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  1. LDN-193189 2HCl

    Catalog No. A22307
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    BMP signaling inhibitor
    LDN193189 HCl (DM-3189) is the hydrochloride salt of LDN193189, which is a selective BMP signaling inhibitor, and inhibits the transcriptional activity of the BMP type I receptors ALK2 and ALK3 with IC50 of 5 nM and 30 nM in C2C12 cell lines, respectively, 200-fold selectivity for BMP versus TGF-β. 了解更多
  2. UK-371804 HCl

    Catalog No. A22379
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    uPA inhibitor
    UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin). 了解更多
  3. Polymyxin B nonapeptide

    Catalog No. A20168
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    Polymyxin B nonapeptide is a cyclic peptide obtained from Polymyxin B by proteolytic removal of its terminal amino acyl residue. Polymyxin B nonapeptide is less toxic, lacks bactericidal activity, and retains its ability to render gram-negative bacteria susceptible to several antibiotics by permeabilizing their outer membranes. 了解更多
  4. Gefapixant

    Catalog No. A19254
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    P2X3R antagonist
    Gefapixant is an orally active P2X3 receptor (P2X3R) antagonist with IC50s of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors. 了解更多
  5. Momelotinib Mesylate

    Catalog No. A21658
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    JAK1/JAK2 inhibitor
    Momelotinib Mesylate (CYT387 Mesylate) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, appr 10-fold selectivity versus JAK3. 了解更多
  6. CDKI-73

    Catalog No. A21467
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    CDK9 inhibitor
    CDKI-73 is a potent CDK9 inhibitor with Ki of 4 nM; shows selective toxicity to CLL cells(LD50=80 nM) versus normal B cell and normal CD34+ cell(LD50>20 uM). 了解更多
  7. CHIR-99021 monohydrochloride

    Catalog No. A21430
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    GSK-3α/β inhibitor
    CHIR-99021 monohydrochloride (CT99021 monohydrochloride) is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM; > 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2, as well as other protein kinases. 了解更多
  8. Tonapofylline

    Catalog No. A21328
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    adenosine A1 receptor antagonist
    Tonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure. 了解更多
  9. Irosustat

    Catalog No. A21287
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    steroid sulfatase inhibitor
    Irosustat is a potent steroid sulfatase inhibitor, with an IC50 of 8 nM, and exhibits anti-breast cancer activity. 了解更多
  10. AZD8329

    Catalog No. A21081
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    11β-HSD1 inhibitor
    AZD8329 is a potent 11β-Hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor with an IC50 of 9 nM for human 11β-HSD1, displays excellent selectivity versus 11β-HSD2, 17β-HSD1 and 17β-HSD3. 了解更多
  11. Ruxolitinib sulfate

    Catalog No. A11467
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    JAK1/2 inhibitor
    Ruxolitinib sulfate (INCB018424 sulfate) is the first potent, selective JAK1/2 inhibitor to enter the clinic with IC50s of 3.3 nM/2.8 nM, and has > 130-fold selectivity for JAK1/2 versus JAK3. 了解更多
  12. Vancomycin hydrochloride

    Catalog No. A16781
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    Vancomycin hydrochloride is an antibiotic for the treatment of bacterial infections. It acts by inhibiting the second stage of cell wall synthesis of susceptible bacteria. 了解更多
  13. MAC glucuronide phenol-linked SN-38

    Catalog No. A18403
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    DNA topoisomerase I inhibitor
    MAC glucuronide phenol-linked SN-38 is a pH-susceptible lactone MAC glucuronide phenol-linked SN-38 (DNA topoisomerase I inhibitor) drug linker. MAC glucuronide phenol-linked SN-38 is cytotoxic across L540cy cells and Ramos cells with IC50 values of 113 and 67 ng/mL, respectively. 了解更多
  14. NaV1.7 inhibitor-1

    Catalog No. A18933
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    NaV 1.7 inhibitor
    NaV1.7 inhibitor-1 is an efficacious voltage-gated sodium channel (NaV) 1.7 inhibitor with an IC50 of 0.6 nM for hNaV1.7, exhibits 80-fold selectivity versus hNaV1.5. 了解更多
  15. SRT 1460

    Catalog No. A19026
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    SIRT1 activator
    SRT 1460, a potent Sirtuin-1 (SIRT1) activator with an EC1.5 value of 2.9 μM, shows good selectivity for activation of SIRT1 versus SIRT2 and SIRT3 (EC1.5>300 μM), and is more potent than Resveratrol and the closest sirtuin homologues. 了解更多
  16. Penicillin V potassium salt

    Catalog No. A17915
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    broad-spectrum penicillin antibiotic
    Penicillin V potassium is a broad-spectrum penicillin antibiotic used orally in the treatment of mild to moderate infections by susceptible gram-positive organisms. 了解更多
  17. Bendazac

    Catalog No. A17607
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    anticataract drug
    Bendazac, also known as Bendazolic acid and AF-983, is an anticataract drug. It has been reported that Bendazac acts by preventing protein denaturation. 了解更多
  18. AZD4573

    Catalog No. A18321
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    CDK9 inhibitor
    AZD4573 is a potent and selective inhibitor of CDK9, with fast-off binding kinetics and high selectivity versus other kinases, including other CDK family kinases. 了解更多
  19. Rantes Rhesus Macaque

    Catalog No. AP5755
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    Rantes Rhesus Macaque Recombinant (CCL5) 了解更多
  20. IP 10 Rhesus macaque

    Catalog No. AP5682
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    IP-10 Rhesus macaque Recombinant (CXCL10) 了解更多
  21. IL 8 Rhesus Macaque

    Catalog No. AP5674
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    Interleukin-8 Rhesus Macaque Recombinant 了解更多
  22. Eotaxin Rhesus Macaque

    Catalog No. AP5638
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    Eotaxin Rhesus Macaque Recombinant (CCL11) 了解更多
  23. TNF a Rhesus Macaque

    Catalog No. AP5575
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    Tumor Necrosis Factor-Alpha Rhesus Macaque Recombinant 了解更多
  24. SAA1 Monkey

    Catalog No. AP5530
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    Serum Amyloid A (APO-SAA1) Rhesus Macaque Recombinant 了解更多
  25. IL 1 alpha Rhesus Macaque

    Catalog No. AP5454
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    Interleukin-1 alpha Rhesus Macaque Recombinant 了解更多
  26. IL 5 Rhesus Macaque

    Catalog No. AP5451
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    Interleukin-5 Rhesus Macaque Recombinant 了解更多
  27. IL 1 beta Monkey

    Catalog No. AP5439
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    Interleukin-1 beta Rhesus Macaque Recombinant 了解更多
  28. IL 13 Rhesus Macaque

    Catalog No. AP5325
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    Interleukin-13 Rhesus Macaque Recombinant 了解更多
  29. IL 6 Rhesus Macaque

    Catalog No. AP5324
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    Interleukin-6 Rhesus Macaque Recombinant 了解更多
  30. IL 4 Rhesus Macaque

    Catalog No. AP5322
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    Interleukin-4 Rhesus Macaque Recombinant 了解更多
  31. IL 3 Rhesus Macaque

    Catalog No. AP5314
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    Interleukin-3 Rhesus Macaque Recombinant 了解更多
  32. IL 16 Rhesus Macaque

    Catalog No. AP5312
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    Interleukin-16 Rhesus Macaque Recombinant 了解更多
  33. Flt3-Ligand Rhesus Macaque

    Catalog No. AP5205
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    Flt3-Ligand Rhesus Macaque Recombinant 了解更多
  34. DUT Pyrococcus Fruriosus

    Catalog No. AP4457
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    Thermostable dUTPase Pyrococcus Fruriosus Recombinant 了解更多
  35. GM CSF Monkey

    Catalog No. AP3366
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    Granulocyte Macrophage-Colony Stimulating Factor Rhesus Macaque Recombinant 了解更多
  36. Procalcitonin Rhesus

    Catalog No. AP3309
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    Procalcitonin Rhesus Recombinant 了解更多
  37. TSG101 Human

    Catalog No. AP2216
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    Tumor Susceptibility Gene 101 Human Recombinant 了解更多
  38. S100b Rhesus Macaque

    Catalog No. AP0438
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    S100 Calcium Binding Protein B Rhesus Macaque Recombinant 了解更多
  39. Ciwujianoside-B

    Catalog No. A14603
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    Ciwujianoside B是从Eleutherococcus senticosus 叶中分离出来的,口服后能够渗透并在大脑中起作用。Ciwujianoside B显着增强识别记忆的能力。 了解更多
  40. Paliperidone

    Catalog No. A10691
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    Dopamine Receptor 拮抗剂
    Paliperidone (Invega)是一种非典型的抗精神病药。 了解更多

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