phosphatase, γ-glutamyl transpeptidase and esterase activity. 了解更多
  6. Adenosine deaminase

    Catalog No. A19330
    Quick View
    Adenosine deaminase is an enzyme that catalyzes the irreversible deamination of adenosine and 2'-deoxyadenosine to inosine and 2'-deoxyinosine, respectively. 了解更多
  7. Hypotaurine

    Catalog No. A20590
    Quick View
    Hypotaurine (2-aminoethanesulfinic acid), an intermediate in taurine biosynthesis from cysteine in astrocytes, is an endogenous inhibitory amino acid of the glycine receptor. 了解更多
  8. Hyaluronidase

    Catalog No. A18232
    Quick View
    local anesthetic additive
    Hyaluronidase (Hyaluronate 4-glycanohydrolase; Hyaluronoglucosaminidase) is a naturally occurring enzyme that depolymerizes hyaluronic acid by cleavage of glycosidic bonds and has been used as a local anesthetic additive. 了解更多
  9. Avelumab

    Catalog No. A18234
    Quick View
    PD-1/PD-L1
    Avelumab is a fully human IgG1 anti-PD-L1 monoclonal antibody with potential antibody-dependent cell-mediated cytotoxicity. 了解更多
  10. HM-43239

    Catalog No. A20826
    Quick View
    FLT3 inhibitor
    HM-43239 is a Novel Potent Small Molecule FLT3 Inhibitor, in Acute Myeloid Leukemia (AML) with FMS-like Tyrosine Kinase 3 (FLT3) Mutations 了解更多
  11. Cinnamylamine

    Catalog No. A20835
    Quick View
    Cinnamylamine can be used for the preparation of Tranylcypromine, a drug that acts as a nonselective and irreversible inhibitor of the enzyme monoamine oxidase (MAO), and is used as an antidepressant and anxiolytic agent. 了解更多
  12. Peptide 401

    Catalog No. A13913
    Quick View
    Peptide 401, a potent mast cell degranulating factor from bee venom, suppresses the increased vascular permeability due to intradermal injection of various smooth muscle spasmogens (histamine, and 5-HT). 了解更多
  13. Exendin-4

    Catalog No. A21580
    Quick View
    glucagon-like peptide-1 receptor agonist
    Exendin-4 (Exenatide), a 39 amino acid peptide, is a long-acting glucagon-like peptide-1 receptor agonist with an IC50 of 3.22 nM. 了解更多
  14. BI-4020

    Catalog No. A22046
    Quick View
    EGFR inhibitor
    BI-4020 is an orally active, non-covalent EGFR inhibitor with IC50 of 0.6 nM and 0.2 nM for EGFR. 了解更多
  15. SR-717

    Catalog No. A22048
    Quick View
    non-nucleotide STING agonist
    SR-717 is a non-nucleotide STING agonist with EC50s of 2.1 μM and 2.2 μM in ISG-THP1 (WT) and ISG-THP1 cGAS KO (cGAS KO) cell lines, respectively. 了解更多
  16. DT2216

    Catalog No. A22050
    Quick View
    BCL-XL degrader
    DT2216 is a potent and selective BCL-XL degrader based on PROTAC technology. 了解更多
  17. BMVC-8C3O

    Catalog No. A22052
    Quick View
    DNA G-quadruplexe (G4) ligand
    BMVC-8C3O is a DNA G-quadruplexe (G4) ligand which can induce topological conversion of non-parallel to parallel forms in human telomeric DNA G4s. 了解更多
  18. LC3-mHTT-IN-AN1

    Catalog No. A22054
    Quick View
    mHTT-LC3 linker compound
    LC3-mHTT-IN-AN1 (Compound AN1) is a mHTT-LC3 linker compound, which interacts with both mutant huntingtin protein (mHTT) and LC3B but not with wtHTT or irrelevant control proteins. 了解更多
  19. APX-115 free base

    Catalog No. A22055
    Quick View
    pan NADPH oxidase (Nox) inhibitor
    APX-115 free base (Ewha-18278 free base) is a potent, orally active pan NADPH oxidase (Nox) inhibitor with Ki values of 1.08 μM, 0.57 μM, and 0.63 μM for Nox1, Nox2 and Nox4, respectively. 了解更多
  20. H-β-Ala-AMC TFA

    Catalog No. A22059
    Quick View
    substrate for aminopeptidase
    H-β-Ala-AMC TFA is a substrate for aminopeptidase. 了解更多
  21. PF9601N

    Catalog No. A22075
    Quick View
    monoamine oxidase B inhibitor
    PF9601N is a selective and potent monoamine oxidase B inhibitor that exhibit anti-Parkinsonian effects in several models of PD. 了解更多
  22. HA155

    Catalog No. A22079
    Quick View
    Autotaxin Inhibitor IV
    HA155, also known as Autotaxin Inhibitor IV, is a boronic acid-based compound that inhibits autotaxin (IC50 = 5.7 nM) by selectively binding to its catalytic threonine. 了解更多
  23. BMS453

    Catalog No. A22082
    Quick View
    RARβ agonist
    BMS453 (BMS-189453), a synthetic retinoid, is a RARβ agonist and a RARα/RARγ antagonist. 了解更多
  24. MCC950

    Catalog No. A22097
    Quick View
    inhibitor of NLRP3 (NOD-like receptor (NLR) family
    MCC950 (CP-456773, CRID3) is a potent and selective inhibitor of NLRP3 (NOD-like receptor (NLR) family, pyrin domain-containing protein 3) with IC50 of 7.5 nM and 8.1 nM in BMDMs and HMDMs, respectively. 了解更多
  25. Creatine riboside

    Catalog No. A22112
    Quick View
    urinary metabolite
    Creatine riboside is a urinary metabolite and is a diagnostic and prognostic biomarker of lung cancer. 了解更多
  26. ONO-8130

    Catalog No. A22113
    Quick View
    antagonist of EP1 receptor
    ONO-8130 is an orally available antagonist of EP1 receptor. 了解更多
  27. FLTX1

    Catalog No. A22120
    Quick View
    antiestrogenic properties
    FLTX1 is a fluorescent Tamoxifen derivative that can specifically label intracellular Tamoxifen-binding sites (estrogen receptors) under permeabilized and non-permeabilized conditions. FLTX1 exhibits the potent antiestrogenic properties of Tamoxifen in breast cancer cells. FLTX1 is devoid of the estrogenic agonistic effect on the uterus. 了解更多
  28. ML198

    Catalog No. A22122
    Quick View
    activator and non-inhibitory chaperone of glucocerebrosidase
    ML198 is a novel activator and non-inhibitory chaperone of glucocerebrosidase. 了解更多
  29. BMS-986188

    Catalog No. A22124
    Quick View
    Positive Allosteric Modulator of the delta-Opioid Receptor
    BMS-986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor. 了解更多
  30. NCGC607

    Catalog No. A22126
    Quick View
    noninhibitory chaperone
    NCGC607 is a a noninhibitory chaperone of glucocerebrosidase (GCase). 了解更多
  31. BGC201531

    Catalog No. A22130
    Quick View
    EP4 antagonist
    BGC201531, also known as GTPL3380 and AP-1531, is a EP4 antagonist for the treatment of acute migraine. 了解更多
  32. Statil

    Catalog No. A22132
    Quick View
    aldose reductase inhibitor
    Ponalrestat, also known as MK-538, is an aldose reductase inhibitor. 了解更多
  33. MDK-1088

    Catalog No. A22133
    Quick View
    Trypanosoma cruzi inhibitor
    MDK-1088 (T.cruzi Inhibitor) is a Trypanosoma cruzi inhibitor. 了解更多
  34. MSA-2

    Catalog No. A22139
    Quick View
    non-nucleotide STING agonist
    MSA-2, a potent and orally available non-nucleotide STING agonist, is bound to STING as a noncovalent dimer with nanomolar affinity. 了解更多
  35. GNE-140 racemic

    Catalog No. A22146
    Quick View
    lactate dehydrogenase (LDHA) inhibitor
    GNE-140 racemic is a novel potent lactate dehydrogenase (LDHA) inhibitor. 了解更多
  36. AA41612

    Catalog No. A22147
    Quick View
    antagonist of melanopsin-mediated phototransduction
    AA41612 is an antagonist of melanopsin-mediated phototransduction. 了解更多
  37. Simetride

    Catalog No. A22153
    Quick View
    non-narcotic analgesic
    Simetride, a non-narcotic analgesic, is an ingredient of Kyorin AP2 which is used to treat low back pain, symptomatic neuralgia, headache, menstrual pain and etc. 了解更多
  38. Adenosine amine congener

    Catalog No. A22193
    Quick View
    A1 adenosine receptor agonist
    Adenosine amine congener (ADAC) is a selective A1 adenosine receptor agonist, can ameliorate noise- and Cisplatin-induced cochlear injury. 了解更多
  39. SR-31747 free base

    Catalog No. A22199
    Quick View
    immunosuppressive and anti-inflammatory properties
    SR-31747 free base is a sigma ligand with immunosuppressive and anti-inflammatory properties. 了解更多
  40. PF-06835919

    Catalog No. A22266
    Quick View
    ketohexokinase (KHK) inhibitor
    PF-06835919, also known as MDK1846, is a potent ketohexokinase (KHK) inhibitor. 了解更多
  41. Sodium oxamate

    Catalog No. A22275
    Quick View
    LDH inhibitor
    Sodium oxamate (SO, Aminooxoacetic acid, Oxamic acid) is an inhibitor of lactate dehydrogenase (LDH) that specificly inhibits LDH?A. 了解更多
  42. Motixafortide

    Catalog No. A22276
    Quick View
    CXCR4 antagonist
    Motixafortide (BKT140 4-fluorobenzoyl) is a novel CXCR4 antagonist with an IC50 vakue of ??1 nM. 了解更多
  43. HA-100 dihydrochloride

    Catalog No. A22289
    Quick View
    PKs inhibitor
    HA-100 is an isoquinoline compound with an added piperazinylsulfonyl group that acts as an inhibitor of protein kinases (PKs), including PKA, PKC, and PKG (IC50s = 8, 12, and 4 ?M, respectively). 了解更多
  44. 3-Hydroxyanthranilic acid

    Catalog No. A22292
    Quick View
    immunomodulatory agent
    3-Hydroxyanthranilic Acid (3-HAA, 3-HANA), a tryptophan metabolite, has an immunomodulatory effect that may result from inhibition of PI3K/Akt/mTOR and NF-κB activity, thereby decreasing the production of pro-inflammatory mediators. 了解更多
  45. Acetosyringone

    Catalog No. A22294
    Quick View
    anti-inflammatory agent
    Acetosyringone is a phenolic natural product with analgesic, antipyretic and anti-inflammatory actions. 了解更多
  46. BD750

    Catalog No. A22300
    Quick View
    JAK3/STAT5 inhibitor
    BD750, an effective immunosuppressant and a JAK3/STAT5 inhibitor, inhibits IL-2-induced JAK3/STAT5-dependent T cell proliferation, with IC50 values of 1.5 μM and 1.1 μM in mouse and human T cells, respectively. 了解更多
  47. SRX3207

    Catalog No. A22305
    Quick View
    Syk/PI3K inhibitor
    SRX3207 is an orally active and first-in-class dual Syk/PI3K inhibitor, with IC50 values of 10.7 nM and 861 nM for Syk and PI3Kα, respectively. SRX3207 relieves tumor immunosuppression. 了解更多
  48. BpV(HOpic)

    Catalog No. A22308
    Quick View
    PTEN inhibitor
    BpV(HOpic) is a potent and selective inhibitor of PTEN with an IC50 of 14 nM. Nanocarrier-BpV(HOpic) has neuroprotective activity. 了解更多
  49. Ferulic acid sodium

    Catalog No. A22310
    Quick View
    FGFR1 inhibitor
    Ferulic acid sodium is a novel fibroblast growth factor receptor 1 (FGFR1) inhibitor with IC50s of 3.78 and 12.5 μM for FGFR1 and FGFR2, respectively. 了解更多
  50. Loureirin A

    Catalog No. A22313
    Quick View
    flavonoid
    Loureirin A is a flavonoid extracted from Dragon's Blood, can inhibit Akt phosphorylation, and has antiplatelet activity. 了解更多

产品 1 到 50 共 2783个

每页
页面:
  1. 1
  2. 2
  3. 3
  4. 4
  5. 5

设置降序顺序
Rewards