ASP3026
Catalog No. A11773
ASP3026是ALK激酶的新型选择性抑制剂。ASP3026在Tyr激酶组中有效抑制ALK激酶活性,并且比克唑替尼更具选择性。
Catalog Num | A11773 |
---|---|
M. Wt | 580.7 |
Formula | C29H40N8O3S |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1097917-15-1 |
Synonyms | ASP 3026, ASP-3026 |
SMILES | CC(C)S(=O)(=O)C1=CC=CC=C1NC2=NC=NC(=N2)NC3=C(C=C(C=C3)N4CCC(CC4)N5CCN(CC5)C)OC |
ASP3026是ALK激酶的新型选择性抑制剂。ASP3026在Tyr激酶组中有效抑制ALK激酶活性,并且比克唑替尼更具选择性。
Targets
ALK | ||||
3.5 nM |
In vitro | DMSO | 13 mg/mL (22.38 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 17.22 mL | 86.1 mL | 172.21 mL |
0.5 mM | 3.44 mL | 17.22 mL | 34.44 mL |
1 mM | 1.72 mL | 8.61 mL | 17.22 mL |
5 mM | 0.34 mL | 1.72 mL | 3.44 mL |
*The above data is based on the productmolecular weight 580.7 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.