“jwh 250”的搜索结果

产品 151 到 200 共 1231个

每页
页面:
  1. 2
  2. 3
  3. 4
  4. 5
  5. 6

设置降序顺序
  1. Centrinone

    Catalog No. A20858
    Quick View
    PLK4 inhibitor
    Centrinone (LCR-263) is a selective and reversible inhibitor of polo-like kinase 4 (PLK4) with a Ki of 0.16 nM. 了解更多
  2. Centrinone-B

    Catalog No. A20855
    Quick View
    PLK4 inhibitor
    Centrinone-B (LCR-323) is a potent and highly selective PLK4 inhibitor, with a Ki of 0.59 nM. 了解更多
  3. Talaporfin sodium

    Catalog No. A18239
    Quick View
    photosensitizer
    Talaporfin (ME2906; NPe6) is a photosensitizer used in photodynamic therapy (PDT). 了解更多
  4. Lesopitron dihydrochloride

    Catalog No. A12950
    Quick View
    5-HT1A receptor agonist
    Lesopitron dihydrochloride is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes. 了解更多
  5. Tyrosine kinase-IN-1

    Catalog No. A12486
    Quick View
    multi-targeted tyrosine kinase inhibitor
    Tyrosine kinase-IN-1 is a multi-targeted tyrosine kinase inhibitor with IC50s of 4, 20, 4, 2 nM for KDR, Flt-1, FGFR1 and PDGFRα, respectively. 了解更多
  6. BACE1-IN-1

    Catalog No. A12183
    Quick View
    BACE1 inhibitor
    BACE1-IN-1 is a potent and highly brain penetrant BACE1 inhibitor with IC50s of 32 and 47 nM for human BACE1 and BACE2, respectively. 了解更多
  7. Pirozadil

    Catalog No. A12501
    Quick View
    Pirozadil is a hypolipidemic agent. 了解更多
  8. TC13172

    Catalog No. A12502
    Quick View
    MLKL inhibitor
    TC13172 is a mixed lineage kinase domain-like protein (MLKL) inhibitor with an EC50 value of 2 nM for HT-29 cells. 了解更多
  9. YM-53601 free base

    Catalog No. A12507
    Quick View
    squalene synthetase inhibitor
    YM-53601 free base is a squalene synthetase inhibitor which suppresses lipogenic biosynthesis and lipid secretion in rodents. 了解更多
  10. MKC3946

    Catalog No. A12508
    Quick View
    IRE1α inhibitor
    MKC3946 is a potent and soluble IRE1α inhibitor, used for cancer research. 了解更多
  11. Famciclovir

    Catalog No. A10380
    Quick View
    Famciclovir(BRL 42810) is a guanine analogue antiviral drug used for the treatment of various herpesvirus infections. 了解更多
  12. Calcitriol D6

    Catalog No. A11376
    Quick View
    Calcitriol D6 is the deuterated form of Calcitriol(1,25-Dihydroxyvitamin D3; Rocaltrol ), which is the hormonally active form of vitamin D, Calcitriol is the active metabolite of vitamin D3 that activates the vitamin D receptor (VDR). 了解更多
  13. NBD-557

    Catalog No. A11509
    Quick View
    HIV-1 inhibitor
    NBD-557 is a potentially HIV-1 inhibitor. 了解更多
  14. DW-1350

    Catalog No. A12250
    Quick View
    LTB4 receptor antagonist
    DW-1350 is a LTB4 receptor antagonist. 了解更多
  15. Y-26763

    Catalog No. A12271
    Quick View
    K+ (KATP) channel activator
    Y-26763 is a K+ channel opener and active metabolite of Y-27152. Y-26763 is an ATP-sensitive K+ (KATP) channel activator. 了解更多
  16. LR-90

    Catalog No. A12296
    Quick View
    AGE inhibitor
    LR-90 is an advanced glycation end product (AGE) inhibitor, inhibits inflammatory responses in human monocytes. LR-90 is also used in the research of diabetic animal model. 了解更多
  17. Bergaptol

    Catalog No. A12303
    Quick View
    CYP3A4 enzyme inhibitor
    Bergaptol is a hydroxylated psoralen that acts as a potent inhibitors of debenzylation activity of CYP3A4 enzyme with an IC50 value of 24.92 uM. Recent studies suggest that it may have antiproliferative and anticancer properties. 了解更多
  18. Pradigastat

    Catalog No. A12475
    Quick View
    DGAT1 inhibitor
    Pradigastat (LCQ-908) is a diacylglycerol acyltransferase 1 (DGAT1) inhibitor. 了解更多
  19. ZINC13466751

    Catalog No. A12522
    Quick View
    HIF-1α/von Hippel-Lindau interaction inhibitor
    ZINC13466751 is a potent inhibitor of HIF-1α/von Hippel-Lindau interaction with an IC50 of 2.0 ?M. 了解更多
  20. Naproxen etemesil

    Catalog No. A13052
    Quick View
    COX-1 and COX-2 inhibitor
    Naproxen etemesil is a lipophilic, non-acidic, inactive prodrug of naproxen that is hydrolysed to pharmacologically active Naproxen once absorbed. Naproxen is a COX-1 and COX-2 inhibitor with IC50s of 8.72 and 5.15 μM, respectively in cell assay. 了解更多
  21. HSL-IN-1

    Catalog No. A13174
    Quick View
    hormone sensitive lipase (HSL) inhibitor
    HSL-IN-1 (compound 24b) is a potent and orally active hormone sensitive lipase (HSL) inhibitor (IC50=2 nM) with a significantly reduced reactive metabolite liability. 了解更多
  22. N2-Methylguanosine

    Catalog No. A13175
    Quick View
    N2-methylguanosine is a modified nucleoside that occurs at several specific locations in many tRNA's. 了解更多
  23. BW 245C

    Catalog No. A13494
    Quick View
    prostanoid DP-receptor (DP1) agonist
    BW 245C is a prostanoid DP-receptor (DP1) agonist, used to treat stroke. 了解更多
  24. PSI-7409

    Catalog No. A13962
    Quick View
    nucleotide analog HCV inhibitor
    PSI-7409 is the active 5'-triphosphate metabolite of Sofosbuvir (PSI-7977). Sofosbuvir (PSI-7977) is a selective and highly active nucleotide analog inhibitor of HCV. 了解更多
  25. FN-1501

    Catalog No. A13559
    Quick View
    FLT3/CDK inhibitor
    FN-1501 is a potent inhibitor of FLT3 and CDK, with IC50s of 2.47, 0.85, 1.96, and 0.28 nM for CDK2/cyclin A, CDK4/cyclin D1, CDK6/cyclin D1 and FLT3, respectively. FN-1501 has anticancer activity. 了解更多
  26. Zamicastat

    Catalog No. A13672
    Quick View
    dopamine β-hydroxylase (DBH) inhibitor
    Zamicastat (BIA 5-1058) is a dopamine β-hydroxylase (DBH) inhibitor that could cross the blood-brain barrier (BBB) and cause central as well as peripheral effects. 了解更多
  27. TES-1025

    Catalog No. A13284
    Quick View
    ACMSD inhibitor
    TES-1025 is a potent and selective human α-amino-β-carboxymuconate-ε-semialdehyde decarboxylase (ACMSD) inhibitor with an IC50 of 13??3 nM. 了解更多
  28. Sipatrigine

    Catalog No. A12943
    Quick View
    neuroprotective agent
    Sipatrigine, a neuroprotective agent, is a glutamate release inhibitor, voltage-dependent sodium channel and calcium channel inhibitor, penetrating the central nervous system. Has potential to treat focal cerebral ischemia and stroke. 了解更多
  29. Antitumor agent-2

    Catalog No. A18430
    Quick View
    Antitumor agent-2 is sourced from patent CN102250203, compound 6a-r, has antitumor action and anti-inflammatory action. 了解更多
  30. I-191

    Catalog No. A18629
    Quick View
    PAR2 antagonist
    I-191 is a potent, selective protease-activated receptor 2 (PAR2) antagonist. 了解更多
  31. Dihydrofolic acid

    Catalog No. A18650
    Quick View
    Dihydrofolic acid is a folic acid derivative acted upon by dihydrofolate reductase to produce tetrahydrofolic acid. 了解更多
  32. BI-671800

    Catalog No. A18902
    Quick View
    CRTH2 antagonist
    BI-671800 is a CRTH2 antagonist that treats patients with asthma. 了解更多
  33. GLP-26

    Catalog No. A18914
    Quick View
    HBV capsid assembly modulator
    GLP-26 is a HBV capsid assembly modulators (CAM), inhibits HBV DNA replication in Hep AD38 system (IC50=3 nM), and reduces cccDNA by >90% at 1 μM. GLP-26 disrupts the encapsidation of pre-genomic RNA, causes nucleocapsid disassembly and reduces cccDNA pools. 了解更多
  34. IDO-IN-12

    Catalog No. A18988
    Quick View
    IDO inhibitor
    IDO-IN-12 is an indoleamine 2,3-dioxygenase (IDO) inhibitor extracted from patent WO 2017181849 A1. 了解更多
  35. Stigmastanol

    Catalog No. A19002
    Quick View
    Stigmastanol is a phytosterol found in a variety of plant sources. 了解更多
  36. Glutarylcarnitine

    Catalog No. A19003
    Quick View
    Glutarylcarnitine is the diagnostic metabolite for malonic aciduria and glutaric aciduria type I monitored in most tandem mass spectrometry newborn screening programmes. 了解更多
  37. Bis-PEG4-acid

    Catalog No. A19036
    Quick View
    PEG PROTAC linker
    Bis-PEG4-acid is a PEG PROTAC linker. 了解更多
  38. SBI-797812

    Catalog No. A19058
    Quick View
    NAMPT activator
    SBI-797812 is a novel NAMPT activator, elevating liver NAD+, turning NAMPT into a "super catalyst" that more efficiently generates NMN. 了解更多
  39. RK-287107

    Catalog No. A19113
    Quick View
    Tankyrase inhibitor
    RK-287107 is a potent and specific tankyrase inhibitor with IC50s of 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively. RK-287107 blocks colorectal cancer cell growth. 了解更多
  40. INH14

    Catalog No. A19119
    Quick View
    IKKα/IKKβ inhibitor
    INH14 is a cell permeable inhibitor of IKKα/IKKβ, with IC50s of 8.97 and 3.59 μM, respectively. 了解更多
  41. MSDC-0602

    Catalog No. A19368
    Quick View
    MPC inhibitor
    MSDC-0602, a PPARγ-sparing thiazolidinedione (TZD), interacts with the mitochondrial pyruvate carrier (MPC) and inhibits its activity and are effective for treatment of type 2 diabetes with reducing risk of PPARγ-mediated side effects. 了解更多
  42. GSK2982772

    Catalog No. A19380
    Quick View
    RIP1 kinase inhibitor
    GSK2982772 is a potent, orally active and ATP competitive RIP1 kinase inhibitor with IC50 values of 16 nM and 20 nM for human and monkey RIP1, respectively. 了解更多
  43. GSK5182

    Catalog No. A19383
    Quick View
    ERRγ agonist
    GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα. 了解更多
  44. Acrizanib

    Catalog No. A19384
    Quick View
    VEGFR-2 抑制剂
    Acrizanib is a VEGFR-2 inhibitor, with an IC50 of 17.4 nM for BaF3-KDR. 了解更多
  45. LHF-535

    Catalog No. A19405
    Quick View
    LHF-535 is an antiviral agent extracted from patent WO2013123215A2, Compound 38, has EC50s of <1 μM, <1 μM, <1 μM, and 1-10 μM for Lassa, Machupo, Junin, and VSVg virus, respectively. 了解更多
  46. AS-35

    Catalog No. A19409
    Quick View
    LTR antagonist
    AS-35 is an orally effective, potent and selective antagonist of leukotrienes, antagonizes LTC4-, LTD4 and LTE4-induced contractions of the ileum with IC50 values of 8 nM, 4 nM and 3 nM, respectively, and has antiallergic activities. 了解更多
  47. MS417

    Catalog No. A19433
    Quick View
    BRD4 inhibitor
    MS417 is a BET-specific BRD4 inhibitor, binds to BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively, with weak selectivity at CBP BRD (IC50, 32.7 μM). 了解更多
  48. LUT014

    Catalog No. A19449
    Quick View
    B-Raf inhibitor
    LUT014 is a B-Raf inhibitor with an IC50 of 11.7 nM, and developed to reduce dose-limiting acneiform lesions associated EGFR Inhibitors treatment. Extracted from patent WO 2019026065A2 . 了解更多
  49. PF-06751979

    Catalog No. A20066
    Quick View
    BACE1 inhibitor
    PF-06751979 is a potent, brain penetrant, β-site amyloid precursor protein cleaving enzyme 1 (BACE1) inhibitor with an IC50 of 7.3 nM in BACE1 binding assay. 了解更多
  50. DMX-5804

    Catalog No. A20199
    Quick View
    MAP4K4 inhibitor
    DMX-5804 is a potent, orally active and selective MAP4K4 inhibitor, with an IC50 of 3 nM, a pIC50 of 8.55 for human MAP4K4, less potent on MINK1/MAP4K6 (pIC50, 8.18), and TNIK/MAP4K7 (pIC50, 7.96). 了解更多

产品 151 到 200 共 1231个

每页
页面:
  1. 2
  2. 3
  3. 4
  4. 5
  5. 6

设置降序顺序
Rewards