Product Data Sheet
CBP-IN-1
Catalog No. A40387
CBP-IN-1 is a potent inhibitor of the CREB-binding protein (CBP) with an IC50 of 1.5 nM. Additionally, it inhibits CBP BRET and BRD4(1), demonstrating IC50 values of 690 nM and 3100 nM, respectively. CBP-IN-1 is valuable for research applications focused on transcriptional regulation and related signal transduction pathways. Its selective inhibitory profile makes it a useful tool in the study of diseases associated with CBP dysregulation.
Chemical Information
| Catalog Num | A40387 |
|---|---|
| M. Wt | 509.59 |
| Formula | C27H33F2N7O |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1936431-44-5 |
| Synonyms | |
| SMILES | O=C(C)N1CC2=C(CC1)N(C3CCNCC3)N=C2N4C5=C(CCC4)C=C(C6=CN(C)N=C6)C(C(F)F)=C5 |
| Storage |
Biological Activity
| Discription | CBP-IN-1 is a potent inhibitor of the CREB-binding protein (CBP) with an IC50 of 1.5 nM. Additionally, it inhibits CBP BRET and BRD4(1), demonstrating IC50 values of 690 nM and 3100 nM, respectively. CBP-IN-1 is valuable for research applications focused on transcriptional regulation and related signal transduction pathways. Its selective inhibitory profile makes it a useful tool in the study of diseases associated with CBP dysregulation. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
