Sildenafil citrate-d8
Catalog No. A31741
Sildenafil citrate-d8 is a deuterium-labeled derivative of Sildenafil citrate, a potent inhibitor of phosphodiesterase type 5 (PDE5) with an IC50 of 5.22 nM. This stable isotope reagent is primarily used for metabolic studies and pharmacokinetic research, facilitating the tracing of drug metabolism and pharmacological profiling in biological systems. Its unique labeling allows for enhanced detection and analysis in various experimental formats.
Chemical Information
| Catalog Num | A31741 |
|---|---|
| M. Wt | 674.75 |
| Formula | C28H30D8N6O11S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1215071-03-6 |
| Synonyms | UK-92480 citrate-d8 |
| SMILES | OC(CC(C(O)=O)(O)CC(O)=O)=O.CCOC1=C(C(NC2=C3N(N=C2CCC)C)=NC3=O)C=C(C=C1)S(=O)(N4C([2H])([2H])C([2H])([2H])N(C([2H])([2H])C4([2H])[2H])C)=O |
| Storage |
Biological Activity
| Discription | Sildenafil citrate-d8 is a deuterium-labeled derivative of Sildenafil citrate, a potent inhibitor of phosphodiesterase type 5 (PDE5) with an IC50 of 5.22 nM. This stable isotope reagent is primarily used for metabolic studies and pharmacokinetic research, facilitating the tracing of drug metabolism and pharmacological profiling in biological systems. Its unique labeling allows for enhanced detection and analysis in various experimental formats. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
