Brompheniramine
Catalog No. A33899
Brompheniramine is a selective histamine H1 receptor antagonist primarily utilized as an antihistamine agent. With a Kd of 6.06 nM, it effectively alleviates symptoms of allergic rhinitis. In addition to its antihistaminic properties, brompheniramine exhibits anticholinergic, antidepressant, and anesthetic effects, making it suitable for various research applications related to allergy and inflammation. The compound also interacts with hERG, calcium, and sodium channels, with IC50 values of 0.90 μM, 16.12 μM, and 21.26 μM, respectively.
Chemical Information
| Catalog Num | A33899 |
|---|---|
| M. Wt | 319.24 |
| Formula | C16H19BrN2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 86-22-6 |
| Synonyms | (±)-Brompheniramine |
| SMILES | CN(C)CCC(C1=CC=C(Br)C=C1)C2=CC=CC=N2 |
| Storage |
Biological Activity
| Discription | Brompheniramine is a selective histamine H1 receptor antagonist primarily utilized as an antihistamine agent. With a Kd of 6.06 nM, it effectively alleviates symptoms of allergic rhinitis. In addition to its antihistaminic properties, brompheniramine exhibits anticholinergic, antidepressant, and anesthetic effects, making it suitable for various research applications related to allergy and inflammation. The compound also interacts with hERG, calcium, and sodium channels, with IC50 values of 0.90 μM, 16.12 μM, and 21.26 μM, respectively. |
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Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
