Rupatadine Fumarate

Catalog No. A12356

Rupatadine Fumarate是PAFR和组胺(H1)受体的抑制剂,Ki分别为550和102 nM。
Catalog Num A12356
M. Wt 532.03
Formula C26H26ClN3.C4H4O4
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 182349-12-8
Synonyms
SMILES CC1=CC(=CN=C1)CN2CCC(=C3C4=C(CCC5=C3N=CC=C5)C=C(C=C4)Cl)CC2.C(=C/C(=O)O)\C(=O)O
Rupatadine Fumarate是PAFR和组胺(H1)受体的抑制剂,Ki分别为550和102 nM。
Targets
Histamine H1 receptor PAFR
102 nM(Ki)550 nM(Ki)
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.8 mL 93.98 mL 187.96 mL
0.5 mM 3.76 mL 18.8 mL 37.59 mL
1 mM 1.88 mL 9.4 mL 18.8 mL
5 mM 0.38 mL 1.88 mL 3.76 mL

*The above data is based on the productmolecular weight 532.03. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.