“jwh 250”的搜索结果

产品 51 到 100 共 1231个

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  1. Pseudolaric Acid B

    Catalog No. A12102
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    anti-fungal agent
    Pseudolaric Acid B, a natural diterpenoid compound isolated from the root and trunk bark of Pseudolaric kaempferi Gordon, has anti-fungal and anti-fertility properties. 了解更多
  2. CFI-402257

    Catalog No. A12037
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    TTK inhibitor
    CFI-402257, a pyrazolopyridin derivative, has been found to be a TTK inhibitor that could influence chromosome segregation and induce cell death so that is significant in anticancer studies. 了解更多
  3. Adooq Payment Adjustment

    Catalog No. ADQPA
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    It is for the online credit card payment only, not for any product order placement. 了解更多
  4. GC7 Sulfate

    Catalog No. A22035
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    DHPS inhibitor
    GC7 Sulfate is a deoxyhypusine synthase (DHPS) inhibitor. 了解更多
  5. Sograzepide

    Catalog No. A22020
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    Gastrin/CCK-B antagonist
    Sograzepide (Netazepide; YF 476; YM-220) is an extremely potent , highly selective and orally active Gastrin/CCK-B antagonist with an IC50 value of 0.1 nM, has inhibitory effect on Gastrin/CCK-A activity with an IC50 of 502 nM. 了解更多
  6. Bisindolylmaleimide X hydrochloride

    Catalog No. A22010
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    PKC inhibitor
    Bisindolylmaleimide X hydrochloride (BIM-X hydrochloride) is a potent and selective protein kinase C (PKC) inhibitor. 了解更多
  7. Deschloroclozapine

    Catalog No. A20801
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    dual dopamine and serotonin receptor antagonist
    Deschloroclozapine is a dual dopamine and serotonin receptor antagonist with Kis of 200, 2500, 420, 39, 84, 40 nM for dopamine D1, D2,D4, and serotonin S2A, S2C, S3, respectively. 了解更多
  8. Ro-24-4736

    Catalog No. A20717
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    PAF antagonist
    Ro 24-4736 is a potent, selective, p.o.-active platelet-activating factor (PAF) antagonist with a long duration of action. 了解更多
  9. NSP-805

    Catalog No. A20716
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    PDE3 inhibitor
    NSP-805 is a potent and selective inhibitor of guinea pig cardiac phosphodiesterase 3 (PDE3), and a cardiotonic agent with vasodilator properties. 了解更多
  10. E-982

    Catalog No. A20698
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    E-982 is extracted from the reference, compound 12. 了解更多
  11. EED226

    Catalog No. A20673
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    PRC2 inhibitor
    EED226 is a polycomb repressive complex 2 (PRC2) inhibitor, which binds to the K27me3-pocket on embryonic ectoderm development (EED) and shows strong antitumor activity in xenograft mice model. 了解更多
  12. Azeliragon

    Catalog No. A20622
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    RAGE inhibitor
    Azeliragon (TTP488) is an orally bioavailable inhibitor of the receptor for advanced glycation end products (RAGE) in development as a potential treatment to slow disease progression in patients with mild Alzheimer??s disease (AD). Azeliragon also can cross the blood-brain barrier (BBB). 了解更多
  13. Allopurinol riboside

    Catalog No. A20572
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    Allopurinol riboside, a metabolite of allopurinol, shows potent activities against parasites. 了解更多
  14. ICI 153110

    Catalog No. A20513
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    phosphodiesterase inhibitor
    ICI 153110 is an orally active phosphodiesterase inhibitor with both vasodilating and inotropic properties which is designed for the treatment of congestive cardiac failure. 了解更多
  15. Cadazolid

    Catalog No. A20481
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    oxazolidinone antibiotic
    Cadazolid (ACT-179811) is a new oxazolidinone antibiotic with potent activity against Clostridium difficile. 了解更多
  16. TM5275 sodium

    Catalog No. A20462
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    plasminogen activator inhibitor
    TM5275 sodium is a plasminogen activator inhibitor (PAI-1) with an IC50 of 6.95 μM. 了解更多
  17. beta-L-D4A

    Catalog No. A20444
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    HIV-1 reverse transcriptase inhibitor
    beta-L-D4A is a nucleoside HIV-1 reverse transcriptase inhibitor. 了解更多
  18. Sulfasymazine

    Catalog No. A20435
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    Sulfasymazine is a sulfonamide drug and displays antibacterial properties. 了解更多
  19. TPI-1

    Catalog No. A20423
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    SHP-1 inhibitor
    TPI-1, also known as Tyrosine Phosphatase Inhibitor 1, is a SHP-1 inhibitor; inhibits recombinant SHP-1 with an IC50 of 40 nM. 了解更多
  20. BGG463

    Catalog No. A20420
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    CDK2 inhibitor
    BGG463 (K03859) is an orally active type II CDK2 inhibitor. 了解更多
  21. Xenalamine

    Catalog No. A20411
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    Xenalamine is a synthetic antiviral agent. 了解更多
  22. Tomivosertib

    Catalog No. A20407
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    MNK1/MNK2 inhibitor
    Tomivosertib (eFT508) is a potent, highly selective, and orally bioavailable MNK1 and MNK2 inhibitor, with IC50s of 1-2 nM against both isoforms. 了解更多
  23. ML329

    Catalog No. A20401
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    MITF inhibitor
    ML329 is a micropthalmia-associated transcription factor (MITF) inhibitor, which inhibits TRPM-1 promoter activity with an IC50 of 1.2 μM. 了解更多
  24. Revizinone

    Catalog No. A20398
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    PDE inhibitor
    Revizinone is a novel selective phosphodiesterase (PDE) inhibitor with IC50 values on this enzyme to 0.036 microM. 了解更多
  25. B220

    Catalog No. A20391
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    B220 is an antiviral agent which can inhibit the growth of HSV-1, HSV-2 and human cytomegalovirus (CMV). 了解更多
  26. DMU2105

    Catalog No. A20389
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    CYP1B1 inhibitor
    DMU2105 is a potent and specific CYP1B1 inhibitor, with IC50s of 10 nM and 742 nM for CYP1B1 and CYP1A1, respectively. 了解更多
  27. SAR-20347

    Catalog No. A20380
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    TYK2/JAK1/JAK2/JAK3 inhibitor
    SAR-20347 is an inhibitor of TYK2, JAK1, JAK2 and JAK3 with IC50s of 0.6, 23, 26 and 41 nM, respectively. 了解更多
  28. RMI 10874

    Catalog No. A20370
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    RMI 10874 is a tilorone analogue. Tilorone is a small-molecule, orally bioavailable antiviral agent. RMI 10874 completely abolishes lung colonization of an H-2 negative (GR9.B9) MCA-induced fibrosarcoma clone. 了解更多
  29. RD3-0028

    Catalog No. A20348
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    RSV replication inhibitor
    RD3-0028 is a potent and selective inhibitor of RSV replication with an EC50 of 4.5 μM. 了解更多
  30. Alsterpaullone

    Catalog No. A20318
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    CDK inhibitor
    Alsterpaullone (9-Nitropaullone;NSC 705701) is a potent CDK inhibitor, with IC50s of 35 nM, 15 nM, 200 nM and 40 nM for CDK1/cyclin B, CDK2/cyclin A, CDK2/cyclin E and CDK5/p35, respectively. 了解更多
  31. Diacylglycerol acyltransferase inhibitor-1

    Catalog No. A20315
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    DGAT1 inhibitor
    Diacylglycerol acyltransferase inhibitor-1 is a diacylglycerol acyltransferase (DGAT1) inhibitor. 了解更多
  32. PTI-428

    Catalog No. A20287
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    CFTR amplifier
    PTI-428 is a specific cystic fibrosis transmembrane conductance regulator (CFTR) amplifier. 了解更多
  33. Boc-C1-PEG2-C4-Cl

    Catalog No. A20263
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    Boc-C1-PEG2-C4-Cl (PROTAC Linker 1) is a PROTAC linker utilized to connect the respective tyrosine kinase inhibitor (TKI) to the E3 recruiting ligand. 了解更多
  34. AGI-25696

    Catalog No. A20250
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    MATA2 inhibitors
    AGI-25696 is a methionine adenosyltransferase 2A (MATA2 ) inhibitors useful for treatment of cancer. AGI-25696 blocks growth of MTAP-deleted tumors in vivo. 了解更多
  35. Ziresovir

    Catalog No. A20179
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    RSV F protein inhibitor
    Ziresovir (AK0529;RO-0529) is a potent, selective, and orally bioavailable respiratory syncytial virus (RSV) fusion (F) protein (RSV F) protein inhibitor. 了解更多
  36. MAT2A inhibitor 2

    Catalog No. A20171
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    MAT2A inhibitor
    MAT2A inhibitor 2 is a methionine adenosyltransferase 2A (MAT2A) inhibitor. 了解更多
  37. Ceftobiprole

    Catalog No. A20135
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    Ceftobiprole is a broad-spectrum cephalosporin with activity against Methicillin-resistant staphylococcus aureus (MRSA) with the MIC90 value of 2 mcg/mL. 了解更多
  38. DAAO inhibitor-1

    Catalog No. A20117
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    DAAO inhibitor
    DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor with an IC50 of 0.12 μM. 了解更多
  39. Imiglitazar

    Catalog No. A20080
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    PPARα/ PPARγ1 agonist
    Imiglitazar (TAK559) is a potent and dual human PPARα and PPARγ1 agonist with EC50 values of 67 and 31 nM. 了解更多
  40. mTOR inhibitor-1

    Catalog No. A20029
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    mTOR inhibitor
    mTOR inhibitor-1 is a novel mTOR pathway inhibitor which can suppress cells proliferation and inducing autophagy. 了解更多
  41. NITD-349

    Catalog No. A20026
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    MmpL3 inhibitor
    NITD-349 is an MmpL3 inhibitor that shows highly potent anti-mycobacterial activity with MIC50 of 23 nM against virulent Mycobacterium tuberculosis H37Rv. 了解更多
  42. IACS-8968

    Catalog No. A20020
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    dual IDO/TDO inhibitor
    IACS-8968 (IDO/TDO Inhibitor) is a dual IDO and TDO inhibitor, with pIC50s of 6.43 for IDO and <5 for TDO, respectively. 了解更多
  43. ML-290

    Catalog No. A20008
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    RXFP1 agonist
    ML-290 is a first-in-class and potent relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes, with an EC50 of 94 nM. 了解更多
  44. A 1070722

    Catalog No. A19973
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    GSK-3 inhibitor
    A 1070722 is a potent and selective glycogen synthase kinase 3 (GSK-3) inhibitor, with a Ki of 0.6 nM for both GSK-3α and GSK-3β. 了解更多
  45. UCB9608

    Catalog No. A19941
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    PI4KIIIβ inhibitor
    UCB9608 is a potent, selective and orally active PI4KIIIβ inhibitor, with an IC50 of 11 nM, selective over PI3KC2 α, β, and γ lipid kinases. 了解更多
  46. AZD7594

    Catalog No. A19866
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    glucocorticoid receptor modulator
    AZD7594 is a potent selective nonsteroidal glucocorticoid receptor modulator, with an IC50 of 0.9 nM. 了解更多
  47. MK-4074

    Catalog No. A19854
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    ACC1/ACC2 inhibitor
    MK-4074 is a liver-specific inhibitor of acetyl-CoA carboxylase ACC1 and ACC2 with IC50 values of approximately 3 nM. 了解更多
  48. BET bromodomain inhibitor

    Catalog No. A19831
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    BET inhibitor
    BET bromodomain inhibitor is a potent BET inhibitor extracted from patent WO/2015/153871A2, compound example 11. 了解更多
  49. GCN2iB

    Catalog No. A19806
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    GCN2 inhibitor
    GCN2iB is an ATP-competitive inhibitor of a serine/threonine-protein kinase general control nonderepressible 2 (GCN2), with an IC50 of 2.4 nM. 了解更多
  50. HFI-142

    Catalog No. A19709
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    IRAP inhibitor
    HFI-142 is an insulin-regulated aminopeptidase (IRAP) inhibitor with a Ki of 2.01 μM. 了解更多

产品 51 到 100 共 1231个

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页面:
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  2. 2
  3. 3
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  5. 5

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