“inhibitor”的搜索结果

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  1. Histone Acetyltransferase Inhibitor II

    Catalog No. A12331
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    cell permeable p300 inhibitor
    Histone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 ?M; Histone Acetyltransferase Inhibitor II can be used in cancer research. 了解更多
  2. Src Inhibitor 1

    Catalog No. A12299
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    Src tyrosine kinase inhibitor
    Src Inhibitor 1 is a potent and selective dual site Src tyrosine kinase inhibitor with IC50 values of 44 nM for Src and 88nM for Lck. 了解更多
  3. CPA inhibitor

    Catalog No. A11369
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    CPA inhibitor
    CPA inhibitor is a potent inhibitor for carboxypeptidase A (CPA). 了解更多
  4. GSK3 Inhibitor XIII

    Catalog No. A22128
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    ATP-binding site inhibitor of GSK-3
    GSK3 Inhibitor XIII (GSK3i XIII) is an ATP-binding site inhibitor of GSK-3. 了解更多
  5. ATR inhibitor 2

    Catalog No. A22162
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    ATR inhibitor
    ATR inhibitor 2 is an ATP-competitive, orally active, and selective ATR inhibitor, with a Ki of <150 pM. 了解更多
  6. LMPTP INHIBITOR 1 dihydrochloride

    Catalog No. A22227
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    LMPTP inhibitor
    LMPTP INHIBITOR 1 (dihydrochloride) is a selective inhibitor of low molecular weight protein tyrosine phosphatase (LMPTP), with an IC50 of 0.8 μM LMPTP-A. 了解更多
  7. VPS34 inhibitor 1 (Compound 19)

    Catalog No. A22378
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    VPS34 inhibitor
    VPS34 inhibitor 1 (Compound 19, PIK-III analogue) is a potent and selective inhibitor of VPS34 with an IC50 of 15 nM. 了解更多
  8. Selective PI3Kδ Inhibitor 1 (compound 7n)

    Catalog No. A22381
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    PI3Kδ inhibitor
    Selective PI3Kδ Inhibitor 1 (compound 7n) is an inhibitor of PI3Kδ with an IC50 of 0.9 nM and >1000-fold selectivity against other class I PI3K isoforms [PI3K α/γ/β=3670/1460/21300 nM]. 了解更多
  9. BTK inhibitor 1 (Compound 27)

    Catalog No. A22445
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    BTK inhibitor
    BTK inhibitor 1 (compound 27) is an inhibitor of BTK with an IC50 of 0.11 nM for Btk and inhibits B cell activation in hWB with an IC50 of 2 nM. 了解更多
  10. Multi-kinase inhibitor 1

    Catalog No. A22645
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    multi-kinase inhibitor
    Multi-kinase inhibitor 1 is a potent multi-kinase inhibitor. Multi-kinase inhibitor 1 has the potential for diseases or disorders associated with abnormal or deregulated tyrosine kinase activity, particularly diseases associated with the activity of PDGF-R, c-Kit and Bcr-abl. 了解更多
  11. Diacylglycerol acyltransferase inhibitor-1

    Catalog No. A20315
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    DGAT1 inhibitor
    Diacylglycerol acyltransferase inhibitor-1 is a diacylglycerol acyltransferase (DGAT1) inhibitor. 了解更多
  12. MAT2A inhibitor 2

    Catalog No. A20171
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    MAT2A inhibitor
    MAT2A inhibitor 2 is a methionine adenosyltransferase 2A (MAT2A) inhibitor. 了解更多
  13. DAAO inhibitor-1

    Catalog No. A20117
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    DAAO inhibitor
    DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor with an IC50 of 0.12 μM. 了解更多
  14. Grp94 Inhibitor-1

    Catalog No. A20073
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    Grp94 inhibitor
    Grp94 Inhibitor-1 is a potent, selective Grp94 inhibitor with an IC50 value of 2 nM, and over 1000-fold selectivity to Grp94 against Hsp90α. 了解更多
  15. mTOR inhibitor-1

    Catalog No. A20029
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    mTOR inhibitor
    mTOR inhibitor-1 is a novel mTOR pathway inhibitor which can suppress cells proliferation and inducing autophagy. 了解更多
  16. Tubulin inhibitor 1

    Catalog No. A19998
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    tubulin inhibitor
    Tubulin inhibitor 1 is a tubulin inhibitor, inhibits tubulin polymerization. 了解更多
  17. YAP/TAZ inhibitor-1

    Catalog No. A19976
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    YAP/TAZ inhibitor
    YAP/TAZ inhibitor-1 is a YAP/TAZ inhibitor extracted from patent WO2017058716A1, Compound 1, has an IC50 of <0.100 μμ in firefly luciferase assay. 了解更多
  18. SIRT5 inhibitor 1

    Catalog No. A19841
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    SIRT5 inhibitor
    SIRT5 inhibitor 1 is a potent Human Sirtuin 5 deacylase inhibitor, with an IC50 of 0.11 μM. 了解更多
  19. BET bromodomain inhibitor

    Catalog No. A19831
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    BET inhibitor
    BET bromodomain inhibitor is a potent BET inhibitor extracted from patent WO/2015/153871A2, compound example 11. 了解更多
  20. TRAF-STOP inhibitor 6877002

    Catalog No. A19758
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    CD40-TRAF6 interaction inhibitor
    TRAF-STOP inhibitor 6877002, is a selective inhibitor of CD40-TRAF6 interaction, compound VII, shows inhibition of NF-κB activation in RAW cells, extracted from patent WO2014033122A1. 了解更多
  21. Glutaminyl Cyclase Inhibitor 1

    Catalog No. A19723
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    glutaminyl cyclase inhibitor
    Glutaminyl Cyclase Inhibitor 1 is a glutaminyl cyclase inhibitor with an IC50 of 0.5 μM. 了解更多
  22. PKC-theta inhibitor

    Catalog No. A19712
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    PKC-θ inhibitor
    PKC-theta inhibitor is a selective PKC-θinhibitor, with an IC50 of 12 nM. 了解更多
  23. LRRK2 inhibitor 1

    Catalog No. A19701
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    LRRK2 inhibitor
    LRRK2 inhibitor 1 is a potent, selective and oral LRRK2 inhibitor with an pIC50 of 6.8 nM. 了解更多
  24. PDGFRα kinase inhibitor 1

    Catalog No. A19632
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    type II PDGFRα kinase inhibitor
    PDGFRα kinase inhibitor 1 is a highly selective type II PDGFRα kinase inhibitor with IC50s of 132 nM and 6115 nM for PDGFRα and PDGFRβ, respectively. 了解更多
  25. HIV-1 integrase inhibitor 3

    Catalog No. A19628
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    INST inhibitor
    HIV-1 integrase inhibitor 3 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 2.7 nM. 了解更多
  26. PI3K/mTOR Inhibitor-2

    Catalog No. A19621
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    dual pan-PI3K/mTOR inhibitor
    PI3K/mTOR Inhibitor-2 is a potent dual pan-PI3K/mTOR inhibitor with IC50s of 3.4/34/16/1 nM for PI3Kα/PI3Kβ/PI3Kδ/PI3Kγ and 4.7 nM for mTOR. Antitumor activity. 了解更多
  27. HIV-1 integrase inhibitor 4

    Catalog No. A19617
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    INST inhibitor
    HIV-1 integrase inhibitor 4 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 3.7 nM. 了解更多
  28. Neurotoxin Inhibitor

    Catalog No. A19507
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    neurotoxin inhibitor
    Neurotoxin Inhibitor is a neurotoxin inhibitor. 了解更多
  29. Aurora Kinase Inhibitor 3

    Catalog No. A19448
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    Aurora A kinase inhibitor
    Aurora Kinase Inhibitor 3 is a strong and selective Aurora A kinase inhibitor with an IC50 of 42 nM, and weakly inhibits EGFR with an IC50>10 μM. 了解更多
  30. p38α inhibitor 1

    Catalog No. A19182
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    p38α inhibitor
    p38α inhibitor 1 is a p38α inhibitor extracted from patent WO 2008076265 A1. 了解更多
  31. Bromodomain inhibitor-8

    Catalog No. A19161
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    BET bromodomain inhibitor
    Bromodomain inhibitor-8 (Intermediate 21) is a BET bromodomain inhibitor for treating autoimmune and inflammatory diseases. 了解更多
  32. FAAH inhibitor 1

    Catalog No. A21841
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    FAAH inhibitor
    FAAH inhibitor 1 (Benzothiazole analog 3) is a potent fatty acid amide hydrolase (FAAH) inhibitor with an IC50 of 18??8 nM. 了解更多
  33. B-Raf inhibitor 1 dihydrochloride

    Catalog No. A21834
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    Raf kinase inhibitor
    B-Raf inhibitor 1 dihydrochloride is a potent Raf kinase inhibitor with Kis of 1 nM, 1 nM, and 0.3 nM for B-RafWT, B-RafV600E, and C-Raf, respectively. 了解更多
  34. Notch inhibitor 1

    Catalog No. A21591
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    Notch inhibitor
    Notch inhibitor 1 is a potent Notch inhibitor, with IC50s of 7.8 and 8.5 nM for Notch 1 and Notch 3, respectively. Used in the research of cancer. 了解更多
  35. β-Secretase Inhibitor IV

    Catalog No. A21346
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    BACE-1 inhibitor
    β-Secretase Inhibitor IV is a potent, cell-active BACE-1 inhibitor with IC50s of 15.6 and 16.3nM under BACE-1 concentrations of 2 nM and 100 pM, respectively. 了解更多
  36. HIV-1 integrase inhibitor 2

    Catalog No. A11447
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    HIV-1 integrase inhibitor
    HIV-1 integrase inhibitor 2, in the treatment of human immunodeficiency virus (HIV) infection. 了解更多
  37. HIV-1 integrase inhibitor

    Catalog No. A11446
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    HIV-1 integrase inhibitor
    HIV-1 integrase inhibitor is uesful for anti-HIV. 了解更多
  38. P-gp inhibitor 1

    Catalog No. A13384
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    P-gp inhibitor
    P-gp inhibitor 1 is a novel inhibitor reversing P-glycoprotein-mediated multidrug resistance. 了解更多
  39. PDE-9 inhibitor

    Catalog No. A11532
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    PDE-9 inhibitor
    PDE-9 inhibitor is useful for neurodegenerative diseases. 了解更多
  40. MMP3 inhibitor 1

    Catalog No. A13185
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    MMP-3 inhibitor
    MMP3 inhibitor 1 is a potent and highly selective MMP-3 inhibitor with an IC50 of 1 nM. 了解更多
  41. Top1 inhibitor 1

    Catalog No. A13304
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    human topoisomerase I (Top1) inhibitor
    Top1 inhibitor 1 (compound 28) is a potent human topoisomerase I (Top1) inhibitor with an IC50 value of 29 nM. 了解更多
  42. HPGDS inhibitor 2

    Catalog No. A18390
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    H-PGDS 抑制剂
    HPGDS inhibitor 2 is a highly potent and selective hematopoietic prostaglandin D synthase (H-PGDS) inhibitor with an IC50 of 9.9 nM. 了解更多
  43. IDH1 Inhibitor 2

    Catalog No. A18420
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    IDH1 inhibitor
    DH1 Inhibitor 2 is a potent IDH1 inhibitor via a direct covalent modification of His315, with an IC50 of 110 nM. 了解更多
  44. KRAS G12C inhibitor 17

    Catalog No. A18441
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    KRAS G12C inhibitor
    KRAS G12C inhibitor 17 is a potent KRAS G12C inhibitor extracted from patent WO2019110751A1, compound 82, has an IC50 of 5 nM. 了解更多
  45. KRAS G12C inhibitor 16

    Catalog No. A18444
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    KRAS G12C inhibitor
    KRAS G12C inhibitor 16 is a potent KRAS G12C inhibitor extracted from patent WO2019110751A1, compound 39, has an IC50 of 97 nM. 了解更多
  46. KRAS G12C inhibitor 15

    Catalog No. A18447
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    KRAS G12C inhibitor
    KRAS G12C inhibitor 15 is a potent KRAS G12C inhibitor extracted from patent WO2019110751A1, compound 22, has an IC50 of 5 nM. 了解更多
  47. PARP14 inhibitor H10

    Catalog No. A18616
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    PARP14 抑制剂
    PARP14 inhibitor H10, compound H 10, is a selective inhibitor against PARP14 (IC50=490 nM), over other PARPs (??24 fold over PARP1). PARP14 inhibitor H10 induces caspase-3/7-mediated cell apoptosis. 了解更多
  48. BRD4 Inhibitor-10

    Catalog No. A18679
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    BRD4-BD1 inhibitor
    BRD4 Inhibitor-10 is a potent BRD4-BD1 inhibitor extracted from patent WO2015022332A1, Compound II-25, has an IC50 of 8 nM. 了解更多
  49. KRAS G12C inhibitor 5

    Catalog No. A18840
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    KRas G12C inhibitor
    KRAS G12C inhibitor 5 is a KRas G12C inhibitor extracted from patent WO2017201161A1, Compound example 147. 了解更多
  50. Tuberculosis inhibitor 1

    Catalog No. A18906
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    trypanosoma brucei growth inhibitor
    Tuberculosis inhibitor 1 is a potent and non-cytotoxic trypanosoma brucei growth inhibitor with an EC50 of 5 nM. 了解更多

产品 1 到 50 共 5361个

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